Design and Synthesis of Androgen Receptor Full Antagonists Bearing a p-Carborane Cage: Promising Ligands for Anti-Androgen Withdrawal Syndrome von Goto, Tokuhito, Ohta, Kiminori, Fujii, Shinya, Ohta, Shigeru, Endo, Yasuyuki

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Facile and Efficient Synthesis of C-Hydroxycarboranes and C,C‘-Dihydroxycarboranes von Ohta, Kiminori, Goto, Tokuhito, Yamazaki, Hiroto, Pichierri, Fabio, Endo, Yasuyuki

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Crystal structure, docking study and structure–activity relationship of carborane-containing androgen receptor antagonist 3-(12-hydroxymethyl-1,12-dicarba- closo-dodecaboran-1-yl)b... von Ohta, Kiminori, Goto, Tokuhito, Fujii, Shinya, Kawahata, Masatoshi, Oda, Akifumi, Ohta, Shigeru, Yamaguchi, Kentaro, Hirono, Shuichi, Endo, Yasuyuki

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Design and synthesis of carborane-containing androgen receptor (AR) antagonist bearing a pyridine ring von Ohta, Kiminori, Goto, Tokuhito, Fijii, Shinya, Suzuki, Tomoharu, Ohta, Shigeru, Endo, Yasuyuki

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Development of androgen receptor ligands by application of ten-vertex para-carborane as a novel hydrophobic core structure von Fujii, Shinya, Ohta, Kiminori, Goto, Tokuhito, Oda, Akifumi, Masuno, Hiroyuki, Endo, Yasuyuki, Kagechika, Hiroyuki

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New synthetic method of 1,2-diaryl-1,2-dicarba- closo-dodecaboranes employing aromatic nucleophilic substitution (S NAr) reaction von Ohta, Kiminori, Goto, Tokuhito, Endo, Yasuyuki

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Novel androgen receptor full antagonists: Design, synthesis, and a docking study of glycerol and aminoglycerol derivatives that contain p-carborane cages von Kaise, Asako, Ohta, Kiminori, Fujii, Shinya, Oda, Akifumi, Goto, Tokuhito, Endo, Yasuyuki

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1,2-Dicarba-closo-dodecaboran-1-yl Naphthalene Derivatives von OHTA, Kiminori, GOTO, Tokuhito, ENDO, Yasuyuki

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A series of novel indazole derivatives of Sirt 1 activator as osteogenic regulators von Atobe, Masakazu, Yamakawa, Natsumi, Wada, Yasuhiro, Goto, Tokuhito, Kawanishi, Masashi, Ito, Takeshi, Saito, Makoto, Takeda, Masahiro, Tabata, Takanori, Arai, Hirokazu

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Acidic heterocycles as novel hydrophilic pharmacophore of androgen receptor ligands with a carborane core structure von Fujii, Shinya, Ohta, Kiminori, Goto, Tokuhito, Kagechika, Hiroyuki, Endo, Yasuyuki

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Potent Androgen Antagonists Based on Carborane as a Hydrophobic Core Structure von Fujii, Shinya, Goto, Tokuhito, Ohta, Kiminori, Hashimoto, Yuichi, Suzuki, Tomoharu, Ohta, Shigeru, Endo, Yasuyuki

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1,2-Dicarba-closo-dodecaboran-1-yl naphthalene derivatives von Ohta, Kiminori, Goto, Tokuhito, Endo, Yasuyuki

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Design and synthesis of novel androgen receptor antagonists with sterically bulky icosahedral carboranes von Goto, Tokuhito, Ohta, Kiminori, Suzuki, Tomoharu, Ohta, Shigeru, Endo, Yasuyuki

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p-Carborane-based androgen antagonists active in LNCaP cells with a mutated androgen receptor von Fujii, Shinya, Yamada, Ayumi, Tomita, Keiko, Nagano, Mao, Goto, Tokuhito, Ohta, Kiminori, Harayama, Takashi, Endo, Yasuyuki, Kagechika, Hiroyuki

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Crystal structure, docking study and structure-activity relationship of carborane-containing androgen receptor antagonist 3-(12-hydroxymethyl-1,12-dicarba-closo-dodecaboran-1-yl)be... von Ohta, Kiminori, Goto, Tokuhito, Fujii, Shinya, Kawahata, Masatoshi, Oda, Akifumi, Ohta, Shigeru, Yamaguchi, Kentaro, Hirono, Shuichi, Endo, Yasuyuki

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1,2-Dicarba-c loso-dodecaboran-1-yl Naphthalene Derivatives von Ohta, Kiminori, Goto, Tokuhito, Endo, Yasuyuki

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Development of androgen receptor ligands by application of ten-vertex para-carborane as a novel hydrophobic core structureElectronic supplementary information (ESI) available. See... von Fujii, Shinya, Ohta, Kiminori, Goto, Tokuhito, Oda, Akifumi, Masuno, Hiroyuki, Endo, Yasuyuki, Kagechika, Hiroyuki

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Phase 2 study of axicabtagene ciloleucel in Japanese patients with relapsed or refractory large B-cell lymphoma von Kato, Koji, Makita, Shinichi, Goto, Hideki, Kanda, Junya, Fujii, Nobuharu, Shimada, Kazuyuki, Akashi, Koichi, Izutsu, Koji, Teshima, Takanori, Fukuda, Natsuko, Sumitani, Tokuhito, Sumi, Hiroyuki, Shimizu, Shinji, Kakurai, Yasuyuki, Yoshikawa, Kenji, Tobinai, Kensei, Usui, Noriko, Hatake, Kiyohiko

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A phase 2 study of axicabtagene ciloleucel in relapsed or refractory large B-cell lymphoma in Japan: 1-year follow-up and biomarker analysis von Kato, Koji, Fujii, Nobuharu, Makita, Shinichi, Goto, Hideki, Kanda, Junya, Shimada, Kazuyuki, Akashi, Koichi, Izutsu, Koji, Teshima, Takanori, Fukuda, Natsuko, Sumitani, Tokuhito, Nakamura, Shota, Sumi, Hiroyuki, Shimizu, Shinji, Kakurai, Yasuyuki, Yoshikawa, Kenji, Tobinai, Kensei, Usui, Noriko, Hatake, Kiyohiko

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Microbolometer Terahertz Focal Plane Array and Camera with Improved Sensitivity in the Sub-Terahertz Region von Oda, Naoki, Kurashina, Seiji, Miyoshi, Masaru, Doi, Kohei, Ishi, Tsutomu, Sudou, Takayuki, Morimoto, Takao, Goto, Hideki, Sasaki, Tokuhito

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