In Vitro and In Vivo Activity of Cabozantinib (XL184), an Inhibitor of RET, MET, and VEGFR2, in a Model of Medullary Thyroid Cancer von Bentzien, Frauke, Zuzow, Marcus, Heald, Nathan, Gibson, Anna, Shi, Yongchang, Goon, Leanne, Yu, Peiwen, Engst, Stefan, Zhang, Wentao, Huang, Donghui, Zhao, Lora, Vysotskaia, Valentina, Chu, Felix, Bautista, Rajana, Cancilla, Belinda, Lamb, Peter, Joly, Alison H., Yakes, F. Michael

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High-content, high-throughput analysis of cell cycle perturbations induced by the HSP90 inhibitor XL888 von Lyman, Susan K, Crawley, Suzanne C, Gong, Ruoyu, Adamkewicz, Joanne I, McGrath, Garth, Chew, Jason Y, Choi, Jennifer, Holst, Charles R, Goon, Leanne H, Detmer, Scott A, Vaclavikova, Jana, Gerritsen, Mary E, Blake, Robert A

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Implementation of the CYP Index for the Design of Selective Tryptophan-2,3-dioxygenase Inhibitors von Parr, Brendan T, Pastor, Richard, Sellers, Benjamin D, Pei, Zhonghua, Jaipuri, Firoz A, Castanedo, Georgette M, Gazzard, Lewis, Kumar, Sanjeev, Li, Xiaokai, Liu, Wen, Mendonca, Rohan, Pavana, Roheeth K, Potturi, Hima, Shao, Cheng, Velvadapu, Venkata, Waldo, Jesse P, Wu, Guosheng, Yuen, Po-wai, Zhang, Zuhui, Zhang, Yamin, Harris, Seth F, Oh, Angela J, DiPasquale, Antonio, Dement, Kevin, La, Hank, Goon, Leanne, Gustafson, Amy, VanderPorten, Erica C, Mautino, Mario R, Liu, Yichin

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Correction: High-Content, High-Throughput Analysis of Cell Cycle Perturbations Induced by the HSP90 Inhibitor XL888 von Lyman, Susan K., Crawley, Suzanne C., Gong, Ruoyu, Adamkewicz, Joanne I., McGrath, Garth, Chew, Jason Y., Choi, Jennifer, Holst, Charles R., Goon, Leanne H., Detmer, Scott A., Vaclavikova, Jana, Gerritsen, Mary E., Blake, Robert A.

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Aminoisoxazoles as Potent Inhibitors of Tryptophan 2,3-Dioxygenase 2 (TDO2) von Pei, Zhonghua, Mendonca, Rohan, Gazzard, Lewis, Pastor, Richard, Goon, Leanne, Gustafson, Amy, VanderPorten, Erica, Hatzivassiliou, Georgia, Dement, Kevin, Cass, Robert, Yuen, Po-wai, Zhang, Yamin, Wu, Guosheng, Lin, Xingyu, Liu, Yichin, Sellers, Benjamin D

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Antibody–Drug Conjugates Derived from Cytotoxic seco-CBI-Dimer Payloads Are Highly Efficacious in Xenograft Models and Form Protein Adducts In Vivo von Su, Dian, Chen, Jinhua, Cosino, Ely, dela Cruz-Chuh, Josefa, Davis, Helen, Del Rosario, Geoffrey, Figueroa, Isabel, Goon, Leanne, He, Jintang, Kamath, Amrita V, Kaur, Surinder, Kozak, Katherine R, Lau, Jeffrey, Lee, Donna, Lee, M. Violet, Leipold, Douglas, Liu, Luna, Liu, Peter, Lu, Guo-Liang, Nelson, Chris, Ng, Carl, Pillow, Thomas H, Polakis, Paul, Polson, Andrew G, Rowntree, Rebecca K, Saad, Ola, Safina, Brian, Stagg, Nicola J, Tercel, Moana, Vandlen, Richard, Vollmar, Breanna S, Wai, John, Wang, Tao, Wei, BinQing, Xu, Keyang, Xue, Juanjuan, Xu, Zijin, Yan, Gang, Yao, Hui, Yu, Shang-Fan, Zhang, Donglu, Zhong, Fiona, Dragovich, Peter S

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Discovery of a Novel Series of Potent and Orally Bioavailable Phosphoinositide 3-Kinase γ Inhibitors von Leahy, James W, Buhr, Chris A, Johnson, Henry W. B, Kim, Byung Gyu, Baik, TaeGon, Cannoy, Jonah, Forsyth, Timothy P, Jeong, Joon Won, Lee, Matthew S, Ma, Sunghoon, Noson, Kevin, Wang, Longcheng, Williams, Matthew, Nuss, John M, Brooks, Eric, Foster, Paul, Goon, Leanne, Heald, Nathan, Holst, Charles, Jaeger, Christopher, Lam, Scott, Lougheed, Julie, Nguyen, Lam, Plonowski, Arthur, Song, Joanne, Stout, Thomas, Wu, Xiang, Yakes, Michael F, Yu, Peiwen, Zhang, Wentao, Lamb, Peter, Raeber, Olivia

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Lysosomal Ca(2+) stores in bovine corneal endothelium von Srinivas, Sangly P, Ong, Angeline, Goon, Leanne, Goon, Levina, Bonanno, Joseph A

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Lysosomal Ca2+ Stores in Bovine Corneal Endothelium von Srinivas, Sangly P, Ong, Angeline, Goon, Leanne, Goon, Levina, Bonanno, Joseph A

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