Challenging the Drug-Likeness Dogma for New Drug Discovery in Tuberculosis von Machado, Diana, Girardini, Miriam, Viveiros, Miguel, Pieroni, Marco

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Preliminary structure−activity relationships analysis on N-(3,5-dichlorophenyl)-4,5-dihydronaphtho[1,2-d]thiazol-2-amine, a disruptor of mycobacterial energetics von Girardini, Miriam, Machado, Diana, Annunziato, Giannamaria, Papotti, Bianca, Palumbo, Marcella, Spaggiari, Chiara, Costantino, Gabriele, Viveiros, Miguel, Pieroni, Marco

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Cereblon versus VHL: Hijacking E3 ligases against each other using PROTACs von Girardini, Miriam, Maniaci, Chiara, Hughes, Scott J., Testa, Andrea, Ciulli, Alessio

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2‑Aminooxazole as a Novel Privileged Scaffold in Antitubercular Medicinal Chemistry von Azzali, Elisa, Girardini, Miriam, Annunziato, Giannamaria, Pavone, Marialaura, Vacondio, Federica, Mori, Giorgia, Pasca, Maria Rosalia, Costantino, Gabriele, Pieroni, Marco

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Expanding the knowledge around antitubercular 5-(2-aminothiazol-4-yl)isoxazole-3-carboxamides: Hit–to–lead optimization and release of a novel antitubercular chemotype via scaffold... von Girardini, Miriam, Ferlenghi, Francesca, Annunziato, Giannamaria, Degiacomi, Giulia, Papotti, Bianca, Marchi, Cinzia, Sammartino, José Camilla, Rasheed, Sari S., Contini, Anna, Pasca, Maria Rosalia, Vacondio, Federica, Evans, Joanna C., Dick, Thomas, Müller, Rolf, Costantino, Gabriele, Pieroni, Marco

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