Localization of histamine H4 receptors in the central nervous system of human and rat von Strakhova, Marina I, Nikkel, Arthur L, Manelli, Arlene M, Hsieh, Gin C, Esbenshade, Timothy A, Brioni, Jorge D, Bitner, Robert S

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Pharmacological modulation of movement-evoked pain in a rat model of osteoarthritis von Chandran, Prasant, Pai, Madhavi, Blomme, Eric A., Hsieh, Gin C., Decker, Michael W., Honore, Prisca

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Indol-3-ylcycloalkyl Ketones: Effects of N1 Substituted Indole Side Chain Variations on CB2 Cannabinoid Receptor Activity von Frost, Jennifer M, Dart, Michael J, Tietje, Karin R, Garrison, Tiffany R, Grayson, George K, Daza, Anthony V, El-Kouhen, Odile F, Yao, Betty B, Hsieh, Gin C, Pai, Madhavi, Zhu, Chang Z, Chandran, Prasant, Meyer, Michael D

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Central and peripheral sites of action for CB2 receptor mediated analgesic activity in chronic inflammatory and neuropathic pain models in rats von Hsieh, Gin C, Pai, Madhavi, Chandran, Prasant, Hooker, Bradley A, Zhu, Chang Z, Salyers, Anita K, Wensink, Erica J, Zhan, CenChen, Carroll, William A, Dart, Michael J, Yao, Betty B, Honore, Prisca, Meyer, Michael D

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Activation of Dopamine D4 Receptors by ABT-724 Induces Penile Erection in Rats von Brioni, Jorge D., Moreland, Robert B., Cowart, Marlon, Hsieh, Gin C., Stewart, Andrew O., Hedlund, Petter, Donnelly-Roberts, Diana L., Nakane, Masaki, Lynch, James J., Kolasa, Teodozyi, Polakowski, James S., Osinski, Mark A., Marsh, Kennan, Andersson, Karl-Erik, Sullivan, James P., Beavo, Joseph A.

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Central and peripheral sites of action for CB 2 receptor mediated analgesic activity in chronic inflammatory and neuropathic pain models in rats von Hsieh, Gin C, Pai, Madhavi, Chandran, Prasant, Hooker, Bradley A, Zhu, Chang Z, Salyers, Anita K, Wensink, Erica J, Zhan, CenChen, Carroll, William A, Dart, Michael J, Yao, Betty B, Honore, Prisca, Meyer, Michael D

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A-412997 is a selective dopamine D4 receptor agonist in rats von MORELAND, Robert B, PATEL, Meena, HSIEH, Gin C, WETTER, Jill M, MARSH, Kennan, BRIONI, Jorge D

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Substituted Indazoles as Nav1.7 Blockers for the Treatment of Pain von Frost, Jennifer M, DeGoey, David A, Shi, Lei, Gum, Rebecca J, Fricano, Meagan M, Lundgaard, Greta L, El-Kouhen, Odile F, Hsieh, Gin C, Neelands, Torben, Matulenko, Mark A, Daanen, Jerome F, Pai, Madhavi, Ghoreishi-Haack, Nayereh, Zhan, Cenchen, Zhang, Xu-Feng, Kort, Michael E

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Effects of selective dopamine receptor subtype agonists on cardiac contractility and regional haemodynamics in rats von Polakowski, James S, Segreti, Jason A, Cox, Bryan F, Hsieh, Gin C, Kolasa, Teodozyj, Moreland, Robert B, Brioni, Jorge D

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YC-1 potentiates the nitric oxide/cyclic GMP pathway in corpus cavernosum and facilitates penile erection in rats von Hsieh, Gin C, O'Neill, Alyssa B, Moreland, Robert B, Sullivan, James P, Brioni, Jorge D

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H4 receptor antagonism exhibits anti-nociceptive effects in inflammatory and neuropathic pain models in rats von HSIEH, Gin C, CHANDRAN, Prasant, WETTER, Jill M, MARSH, Kennan C, HANCOCK, Arthur A, COWART, Marlon D, ESBENSHADE, Timothy A, BRIONI, Jorge D, HONORE, Prisca, SALYERS, Anita K, PAI, Madhavi, ZHU, Chang Z, WENSINK, Erica J, WITTE, David G, MILLER, Thomas R, MIKUSA, Joe P, BAKER, Scott J

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Rotationally Constrained 2,4-Diamino-5,6-disubstituted Pyrimidines: A New Class of Histamine H4 Receptor Antagonists with Improved Druglikeness and in Vivo Efficacy in Pain and Inf... von Cowart, Marlon D, Altenbach, Robert J, Liu, Huaqing, Hsieh, Gin C, Drizin, Irene, Milicic, Ivan, Miller, Thomas R, Witte, David G, Wishart, Neil, Fix-Stenzel, Shannon R, McPherson, Michael J, Adair, Ronald M, Wetter, Jill M, Bettencourt, Brian M, Marsh, Kennan C, Sullivan, James P, Honore, Prisca, Esbenshade, Timothy A, Brioni, Jorge D

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Discovery and biological evaluation of novel cyanoguanidine P2X(7) antagonists with analgesic activity in a rat model of neuropathic pain von Perez-Medrano, Arturo, Donnelly-Roberts, Diana L, Honore, Prisca, Hsieh, Gin C, Namovic, Marian T, Peddi, Sridhar, Shuai, Qi, Wang, Ying, Faltynek, Connie R, Jarvis, Michael F, Carroll, William A

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Indol-3-yl-tetramethylcyclopropyl Ketones: Effects of Indole Ring Substitution on CB2 Cannabinoid Receptor Activity von Frost, Jennifer M, Dart, Michael J, Tietje, Karin R, Garrison, Tiffany R, Grayson, George K, Daza, Anthony V, El-Kouhen, Odile F, Miller, Loan N, Li, Lanlan, Yao, Betty B, Hsieh, Gin C, Pai, Madhavi, Zhu, Chang Z, Chandran, Prasant, Meyer, Michael D

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Structure−Activity Studies on a Series of a 2-Aminopyrimidine-Containing Histamine H4 Receptor Ligands von Altenbach, Robert J, Adair, Ronald M, Bettencourt, Brian M, Black, Lawrence A, Fix-Stenzel, Shannon R, Gopalakrishnan, Sujatha M, Hsieh, Gin C, Liu, Huaqing, Marsh, Kennan C, McPherson, Michael J, Milicic, Ivan, Miller, Thomas R, Vortherms, Timothy A, Warrior, Usha, Wetter, Jill M, Wishart, Neil, Witte, David G, Honore, Prisca, Esbenshade, Timothy A, Hancock, Arthur A, Brioni, Jorge D, Cowart, Marlon D

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Discovery and Biological Evaluation of Novel Cyanoguanidine P2X7 Antagonists with Analgesic Activity in a Rat Model of Neuropathic Pain von Perez-Medrano, Arturo, Donnelly-Roberts, Diana L, Honore, Prisca, Hsieh, Gin C, Namovic, Marian T, Peddi, Sridhar, Shuai, Qi, Wang, Ying, Faltynek, Connie R, Jarvis, Michael F, Carroll, William A

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Antinociceptive effects of histamine H3 receptor antagonist in the preclinical models of pain in rats and the involvement of central noradrenergic systems von Hsieh, Gin C, Honore, Prisca, Pai, Madhavi, Wensink, Erica J, Chandran, Prasant, Salyers, Anita K, Wetter, Jill M, Zhao, Chen, Liu, Huaqing, Decker, Michael W, Esbenshade, Timothy A, Cowart, Marlon D, Brioni, Jorge D

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cis-4-(Piperazin-1-yl)-5,6,7a,8,9,10,11,11a-octahydrobenzofuro[2,3-h]quinazolin-2-amine (A-987306), A New Histamine H4R Antagonist that Blocks Pain Responses against Carrageenan-In... von Liu, Huaqing, Altenbach, Robert J, Carr, Tracy L, Chandran, Prasant, Hsieh, Gin C, Lewis, La Geisha R, Manelli, Arlene M, Milicic, Ivan, Marsh, Kennan C, Miller, Thomas R, Strakhova, Marina I, Vortherms, Timothy A, Wakefield, Brian D, Wetter, Jill M, Witte, David G, Honore, Prisca, Esbenshade, Timothy A, Brioni, Jorge D, Cowart, Marlon D

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Synthesis and evaluation of 2-amido-3-carboxamide thiophene CB2 receptor agonists for pain management von Nelson, Derek W., Frost, Jennifer M., Tietje, Karin R., Florjancic, Alan S., Ryther, Keith, Carroll, William A., Dart, Michael J., Daza, Anthony V., Hooker, Bradley A., Grayson, George K., Fan, Yihong, Garrison, Tiffany R., El-Kouhen, Odile F., Yao, Betty, Pai, Madhavi, Chandran, Prasant, Zhu, Chang, Hsieh, Gin C., Meyer, Michael D.

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Diaryldiamines with Dual Inhibition of the Histamine H3 Receptor and the Norepinephrine Transporter and the Efficacy of 4-(3-(Methylamino)-1-phenylpropyl)-6-(2-(pyrrolidin-1-yl)eth... von Altenbach, Robert J, Black, Lawrence A, Strakhova, Marina I, Manelli, Arlene M, Carr, Tracy L, Marsh, Kennan C, Wetter, Jill M, Wensink, Erica J, Hsieh, Gin C, Honore, Prisca, Garrison, Tiffany Runyan, Brioni, Jorge D, Cowart, Marlon D

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