The evolution of amidine-based brain penetrant BACE1 inhibitors von Oehlrich, Daniel, Prokopcova, Hana, Gijsen, Harrie J.M.

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3,3-Difluoro-3,4,5,6-tetrahydropyridin-2-amines: Potent and permeable BACE-1 inhibitors von Peschiulli, Aldo, Oehlrich, Daniel, Rombouts, Frederik, Vos, Ann, Gijsen, Harrie JM

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Tricyclic 3,4-dihydropyrimidine-2-thione derivatives as potent TRPA1 antagonists von Gijsen, Harrie J.M., Berthelot, Didier, De Cleyn, Michel A.J., Geuens, Ivo, Brône, Bert, Mercken, Marc

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5-Sulfonyl-benzimidazoles as selective CB2 agonists-Part 2 von Gijsen, Harrie J.M., De Cleyn, Michel A.J., Surkyn, Michel, Van Lommen, Guy R.E., Verbist, Bie M.P., Nijsen, Marjoleen J.M.A., Meert, Theo, Wauwe, Jean Van, Aerssens, Jeroen

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5-Sulfonyl-benzimidazoles as selective CB2 agonists von Verbist, Bie M.P., De Cleyn, Michel A.J., Surkyn, Michel, Fraiponts, Erwin, Aerssens, Jeroen, Nijsen, Marjoleen J.M.A., Gijsen, Harrie J.M.

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Discovery of brain permeable 2-Azabicyclo[2.2.2]octane sulfonamides as a novel class of presenilin-1 selective γ-secretase inhibitors von Narlawar, Rajeshwar, Serneels, Lutgarde, Gaffric, Celia, Gijsen, Harrie JM, De Strooper, Bart, Bischoff, François

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Selective inhibitors of the PSEN1–gamma-secretase complex von Serneels, Lutgarde, Narlawar, Rajeshwar, Perez-Benito, Laura, Municoy, Marti, Guallar, Victor, T'Syen, Dries, Dewilde, Maarten, Bischoff, François, Fraiponts, Erwin, Tresadern, Gary, Roevens, Peter WM, Gijsen, Harrie JM, De Strooper, Bart

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