Discovery of 4-Amino-5-(3-bromophenyl)-7-(6-morpholino-pyridin- 3-yl)pyrido[2,3-d]pyrimidine, an Orally Active, Non-Nucleoside Adenosine Kinase Inhibitor von Lee, Chih-Hung, Jiang, Meiqun, Cowart, Marlon, Gfesser, Greg, Perner, Richard, Kim, Ki Hwan, Gu, Yu Gui, Williams, Michael, Jarvis, Michael F, Kowaluk, Elizabeth A, Stewart, Andrew O, Bhagwat, Shripad S

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Fluorescent benzofuran histamine H3 receptor antagonists with sub-nanomolar potency von Cowart, M., Gfesser, G. A., Bhatia, K., Esser, R., Sun, M., Miller, T. R., Krueger, K., Witte, D., Esbenshade, T. A., Hancock, A. A.

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Achievement of behavioral efficacy and improved potency in new heterocyclic analogs of benzofuran H3 antagonists von Cowart, M, Faghih, R, Gfesser, G, Curtis, M, Sun, M, Zhao, C, Bennani, Y, Wetter, J, Marsh, K, Miller, T R, Krueger, K, Pan, J B, Drescher, K, Fox, G B, Esbenshade, T A, Hancock, A A

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Synthesis and Pharmacology of (Pyridin-2-yl)methanol Derivatives as Novel and Selective Transient Receptor Potential Vanilloid 3 Antagonists von Gomtsyan, Arthur, Schmidt, Robert G, Bayburt, Erol K, Gfesser, Gregory A, Voight, Eric A, Daanen, Jerome F, Schmidt, Diana L, Cowart, Marlon D, Liu, Huaqing, Altenbach, Robert J, Kort, Michael E, Clapham, Bruce, Cox, Phil B, Shrestha, Anurupa, Henry, Rodger, Whittern, David N, Reilly, Regina M, Puttfarcken, Pamela S, Brederson, Jill-Desiree, Song, Ping, Li, Bin, Huang, Susan M, McDonald, Heath A, Neelands, Torben R, McGaraughty, Steve P, Gauvin, Donna M, Joshi, Shailen K, Banfor, Patricia N, Segreti, Jason A, Shebley, Mohamad, Faltynek, Connie R, Dart, Michael J, Kym, Philip R

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Structure–activity studies of 5-substituted pyridopyrimidines as adenosine kinase inhibitors von Cowart, Marlon, Lee, Chih-Hung, Gfesser, Gregory A., Bayburt, Erol K., Bhagwat, Shripad S., Stewart, Andrew O., Yu, Haixia, Kohlhaas, Kathy L., McGaraughty, Steve, Wismer, Carol T., Mikusa, Joseph, Zhu, Chang, Alexander, Karen M., Jarvis, Michael F., Kowaluk, Elizabeth A.

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The medicinal chemistry of novel H 3 antagonists von Cowart, M., Faghih, R., Gfesser, G., Curtis, M., Pratt, J. K., Bennani, Y., Fox, G. B., Esbenshade, T. A., Hancock, A. A.

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Novel heterocyclic-substituted benzofuran histamine H3 receptor antagonists: in vitro properties, drug-likeness, and behavioral activity von Cowart, Marlon, Gfesser, Gregory A, Browman, Kaitlin E, Faghih, Ramin, Miller, Thomas R, Milicic, Ivan, Baranowski, John L, Krueger, Kathleen M, Witte, David G, Molesky, Angela L, Komater, Victoria A, Buckley, Michael J, Diaz, Gilbert J, Gagne, Gerard D, Zhou, Deliang, Deng, Xiaoqing, Pan, Liping, Roberts, Ellen M, Diehl, Marilyn S, Wetter, Jill M, Marsh, Kennan C, Fox, Gerard B, Brioni, Jorge D, Esbenshade, Timothy A, Hancock, Arthur A

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4-(2-[2-(2( R )-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl)benzonitrile and Related 2-Aminoethylbenzofuran H 3 Receptor Antagonists Potently Enhance Cognition and Attention von Cowart, Marlon, Faghih, Ramin, Curtis, Michael P., Gfesser, Gregory A., Bennani, Youssef L., Black, Lawrence A., Pan, Liping, Marsh, Kennan C., Sullivan, James P., Esbenshade, Timothy A., Fox, Gerard B., Hancock, Arthur A.

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Synthesis and SAR of 5-Amino- and 5-(Aminomethyl)benzofuran Histamine H 3 Receptor Antagonists with Improved Potency von Sun, Minghua, Zhao, Chen, Gfesser, Gregory A., Thiffault, Christine, Miller, Thomas R., Marsh, Kennan, Wetter, Jill, Curtis, Michael, Faghih, Ramin, Esbenshade, Timothy A., Hancock, Arthur A., Cowart, Marlon

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5-(3-Bromophenyl)-7-(6-morpholin-4-ylpyridin-3-yl)pyrido[2,3-d]pyrimidin-4-ylamine: structure–activity relationships of 7-substituted heteroaryl analogs as non-nucleoside adenosine... von Matulenko, Mark A., Lee, Chih-Hung, Jiang, Meiqun, Frey, Robin R., Cowart, Marlon D., Bayburt, Erol K., DiDomenico, Stanley, Gfesser, Gregory A., Gomtsyan, Arthur, Zheng, Guo Zhu, McKie, Jeffery A., Stewart, Andrew O., Yu, Haixia, Kohlhaas, Kathy L., Alexander, Karen M., McGaraughty, Steve, Wismer, Carol T., Mikusa, Joseph, Marsh, Kennan C., Snyder, Ronald D., Diehl, Marilyn S., Kowaluk, Elizabeth A., Jarvis, Michael F., Bhagwat, Shripad S.

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Evaluation of a synthetic route to ε-viniferin based on a new method for the stereoselective preparation of 2,3-diaryl-2,3-dihydrobenzofurans von Engler, Thomas A., Draney, Bill W., Gfesser, Gregory A.

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Fluorescent benzofuran histamine H(3) receptor antagonists with sub-nanomolar potency von Cowart, M, Gfesser, G A, Bhatia, K, Esser, R, Sun, M, Miller, T R, Krueger, K, Witte, D, Esbenshade, T A, Hancock, A A

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4-(2-[2-(2(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl)benzonit rile and Related 2-Aminoethylbenzofuran H sub(3) Receptor Antagonists Potently Enhance Cognition and Attention von Cowart, M, Faghih, R, Curtis, M P, Gfesser, G A, Bennani, Y L, Black, LA, Pan, L, Marsh, K C, Sullivan, J P, Esbenshade, T A, Fox, G B, Hancock, A A

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Adenosine kinase inhibitors: polar 7-Substitutent of pyridopyrimidine derivatives improving their locomotor selectivity von Zheng, Guo Zhu, Mao, Yue, Lee, Chih-Hung, Pratt, John K., Koenig, John R., Perner, Richard J., Cowart, Marlon D., Gfesser, Gregory A., McGaraughty, Steve, Chu, Katharine L., Zhu, Chang, Yu, Haixia, Kohlhaas, Kathy, Alexander, Karen M., Wismer, Carol T., Mikusa, Joseph, Jarvis, Michael F., Kowaluk, Elizabeth A., Stewart, Andrew O.

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Synthesis and structure-activity relationships of 5-heteroatom-substituted pyridopyrimidines as adenosine kinase inhibitors von Gfesser, Gregory A, Bayburt, Erol K, Cowart, Marlon, DiDomenico, Stanley, Gomtsyan, Arthur, Lee, Chih-Hung, Stewart, Andrew O, Jarvis, Michael F, Kowaluk, Elizabeth A, Bhagwat, Shripad S

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The medicinal chemistry of novel H(3) antagonists von Cowart, M, Faghih, R, Gfesser, G, Curtis, M, Pratt, J K, Bennani, Y, Fox, G B, Esbenshade, T A, Hancock, A A

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Structure–activity relationships of non-imidazole H 3 receptor ligands. Part 3: 5-Substituted 3-phenyl-1,2,4-oxadiazoles as potent antagonists von Gfesser, Gregory A., Zhang, Henry, Dinges, Jurgen, Fox, Gerard B., Pan, Jia Bao, Esbenshade, Timothy A., Yao, Betty B., Witte, David, Miller, Thomas R., Kang, Chae-Hee, Krueger, Kathy M., Bennani, Youssef L., Hancock, Arthur A., Faghih, Ramin

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Lewis Acid-Promoted Reactions of Unsymmetrically Substituted Stilbenes with 2-Methoxy-1,4-benzoquinones: Stereoselective Synthesis of trans-2,3-Diaryl-2,3-dihydrobenzofurans von Engler, Thomas A, Gfesser, Gregory A, Draney, Bill W

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Common EIF4E variants modulate risk for autism spectrum disorders in the high-functioning range von Waltes, Regina, Gfesser, Johannes, Haslinger, Denise, Schneider-Momm, Katja, Biscaldi, Monica, Voran, Anette, Freitag, Christine M., Chiocchetti, Andreas G.

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AMbER - Adaptive Instructional Systems as a Use Case for the Holistic Assessment Platform von Witte, Thomas E. F., Gfesser, Torsten, Schwarz, Jessica

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