Inhibition of demethylases by GSK-J1/J4 von Heinemann, Bo, Nielsen, Jesper Morten, Hudlebusch, Heidi Rye, Lees, Michael J., Larsen, Dorthe Vang, Boesen, Thomas, Labelle, Marc, Gerlach, Lars-Ole, Birk, Peter, Helin, Kristian

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GPR39 Signaling Is Stimulated by Zinc Ions But Not by Obestatin von Holst, Birgitte, Egerod, Kristoffer L, Schild, Enrico, Vickers, Steve P, Cheetham, Sharon, Gerlach, Lars-Ole, Storjohann, Laura, Stidsen, Carsten E, Jones, Rob, Beck-Sickinger, Annette G, Schwartz, Thue W

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Molecular Mechanism of Action of Monocyclam Versus Bicyclam Non-peptide Antagonists in the CXCR4 Chemokine Receptor von Rosenkilde, Mette M., Gerlach, Lars-Ole, Hatse, Sigrid, Skerlj, Renato T., Schols, Dominique, Bridger, Gary J., Schwartz, Thue W.

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Long-Acting Lipidated Analogue of Human Pancreatic Polypeptide Is Slowly Released into Circulation von Bellmann-Sickert, Kathrin, Elling, Christian E, Madsen, Andreas N, Little, Paul B, Lundgren, Karsten, Gerlach, Lars-Ole, Bergmann, Ralf, Holst, Birgitte, Schwartz, Thue W, Beck-Sickinger, Annette G

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Molecular mechanism of AMD3100 antagonism in the CXCR4 receptor: transfer of binding site to the CXCR3 receptor von Rosenkilde, Mette M, Gerlach, Lars-Ole, Jakobsen, Janus S, Skerlj, Renato T, Bridger, Gary J, Schwartz, Thue W

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Metal Ion Site Engineering Indicates a Global Toggle Switch Model for Seven-transmembrane Receptor Activation von Elling, Christian E., Frimurer, Thomas M., Gerlach, Lars-Ole, Jorgensen, Rasmus, Holst, Birgitte, Schwartz, Thue W.

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Model-Based Discovery of Synthetic Agonists for the Zn2+-Sensing G‑Protein-Coupled Receptor 39 (GPR39) Reveals Novel Biological Functions von Frimurer, Thomas M, Mende, Franziska, Graae, Anne-Sofie, Engelstoft, Maja S, Egerod, Kristoffer L, Nygaard, Rie, Gerlach, Lars-Ole, Hansen, Jakob Bondo, Schwartz, Thue W, Holst, Birgitte

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Inhibition of Human Immunodeficiency Virus Replication by a Dual CCR5/CXCR4 Antagonist von PRINCEN, Katrien, HATSE, Sigrid, SCHOLS, Dominique, VERMEIRE, Kurt, AQUARO, Stefano, DE CLERCQ, Erik, GERLACH, Lars-Ole, ROSENKILDE, Mette, SCHWARTZ, Thue W, SKERLJ, Renato, BRIDGER, Gary

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A physicogenetic method to assign ligand-binding relationships between 7TM receptors von Frimurer, Thomas M., Ulven, Trond, Elling, Christian E., Gerlach, Lars-Ole, Kostenis, Evi, Högberg, Thomas

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Molecular Interactions of Cyclam and Bicyclam Non-peptide Antagonists with the CXCR4 Chemokine Receptor von Gerlach, L O, Skerlj, R T, Bridger, G J, Schwartz, T W

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Novel Selective Orally Active CRTH2 Antagonists for Allergic Inflammation Developed from in Silico Derived Hits von Ulven, Trond, Receveur, Jean-Marie, Grimstrup, Marie, Rist, Øystein, Frimurer, Thomas M, Gerlach, Lars-Ole, Mathiesen, Jesper Mosolff, Kostenis, Evi, Uller, Lena, Högberg, Thomas

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Identification of Indole Derivatives Exclusively Interfering with a G Protein-Independent Signaling Pathway of the Prostaglandin D2 Receptor CRTH2 von Mathiesen, Jesper Mosolff, Ulven, Trond, Martini, Lene, Gerlach, Lars Ole, Heinemann, Akos, Kostenis, Evi

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Mutations at the CXCR4 interaction sites for AMD3100 influence anti-CXCR4 antibody binding and HIV-1 entry von Hatse, Sigrid, Princen, Katrien, Vermeire, Kurt, Gerlach, Lars-Ole, Rosenkilde, Mette M., Schwartz, Thue W., Bridger, Gary, De Clercq, Erik, Schols, Dominique

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HER2-positive breast-cancer cell lines are sensitive to KDM5 inhibition: definition of a gene-expression model for the selection of sensitive cases von Paroni, Gabriela, Bolis, Marco, Zanetti, Adriana, Ubezio, Paolo, Helin, Kristian, Staller, Peter, Gerlach, Lars Ole, Fratelli, Maddalena, Neve, Richard M., Terao, Mineko, Garattini, Enrico

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Preparation and evaluation of sulfur-containing metal chelators von Clavier, Sylvain, Rist, Oystein, Hansen, Stina, Gerlach, Lars-Ole, Högberg, Thomas, Bergman, Jan

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Model-Based Discovery of Synthetic Agonists for the Zn 2+ -Sensing G-Protein-Coupled Receptor 39 (GPR39) Reveals Novel Biological Functions von Frimurer, Thomas M, Mende, Franziska, Graae, Anne-Sofie, Engelstoft, Maja S, Egerod, Kristoffer L, Nygaard, Rie, Gerlach, Lars-Ole, Hansen, Jakob Bondo, Schwartz, Thue W, Holst, Birgitte

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Abstract 5161: The development of therapeutic inhibitors of the KDM5 histone demethylases von Hudlebusch, Heidi R., Heinemann, Bo, Nielsen, Jesper M., Kleine-Kohlbrecher, Daniela, Hauge, Camilla, Boesen, Thomas, Labelle, Marc, Gerlach, Lars-Ole, Staller, Peter, Birk, Peter

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A 4-year non-randomized comparative phase-IV study of early rheumatoid arthritis: integrative anthroposophic medicine for patients with preference against DMARDs versus conventiona... von Hamre, Harald J, Pham, Van N, Kern, Christian, Rau, Rolf, Klasen, Jörn, Schendel, Ute, Gerlach, Lars, Drabik, Attyla, Simon, Ludger

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Molecular Mechanism of AMD3100 Antagonism in the CXCR4 Receptor von Rosenkilde, Mette M., Gerlach, Lars-Ole, Jakobsen, Janus S., Skerlj, Renato T., Bridger, Gary J., Schwartz, Thue W.

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Mutation of Asp(171) and Asp(262) of the chemokine receptor CXCR4 impairs its coreceptor function for human immunodeficiency virus-1 entry and abrogates the antagonistic activity o... von Hatse, S, Princen, K, Gerlach, L O, Bridger, G, Henson, G, De Clercq, E, Schwartz, T W, Schols, D

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