Two Approaches to a Trifluoromethyl Triazole: A Fit-for-Purpose Trifluoromethylation in Flow-Mode and a Long-Term Decarboxylative Click Approach von Ayothiraman, Rajaram, Gangu, Aravind S, Bandaru, Durgarao, Guturi, Siva Krishna, Lakshminarasimhan, Thirumalai, Jaleel, Mohamed, Kanagavel, Kishorekumar, Rangaswamy, Sundaramurthy, Cuniere, Nicolas L, Zaretsky, Serge, Camacho, Kathryn, Eastgate, Martin D, Vaidyanathan, Rajappa

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Development of a Scalable Synthetic Route to BMS-986251. Part 1: Synthesis of the Cyclohexane Dicarboxylate Fragment von Kuppusamy, Sankar, Gangu, Aravind S, Kalidindi, Srinivas, Ponnusamy, Muthukrishnan, Tendulkar, Shankar, Venu, Alla, Palani, Senthil, Nagappan, Vedhachalam, Vinodini, Arun, Mudryk, Boguslaw, Rupasinghe, Sanjeewa, Joe, Candice L, Coombs, John R, Gallagher, William P, Kopp, Nathaniel, Gonzalez-Bobes, Francisco, Eastgate, Martin D, Vaidyanathan, Rajappa

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Development of a Scalable Synthetic Route to BMS-986251, Part 2: Synthesis of the Tricyclic Core and the API von Kalidindi, Srinivas, Gangu, Aravind S, Kuppusamy, Sankar, Sathasivam, Shunmugaraj, Shekarappa, Vijaykumar, Murugan, Saravanan, Bondigela, Sivasankar, Kandasamy, Moorthy, Ghanta, Kishore, Vinodini, Arun, Shrikant, Abhishek, Ramachandran, Ravikumar, Gallagher, William P, Kopp, Nathaniel, González-Bobes, Francisco, Eastgate, Martin D, Vaidyanathan, Rajappa

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Development of Continuous Flow Processes to Access Pyrrolo[2,1‑f][1,2,4]triazin-4-amine: An RSM for the Synthesis of Antiviral Drugs von Vasilev, Maksim, Gangu, Aravind S., Gajula, Praveen, Kaetzel, Nathaniel D., Natarajan, Vasudevan, Desai, Bimbisar, Sirasani, Gopal, Qu, Bo, Senanayake, Chris H.

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Development and Execution of an Ni(II)-Catalyzed Reductive Cross-Coupling of Substituted 2-Chloropyridine and Ethyl 3-Chloropropanoate von Nimmagadda, Krishna, Korapati, Satish, Dasgupta, Debottam, Malik, Noormohamed Abdul, Vinodini, Arun, Gangu, Aravind S., Kalidindi, Srinivas, Maity, Prantik, Bondigela, Siva Sankar, Venu, Alla, Gallagher, William P., Aytar, Selin, Gonzalez-Bobes, Francisco, Vaidyanathan, Rajappa

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Development of a Safer Continuous Flow Process for B 2 (OH) 4 -Mediated Chemoselective Reduction of Nitroarenes to Anilines von Revu, Omkar, Vasilev, Maksim, Gajula, Praveen, Kalikinidi, Nageswara Rao, Gadi, Madhusudhan Reddy, Zhao, Huiping, Gamage, Shanika M. P., Hibbert, Graham, Ravikumar, Ongolu, Gummidi, Lalitha, Nasipireddy, Venkatarathnam, Vinodini, Arun, Bietsch, Jonathan, Wang, Zhirui, Brown, Jack D., Sirasani, Gopal, Armstrong, Joseph D., Gangu, Aravind S., Qu, Bo, Senanayake, Chris H.

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Development of a Safer Continuous Flow Process for B2(OH)4‑Mediated Chemoselective Reduction of Nitroarenes to Anilines von Revu, Omkar, Vasilev, Maksim, Gajula, Praveen, Kalikinidi, Nageswara Rao, Gadi, Madhusudhan Reddy, Zhao, Huiping, Gamage, Shanika M. P., Hibbert, Graham, Ravikumar, Ongolu, Gummidi, Lalitha, Nasipireddy, Venkatarathnam, Vinodini, Arun, Bietsch, Jonathan, Wang, Zhirui, Brown, Jack D., Sirasani, Gopal, Armstrong, Joseph D., Gangu, Aravind S., Qu, Bo, Senanayake, Chris H.

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Synthesis of Chiral 1,2-Amino Alcohol-Containing Compounds Utilizing Ruthenium-Catalyzed Asymmetric Transfer Hydrogenation of Unprotected α‑Ketoamines von Mangunuru, Hari P. R., Terrab, Leila, Janganati, Venumadhav, Kalikinidi, Nageswara Rao, Tenneti, Srinivasarao, Natarajan, Vasudevan, Shada, Arun D. R., Naini, Santhosh Reddy, Gajula, Praveen, Lee, Daniel, Samankumara, Lalith P., Mamunooru, Manasa, Jayaraman, Aravindan, Sahani, Rajkumar Lalji, Yin, Jinya, Hewa-Rahinduwage, Chathuranga C., Gangu, Aravind, Chen, Anji, Wang, Zhirui, Desai, Bimbisar, Yue, Tai Y., Wannere, Chaitanya S., Armstrong, Joseph D., Donsbach, Kai O., Sirasani, Gopal, Gupton, B. Frank, Qu, Bo, Senanayake, Chris H.

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Alternative Approach to the Large-Scale Synthesis of the Densely Functionalized Pyrrolidone BMT-415200 von Rakshit, Souvik, Sathasivam, Shunmugaraj, Reddy, Raghurami, Rao, Saladi V., Shekarappa, Vijaykumar, Kandasamy, Moorthy, Jaleel, Mohamed, Murugan, Saravanan, Bhat, Anuradha, Subramani, Tamilarasan, Lakshminarasimhan, Thirumalai, Gangu, Aravind, Wisniewski, Steven R., Kopp, Nathaniel, Hale, Ian, Stevens, Jason M., Rosso, Victor W., Eastgate, Martin D., Vaidyanathan, Rajappa

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Facile and Scalable Methodology for the Pyrrolo[2,1‑f][1,2,4]triazine of Remdesivir von Roy, Sarabindu, Yadaw, Ajay, Roy, Subho, Sirasani, Gopal, Gangu, Aravind, Brown, Jack D, Armstrong, Joseph D, Stringham, Rodger W, Gupton, B. Frank, Senanayake, Chris H, Snead, David R

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