Compounds that block both intermediate‐conductance (IKCa) and small‐conductance (SKCa) calcium‐activated potassium channels von Malik‐Hall, M, Ganellin, C R, Galanakis, D, Jenkinson, D H

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Distinct pharmacology of rat and human histamine H3 receptors: role of two amino acids in the third transmembrane domain von Ligneau, X, Morisset, S, Tardivel‐Lacombe, J, Gbahou, F, Ganellin, C R, Stark, H, Schunack, W, Schwartz, J ‐C, Arrang, J ‐M

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Clotrimazole analogues: effective blockers of the slow afterhyperpolarization in cultured rat hippocampal pyramidal neurones von Shah, M M, Miscony, Z, Javadzadeh‐Tabatabaie, M, Ganellin, C R, Haylett, D G

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Distinct pharmacology of rat and human histamine H 3 receptors: role of two amino acids in the third transmembrane domain von Ligneau, X, Morisset, S, Tardivel‐Lacombe, J, Gbahou, F, Ganellin, C R, Stark, H, Schunack, W, Schwartz, J ‐C, Arrang, J ‐M

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Glossary of terms used in medicinal chemistry (IUPAC Recommendations 1998) von Wermuth, C. G., Ganellin, C. R., Lindberg, P., Mitscher, L. A.

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Correlation between log POCT/H2O and pKB estimates for a series of muscarinic and histamine H2‐receptor antagonists von Shankley, N.P., Black, J.W., Ganellin, C.R., Mitchell, R.C.

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Differences in the actions of some blockers of the calcium‐activated potassium permeability in mammalian red cells von Benton, D C H, Roxburgh, C J, Ganellin, C R, Shiner, M A R, Jenkinson, D H

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Synthesis, molecular modeling, and pharmacological testing of bis-quinolinium cyclophanes: potent, non-peptidic blockers of the apamin-sensitive Ca(2+)-activated K(+) channel von Campos Rosa, J, Galanakis, D, Piergentili, A, Bhandari, K, Ganellin, C R, Dunn, P M, Jenkinson, D H

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Sedation and histamine H1‐receptor antagonism: studies in man with the enantiomers of chlorpheniramine and dimethindene von Nicholson, A.N., Pascoe, Peta A., Turner, Claire, Ganellin, C.R., Greengrass, P.M., Casy, A.F., Mercer, Amanda D.

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Histamine H1‐Receptor in Heart: Unique Electrophoretic Mobility and Autoradiographic Localization von Ruat, M., Bouthenet, M. L., Schwartz, J.‐C., Ganellin, C. R.

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Bis-quinolinium cyclophanes: 6,10-diaza-3(1,3),8(1,4)-dibenzena-1,5(1,4)- diquinolinacyclodecaphane (UCL 1684), the first nanomolar, non-peptidic blocker of the apamin-sensitive Ca... von Rosa, J C, Galanakis, D, Ganellin, C R, Dunn, P M, Jenkinson, D H

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Zolantidine (SK&F 95282) is a potent selective brain‐penetrating histamine H2‐receptor antagonist von Calcutt, C.R., Ganellin, C.R., Griffiths, R., Leigh, B.K., Maguire, J.P., Mitchell, R.C., Mylek, M.E., Parsons, M.E., Smith, I.R., Young, R.C.

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Molecule-Receptor Specificity von Richards, W. G., Clarkson, R., Ganellin, C. R.

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Characterization and inhibition of a cholecystokinin-inactivating serine peptidase von Rose, Christiane, Vargas, Froylan, Facchinetti, Patricia, Bourgeat, Pierre, Bambal, Ramesh B, Bishop, Paul B, Chan, Suzanne M. T, Moore, Andrew N. J, Ganellin, C. Robin, Schwartz, Jean-Charles

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Characterization and development of cimetidine as a histamine H2-receptor antagonist von Brimblecombe, R.W., Duncan, W.A.M., Durant, G.J., Emmett, J.C., Ganellin, C.R., Leslie, G.B., Parsons, M.E.

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Conformation of histamine derivatives. 3. A relationship between conformation and pharmacological activity von Ganellin, C R

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Medicinal chemistry in the development of societies: Biodiversity and natural products von Monge, A., Chorghade, M., Erhardt, P.W., Ganellin, C.R., Koga, N., Lindberg, P., Perun, T.J., Topliss, J.G., Trivedi, B.K., Wermuth, C.G.

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Evidence for low brain penetration by the H1-receptor antagonist temelastine (SK&F 93944) von CALCUTT, C. R, GANELLIN, C. R, JACKSON, B, LEIGH, B. K, OWEN, D. A. A, SMITH, I. R

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Compounds Affecting the Central Nervous System. I. 4-Piperidones and Related Compounds von Ganellin, C. R, Spickett, R. G. W

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A Novel Series of (Phenoxyalkyl)imidazoles as Potent H3-Receptor Histamine Antagonists von Ganellin, C. Robin, Fkyerat, Abdellatif, Bang-Andersen, Benny, Athmani, Salah, Tertiuk, Wasyl, Garbarg, Monique, Ligneau, Xavier, Schwartz, Jean-Charles

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