Glossary of terms used in medicinal chemistry (IUPAC Recommendations 1998) von Wermuth, C. G., Ganellin, C. R., Lindberg, P., Mitscher, L. A.

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Compounds that block both intermediate‐conductance (IKCa) and small‐conductance (SKCa) calcium‐activated potassium channels von Malik‐Hall, M, Ganellin, C R, Galanakis, D, Jenkinson, D H

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Distinct pharmacology of rat and human histamine H3 receptors: role of two amino acids in the third transmembrane domain von Ligneau, X, Morisset, S, Tardivel‐Lacombe, J, Gbahou, F, Ganellin, C R, Stark, H, Schunack, W, Schwartz, J ‐C, Arrang, J ‐M

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Synthesis, molecular modeling, and pharmacological testing of bis-quinolinium cyclophanes: potent, non-peptidic blockers of the apamin-sensitive Ca(2+)-activated K(+) channel von Campos Rosa, J, Galanakis, D, Piergentili, A, Bhandari, K, Ganellin, C R, Dunn, P M, Jenkinson, D H

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Distinct pharmacology of rat and human histamine H 3 receptors: role of two amino acids in the third transmembrane domain von Ligneau, X, Morisset, S, Tardivel‐Lacombe, J, Gbahou, F, Ganellin, C R, Stark, H, Schunack, W, Schwartz, J ‐C, Arrang, J ‐M

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Clotrimazole analogues: effective blockers of the slow afterhyperpolarization in cultured rat hippocampal pyramidal neurones von Shah, M M, Miscony, Z, Javadzadeh‐Tabatabaie, M, Ganellin, C R, Haylett, D G

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Bis-quinolinium cyclophanes: 6,10-diaza-3(1,3),8(1,4)-dibenzena-1,5(1,4)- diquinolinacyclodecaphane (UCL 1684), the first nanomolar, non-peptidic blocker of the apamin-sensitive Ca... von Rosa, J C, Galanakis, D, Ganellin, C R, Dunn, P M, Jenkinson, D H

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Characterization and inhibition of a cholecystokinin-inactivating serine peptidase von Rose, Christiane, Vargas, Froylan, Facchinetti, Patricia, Bourgeat, Pierre, Bambal, Ramesh B, Bishop, Paul B, Chan, Suzanne M. T, Moore, Andrew N. J, Ganellin, C. Robin, Schwartz, Jean-Charles

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Histamine H1‐Receptor in Heart: Unique Electrophoretic Mobility and Autoradiographic Localization von Ruat, M., Bouthenet, M. L., Schwartz, J.‐C., Ganellin, C. R.

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Differences in the actions of some blockers of the calcium‐activated potassium permeability in mammalian red cells von Benton, D C H, Roxburgh, C J, Ganellin, C R, Shiner, M A R, Jenkinson, D H

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Calcium-activated potassium channels sustain calcium signaling in T lymphocytes. Selective blockers and manipulated channel expression levels von Fanger, C M, Rauer, H, Neben, A L, Miller, M J, Wulff, H, Rosa, J C, Ganellin, C R, Chandy, K G, Cahalan, M D

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Medicinal chemistry in the development of societies: Biodiversity and natural products von Monge, A., Chorghade, M., Erhardt, P.W., Ganellin, C.R., Koga, N., Lindberg, P., Perun, T.J., Topliss, J.G., Trivedi, B.K., Wermuth, C.G.

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The pharmacology of cimetidine, a new histamine H 2 ‐receptor antagonist von Brimblecombe, RW, Duncan, WAM, Durant, GJ, Ganellin, CR, Parsons, ME, Black, JW

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Correlation between log POCT/H2O and pKB estimates for a series of muscarinic and histamine H2‐receptor antagonists von Shankley, N.P., Black, J.W., Ganellin, C.R., Mitchell, R.C.

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A Novel Series of (Phenoxyalkyl)imidazoles as Potent H3-Receptor Histamine Antagonists von Ganellin, C. Robin, Fkyerat, Abdellatif, Bang-Andersen, Benny, Athmani, Salah, Tertiuk, Wasyl, Garbarg, Monique, Ligneau, Xavier, Schwartz, Jean-Charles

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Sedation and histamine H1‐receptor antagonism: studies in man with the enantiomers of chlorpheniramine and dimethindene von Nicholson, A.N., Pascoe, Peta A., Turner, Claire, Ganellin, C.R., Greengrass, P.M., Casy, A.F., Mercer, Amanda D.

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Influence of imidazole replacement in different structural classes of histamine H(3)-receptor antagonists von Meier, G, Apelt, J, Reichert, U, Grassmann, S, Ligneau, X, Elz, S, Leurquin, F, Ganellin, C R, Schwartz, J C, Schunack, W, Stark, H

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Inhibitors of Tripeptidyl Peptidase II. 2. Generation of the First Novel Lead Inhibitor of Cholecystokinin-8-Inactivating Peptidase:  A Strategy for the Design of Peptidase Inhibit... von Ganellin, C. Robin, Bishop, Paul B, Bambal, Ramesh B, Chan, Suzanne M. T, Law, James K, Marabout, Benoit, Luthra, Pratibha Mehta, Moore, Andrew N. J, Peschard, Olivier, Bourgeat, Pierre, Rose, Christiane, Vargas, Froylan, Schwartz, Jean-Charles

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Synthesis and Structure-Activity Relationships of Dequalinium Analogs as K+ Channel Blockers. Investigations on the Role of the Charged Heterocycle von Galanakis, Dimitrios, Davis, Carole A, Herrero, Benedicto Del Rey, Ganellin, C. Robin, Dunn, Philip M, Jenkinson, Donald H

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Synthesis and quantitative structure-activity relationships of dequalinium analogues as K+ channel blockers : investigation into the role of the substituent at position 4 of the qu... von GALANAKIS, D, CALDER, J. A. D, GANELLIN, C. R, OWEN, C. S, DUNN, P. M

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