Design, Synthesis, and Structural Characterization of Lysine Covalent BH3 Peptides Targeting Mcl‑1 von Gambini, Luca, Udompholkul, Parima, Baggio, Carlo, Muralidharan, Aruljothi, Kenjić, Nikola, Assar, Zahra, Perry, J. Jefferson P, Pellecchia, Maurizio

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Reduction of Circulating Cancer Cells and Metastases in Breast-Cancer Models by a Potent EphA2-Agonistic Peptide–Drug Conjugate von Salem, Ahmed F, Wang, Si, Billet, Sandrine, Chen, Jie-Fu, Udompholkul, Parima, Gambini, Luca, Baggio, Carlo, Tseng, Hsian-Rong, Posadas, Edwin M, Bhowmick, Neil A, Pellecchia, Maurizio

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Potential Therapeutic Targeting of Coronavirus Spike Glycoprotein Priming von Barile, Elisa, Baggio, Carlo, Gambini, Luca, Shiryaev, Sergey A., Strongin, Alex Y., Pellecchia, Maurizio

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Effective Tumor Targeting by EphA2-Agonist-Biotin-Streptavidin Conjugates von Udompholkul, Parima, Baggio, Carlo, Gambini, Luca, Sun, Yu, Zhao, Ming, Hoffman, Robert M., Pellecchia, Maurizio

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NMR Fingerprints of the Drug-like Natural-Product Space Identify Iotrochotazine A: A Chemical Probe to Study Parkinson's Disease von Grkovic, Tanja, Pouwer, Rebecca H., Vial, Marie-Laure, Gambini, Luca, Noël, Alba, Hooper, John N. A., Wood, Stephen A., Mellick, George D., Quinn, Ronald J.

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Therapeutic Targeting of Pancreatic Cancer via EphA2 Dimeric Agonistic Agents von Salem, Ahmed F., Gambini, Luca, Udompholkul, Parima, Baggio, Carlo, Pellecchia, Maurizio

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Picomolar Inhibition of Plasmepsin V, an Essential Malaria Protease, Achieved Exploiting the Prime Region von Gambini, Luca, Rizzi, Luca, Pedretti, Alessandro, Taglialatela-Scafati, Orazio, Carucci, Mario, Pancotti, Andrea, Galli, Corinna, Read, Martin, Giurisato, Emanuele, Romeo, Sergio, Russo, Ilaria

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Correction: Picomolar Inhibition of Plasmepsin V, an Essential Malaria Protease, Achieved Exploiting the Prime Region von Gambini, Luca, Rizzi, Luca, Pedretti, Alessandro, Taglialatela-Scafati, Orazio, Carucci, Mario, Pancotti, Andrea, Galli, Corinna, Read, Martin, Giurisato, Emanuele, Romeo, Sergio, Russo, Ilaria

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Lysine Covalent Antagonists of Melanoma Inhibitors of Apoptosis Protein von Udompholkul, Parima, Baggio, Carlo, Gambini, Luca, Alboreggia, Giulia, Pellecchia, Maurizio

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Targefrin: A Potent Agent Targeting the Ligand Binding Domain of EphA2 von Baggio, Carlo, Udompholkul, Parima, Gambini, Luca, Pellecchia, Maurizio

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Covalent Inhibitors of Protein–Protein Interactions Targeting Lysine, Tyrosine, or Histidine Residues von Gambini, Luca, Baggio, Carlo, Udompholkul, Parima, Jossart, Jennifer, Salem, Ahmed F, Perry, J. Jefferson P, Pellecchia, Maurizio

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Aryl-fluorosulfate-based Lysine Covalent Pan-Inhibitors of Apoptosis Protein (IAP) Antagonists with Cellular Efficacy von Baggio, Carlo, Udompholkul, Parima, Gambini, Luca, Salem, Ahmed F, Jossart, Jennifer, Perry, J. Jefferson P, Pellecchia, Maurizio

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Stability and Cell Permeability of Sulfonyl Fluorides in the Design of Lys‐Covalent Antagonists of Protein‐Protein Interactions von Gambini, Luca, Udompholkul, Parima, Salem, Ahmed F., Baggio, Carlo, Pellecchia, Maurizio

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Design of Potent pan-IAP and Lys-Covalent XIAP Selective Inhibitors Using a Thermodynamics Driven Approach von Baggio, Carlo, Gambini, Luca, Udompholkul, Parima, Salem, Ahmed F, Aronson, Alexander, Dona, Ada, Troadec, Estelle, Pichiorri, Flavia, Pellecchia, Maurizio

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Human resistin protects against endotoxic shock by blocking LPS–TLR4 interaction von Jang, Jessica C., Li, Jiang, Gambini, Luca, Batugedara, Hashini M., Sati, Sandeep, Lazar, Mitchell A., Fan, Li, Pellecchia, Maurizio, Nair, Meera G.

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Abstract 3911: Targeting the EphA2-ligand binding domain for the design of innovative cancer therapeutics von Udompholkul, Parima, Gambini, Luca, Salem, Ahmed F., Baggio, Carlo, Pellecchia, Maurizio

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Aryl-fluorosulfate-based Lysine Covalent pan-Inhibitors of Apoptosis Proteins (IAP) Antagonists with Cellular Efficacy von Baggio, Carlo, Udompholkul, Parima, Gambini, Luca, Salem, Ahmed F., Jossart, Jennifer, Perry, J. Jefferson P., Pellecchia, Maurizio

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Structure-Based Design of Novel EphA2 Agonistic Agents with Nanomolar Affinity in Vitro and in Cell von Gambini, Luca, Salem, Ahmed F, Udompholkul, Parima, Tan, Xiao-Feng, Baggio, Carlo, Shah, Neh, Aronson, Alexander, Song, Jikui, Pellecchia, Maurizio

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Theranostic Nanocages for Imaging and Photothermal Therapy of Prostate Cancer Cells by Active Targeting of Neuropeptide‑Y Receptor von Avvakumova, Svetlana, Galbiati, Elisabetta, Sironi, Laura, Locarno, Silvia A, Gambini, Luca, Macchi, Chiara, Pandolfi, Laura, Ruscica, Massimiliano, Magni, Paolo, Collini, Maddalena, Colombo, Miriam, Corsi, Fabio, Chirico, Giuseppe, Romeo, Sergio, Prosperi, Davide

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N‐locking stabilization of covalent helical peptides: Application to Bfl‐1 antagonists von Baggio, Carlo, Udompholkul, Parima, Gambini, Luca, Jossart, Jennifer, Salem, Ahmed F., Håkansson, Maria, Perry, J. Jefferson P., Pellecchia, Maurizio

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