Prospective discovery of small molecule enhancers of an E3 ligase-substrate interaction von Simonetta, Kyle R., Taygerly, Joshua, Boyle, Kathleen, Basham, Stephen E., Padovani, Chris, Lou, Yan, Cummins, Thomas J., Yung, Stephanie L., von Soly, Szerenke Kiss, Kayser, Frank, Kuriyan, John, Rape, Michael, Cardozo, Mario, Gallop, Mark A., Bence, Neil F., Barsanti, Paul A., Saha, Anjanabha

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Arbaclofen Placarbil, a Novel R-Baclofen Prodrug: Improved Absorption, Distribution, Metabolism, and Elimination Properties Compared with R-Baclofen von Lal, Ritu, Sukbuntherng, Juthamas, Tai, Ezra H.L., Upadhyay, Shubhra, Yao, Fenmei, Warren, Mark S., Luo, Wendy, Bu, Lin, Nguyen, Son, Zamora, Jeanelle, Peng, Ge, Dias, Tracy, Bao, Ying, Ludwikow, Maria, Phan, Thu, Scheuerman, Randall A., Yan, Hui, Gao, Mark, Wu, Quincey Q., Annamalai, Thamil, Raillard, Stephen P., Koller, Kerry, Gallop, Mark A., Cundy, Kenneth C.

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Orally Absorbed Derivatives of the β‑Lactamase Inhibitor Avibactam. Design of Novel Prodrugs of Sulfate Containing Drugs von Gordon, Eric M, Duncton, Matthew A. J, Gallop, Mark A

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Acamprosate Produces Its Anti-Relapse Effects Via Calcium von SPANAGEL, Rainer, VENGELIENE, Valentina, JANDELEIT, Bernd, FISCHER, Wolf-Nicolas, GRINDSTAFF, Kent, XUEXIANG ZHANG, GALLOP, Mark A, KRSTEW, Elena V, LAWRENCE, Andrew J, KIEFER, Falk

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Applications of Combinatorial Technologies to Drug Discovery. 2. Combinatorial Organic Synthesis, Library Screening Strategies, and Future Directions von Gordon, Eric M, Barrett, Ronald W, Dower, William J, Fodor, Stephen P. A, Gallop, Mark A

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Applications of Combinatorial Technologies to Drug Discovery. 1. Background and Peptide Combinatorial Libraries von Gallop, Mark A, Barrett, Ronald W, Dower, William J, Fodor, Stephen P. A, Gordon, Eric M

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Combinatorial Organic Synthesis of Highly Functionalized Pyrrolidines: Identification of a Potent Angiotensin Converting Enzyme Inhibitor from a Mercaptoacyl Proline Library von Murphy, Martin M, Schullek, John R, Gordon, Eric M, Gallop, Mark A

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Solid-Phase Synthesis of 3,5-Disubstituted 2,3-Dihydro-1,5-benzothiazepin-4(5H)-ones von Schwarz, Matthias K, Tumelty, David, Gallop, Mark A

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Stereoselective Solid-Phase Synthesis of a Triaza Tricyclic Ring System:  A New Chemotype for Lead Discovery von Peng, Ge, Sohn, Amy, Gallop, Mark A

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Discovery of a novel potent GABA(B) receptor agonist von Xu, Feng, Peng, Ge, Phan, Thu, Dilip, Usha, Chen, Jian Lu, Chernov-Rogan, Tania, Zhang, Xuexiang, Grindstaff, Kent, Annamalai, Thamil, Koller, Kerry, Gallop, Mark A, Wustrow, David J

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Discovery of a novel potent GABAB receptor agonist von Xu, Feng, Peng, Ge, Phan, Thu, Dilip, Usha, Chen, Jian Lu, Chernov-Rogan, Tania, Zhang, Xuexiang, Grindstaff, Kent, Annamalai, Thamil, Koller, Kerry, Gallop, Mark A, Wustrow, David J

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Strategies for the Synthesis and Screening of Glycoconjugates. 1. A Library of Glycosylamines von Vetter, Dirk, Gallop, Mark A

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New methods for analyzing compounds on polymeric supports von Gallop, Mark A, Fitch, William L

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Solid-Supported Combinatorial Synthesis of Structurally Diverse β-Lactams von Ruhland, Beatrice, Bhandari, Ashok, Gordon, Eric M, Gallop, Mark A

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Solid-Phase Synthesis of 4-Arylazetidin-2-ones via Suzuki and Heck Cross-Coupling Reactions von Ruhland, Beatrice, Bombrun, Agnes, Gallop, Mark A

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Validation of tele-otology to diagnose ear disease in children von Eikelboom, Robert H., Mbao, Mathew N., Coates, Harvey L., Atlas, Marcus D., Gallop, Mark A.

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Synthesis and biological evaluation of novel steroidal pyrazoles as substrates for bile acid transporters von Bhat, Laxminarayan, Jandeleit, Bernd, Dias, Tracy M., Moors, Tristen L., Gallop, Mark A.

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Trimethylorthoformate: A mild and effective dehydrating reagent for solution and solid phase imine formation von Look, Gary C., Murphy, Martin M., Campbell, David A., Gallop, Mark A.

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Strategies for Combinatorial Organic Synthesis: Solution and Polymer-Supported Synthesis of 4-Thiazolidinones and 4-Metathiazanones Derived from Amino Acids von Holmes, Christopher P, Chinn, Jason P, Look, Gary C, Gordon, Eric M, Gallop, Mark A

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A face-capping bonding mode for benzene in triosmium carbonyl cluster complexes von Gallop, Mark A, Gomez-Sal, M. Pilar, Housecroft, Catherine E, Johnson, Brian F. G, Lewis, Jack, Owen, Steven M, Raithby, Paul R, Wright, Anthony H

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