Acute Cholesterol Depletion Inhibits Clathrin-Coated Pit Budding von Subtil, Agathe, Gaidarov, Ibragim, Kobylarz, Keith, Lampson, Michael A., Keen, James H., McGraw, Timothy E.

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Phosphoinositide-AP-2 Interactions Required for Targeting to Plasma Membrane Clathrin-Coated Pits von Gaidarov, Ibragim, Keen, James H.

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Discovery of APD371: Identification of a Highly Potent and Selective CB2 Agonist for the Treatment of Chronic Pain von Han, Sangdon, Thoresen, Lars, Jung, Jae-Kyu, Zhu, Xiuwen, Thatte, Jayant, Solomon, Michelle, Gaidarov, Ibragim, Unett, David J, Yoon, Woo Hyun, Barden, Jeremy, Sadeque, Abu, Usmani, Amin, Chen, Chuan, Semple, Graeme, Grottick, Andrew J, Al-Shamma, Hussein, Christopher, Ronald, Jones, Robert M

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Spatial control of coated-pit dynamics in living cells von Santini, Francesca, Warren, Robin A, Keen, James H, Gaidarov, Ibragim

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Nicotinic Acid Receptor Agonists Differentially Activate Downstream Effectors von Richman, Jeremy G., Kanemitsu-Parks, Martha, Gaidarov, Ibragim, Cameron, Jill S., Griffin, Peter, Zheng, Hong, Guerra, Nuvia C., Cham, Linda, Maciejewski-Lenoir, Dominique, Behan, Dominic P., Boatman, Doug, Chen, Ruoping, Skinner, Philip, Ornelas, Pricilla, Waters, M. Gerard, Wright, Samuel D., Semple, Graeme, Connolly, Daniel T.

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G Protein-Coupled Receptor/Arrestin3 Modulation of the Endocytic Machinery von Santini, Francesca, Gaidarov, Ibragim, Keen, James H.

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Arrestin function in G protein-coupled receptor endocytosis requires phosphoinositide binding von Gaidarov, Ibragim, Krupnick, Jason G., Falck, John R., Benovic, Jeffrey L., Keen, James H.

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Myocardial expression, signaling, and function of GPR22: a protective role for an orphan G protein-coupled receptor von Adams, John W, Wang, Jianming, Davis, James R, Liaw, Chen, Gaidarov, Ibragim, Gatlin, Joel, Dalton, Nancy D, Gu, Yusu, Ross, John, Jr, Behan, Dominic, Chien, Ken, Connolly, Daniel

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Angiotensin (1–7) does not interact directly with MAS1, but can potently antagonize signaling from the AT1 receptor von Gaidarov, Ibragim, Adams, John, Frazer, John, Anthony, Todd, Chen, Xiaohua, Gatlin, Joel, Semple, Graeme, Unett, David J.

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Etrasimod, a Novel Sphingosine‐1‐Phosphate Receptor (S1PR1) Modulator, Lacks Functional Activity at S1P2 Receptors von Adams, John W, Unett, David J., Chen, Xiaohua, Gaidarov, Ibragim

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Functional Activity of Etrasimod and a Diverse Panel of Sphingosine‐1‐Phosphate Receptor (S1PR1) Modulators at S1P4 Receptors von Adams, John W, Unett, David J, Chen, Xiaohua, Gaidarov, Ibragim

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Differential tissue and ligand-dependent signaling of GPR109A receptor: Implications for anti-atherosclerotic therapeutic potential von Gaidarov, Ibragim, Chen, Xiaohua, Anthony, Todd, Maciejewski-Lenoir, Dominique, Liaw, Chen, Unett, David J.

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Etrasimod, a Selective S1P 1,4,5 Receptor Modulator, Exhibits Differential G Protein Signaling Compared to Other S1P Receptor Modulators von Komori, H. Kiyomi, Gaidarov, Ibragim, Bruinsma, Karin, Karimi-Naser, Lisa, Ton, Anh-Tuan, Indersmitten, Tim, Abi-Gerges, Najah, Miller, Paul E., Unett, David, Dang, Huong, Chen, Xiaohua, Adams, John W.

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Kinetics of 5-HT2B receptor signaling: profound agonist-dependent effects on signaling onset and duration von Unett, David J, Gatlin, Joel, Anthony, Todd L, Buzard, Daniel J, Chang, Steve, Chen, Chuan, Chen, Xiaohua, Dang, Huong T-M, Frazer, John, Le, Minh K, Sadeque, Abu J M, Xing, Charles, Gaidarov, Ibragim

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Unique pharmacological properties of etrasimod among S1P receptor modulators von Gaidarov, Ibragim, Komori, H. Kiyomi, Stepniak, Dariusz T., Bruinsma, Karin, Dang, Huong, Chen, Xiaohua, Anthony, Todd, Gatlin, Joel, Karimi‐Naser, Lisa, Ton, Anh‐Tuan, Indersmitten, Tim, Miller, Paul E., Ghetti, Andre, Abi‐Gerges, Najah, Unett, David, Al‐Shamma, Hussien, Rabbat, Christopher J., Crosby, Catherine, Adams, John W.

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Embelin and its derivatives unravel the signaling, proinflammatory and antiatherogenic properties of GPR84 receptor von Gaidarov, Ibragim, Anthony, Todd, Gatlin, Joel, Chen, Xiaohua, Mills, David, Solomon, Michelle, Han, Sangdon, Semple, Graeme, Unett, David J.

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The Class II Phosphoinositide 3-Kinase C2α Is Activated by Clathrin and Regulates Clathrin-Mediated Membrane Trafficking von Gaidarov, Ibragim, Smith, Mary E.K, Domin, Jan, Keen, James H

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Phosphoinositide 3-Kinase C2α Links Clathrin to Microtubule-dependent Movement von Zhao, Yanqiu, Gaidarov, Ibragim, Keen, James H.

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Discovery of 2‑(((1r,4r)‑4-(((4-Chlorophenyl)­(phenyl)­carbamoyl)­oxy)­methyl)­cyclohexyl)­methoxy)­acetate (Ralinepag): An Orally Active Prostacyclin Receptor Agonist for the Trea... von Tran, Thuy-Anh, Kramer, Bryan, Shin, Young-Jun, Vallar, Pureza, Boatman, P. Douglas, Zou, Ning, Sage, Carleton R, Gharbaoui, Tawfik, Krishnan, Ashwin, Pal, Biman, Shakya, Sagar R, Garrido Montalban, Antonio, Adams, John W, Ramirez, Juan, Behan, Dominic P, Shifrina, Anna, Blackburn, Anthony, Leakakos, Tina, Shi, Yunqing, Morgan, Michael, Sadeque, Abu, Chen, Weichao, Unett, David J, Gaidarov, Ibragim, Chen, Xiaohua, Chang, Steve, Shu, Hsin-Hui, Tung, Shiu-Feng, Semple, Graeme

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Individual Phosphoinositide 3-Kinase C2α Domain Activities Independently Regulate Clathrin Function von Gaidarov, Ibragim, Zhao, Yanqiu, Keen, James H.

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