Discovery of [cis-3-({(5R)‑5-[(7-Fluoro-1,1-dimethyl-2,3-dihydro‑1H‑inden-5-yl)carbamoyl]-2-methoxy-7,8-dihydro-1,6-naphthyridin-6(5H)‑yl}carbonyl)­cyclobutyl]­acetic Acid (TAK-828... von Kono, Mitsunori, Ochida, Atsuko, Oda, Tsuneo, Imada, Takashi, Banno, Yoshihiro, Taya, Naohiro, Masada, Shinichi, Kawamoto, Tetsuji, Yonemori, Kazuko, Nara, Yoshi, Fukase, Yoshiyuki, Yukawa, Tomoya, Tokuhara, Hidekazu, Skene, Robert, Sang, Bi-Ching, Hoffman, Isaac D, Snell, Gyorgy P, Uga, Keiko, Shibata, Akira, Igaki, Keiko, Nakamura, Yoshiki, Nakagawa, Hideyuki, Tsuchimori, Noboru, Yamasaki, Masashi, Shirai, Junya, Yamamoto, Satoshi

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Structural Basis for the Autoinhibition and STI-571 Inhibition of c-Kit Tyrosine Kinase von Mol, Clifford D, Dougan, Douglas R, Schneider, Thomas R, Skene, Robert J, Kraus, Michelle L, Scheibe, Daniel N, Snell, Gyorgy P, Zou, Hua, Sang, Bi-Ching, Wilson, Keith P

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Tangling Schedules Eases Hardware Connectivity Requirements for Quantum Error Correction von Gehér, György P., Crawford, Ophelia, Campbell, Earl T.

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2-{3-[4-(Alkylsulfinyl)phenyl]-1-benzofuran-5-yl}-5-methyl-1,3,4-oxadiazole Derivatives as Novel Inhibitors of Glycogen Synthase Kinase-3β with Good Brain Permeability von Saitoh, Morihisa, Kunitomo, Jun, Kimura, Eiji, Iwashita, Hiroki, Uno, Yumiko, Onishi, Tomohiro, Uchiyama, Noriko, Kawamoto, Tomohiro, Tanaka, Toshimasa, Mol, Clifford D, Dougan, Douglas R, Textor, Garret P, Snell, Gyorgy P, Takizawa, Masayuki, Itoh, Fumio, Kori, Masakuni

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Design and Synthesis of Potent Inhibitor of Apoptosis (IAP) Proteins Antagonists Bearing an Octahydropyrrolo[1,2‑a]pyrazine Scaffold as a Novel Proline Mimetic von Hashimoto, Kentaro, Saito, Bunnai, Miyamoto, Naoki, Oguro, Yuya, Tomita, Daisuke, Shiokawa, Zenyu, Asano, Moriteru, Kakei, Hiroyuki, Taya, Naohiro, Kawasaki, Masanori, Sumi, Hiroyuki, Yabuki, Masato, Iwai, Kenichi, Yoshida, Sei, Yoshimatsu, Mie, Aoyama, Kazunobu, Kosugi, Yohei, Kojima, Takashi, Morishita, Nao, Dougan, Douglas R, Snell, Gyorgy P, Imamura, Shinichi, Ishikawa, Tomoyasu

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Design, synthesis, and biological activities of novel hexahydropyrazino[1,2-a]indole derivatives as potent inhibitors of apoptosis (IAP) proteins antagonists with improved membrane... von Shiokawa, Zenyu, Hashimoto, Kentaro, Saito, Bunnai, Oguro, Yuya, Sumi, Hiroyuki, Yabuki, Masato, Yoshimatsu, Mie, Kosugi, Yohei, Debori, Yasuyuki, Morishita, Nao, Dougan, Douglas R., Snell, Gyorgy P., Yoshida, Sei, Ishikawa, Tomoyasu

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Identification of Novel, Potent, and Orally Available GCN2 Inhibitors with Type I Half Binding Mode von Fujimoto, Jun, Kurasawa, Osamu, Takagi, Terufumi, Liu, Xin, Banno, Hiroshi, Kojima, Takuto, Asano, Yasutomi, Nakamura, Akito, Nambu, Tadahiro, Hata, Akito, Ishii, Tsuyoshi, Sameshima, Tomoya, Debori, Yasuyuki, Miyamoto, Maki, Klein, Michael G, Tjhen, Richard, Sang, Bi-Ching, Levin, Irena, Lane, Scott Weston, Snell, Gyorgy P, Li, Ke, Kefala, Georgia, Hoffman, Isaac D, Ding, Steve C, Cary, Douglas R, Mizojiri, Ryo

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Structural and Kinetic Analysis of the Substrate Specificity of Human Fibroblast Activation Protein α von Aertgeerts, Kathleen, Levin, Irena, Shi, Lihong, Snell, Gyorgy P., Jennings, Andy, Prasad, G. Sridhar, Zhang, Yanming, Kraus, Michelle L., Salakian, Shant, Sridhar, Vandana, Wijnands, Robert, Tennant, Mike G.

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Design, synthesis and structure–activity relationships of 1,3,4-oxadiazole derivatives as novel inhibitors of glycogen synthase kinase-3β von Saitoh, Morihisa, Kunitomo, Jun, Kimura, Eiji, Hayase, Yoji, Kobayashi, Hiromi, Uchiyama, Noriko, Kawamoto, Tomohiro, Tanaka, Toshimasa, Mol, Clifford D., Dougan, Douglas R., Textor, Garret S., Snell, Gyorgy P., Itoh, Fumio

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A new class of non-thiazolidinedione, non-carboxylic-acid-based highly selective peroxisome proliferator-activated receptor (PPAR) γ agonists: Design and synthesis of benzylpyrazol... von Rikimaru, Kentaro, Wakabayashi, Takeshi, Abe, Hidenori, Imoto, Hiroshi, Maekawa, Tsuyoshi, Ujikawa, Osamu, Murase, Katsuhito, Matsuo, Takanori, Matsumoto, Mitsuharu, Nomura, Chisako, Tsuge, Hiroko, Arimura, Naoto, Kawakami, Kazutoshi, Sakamoto, Junichi, Funami, Miyuki, Mol, Clifford D., Snell, Gyorgy P., Bragstad, Kenneth A., Sang, Bi-Ching, Dougan, Douglas R., Tanaka, Toshimasa, Katayama, Nozomi, Horiguchi, Yoshiaki, Momose, Yu

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An optimization-based design approach for a novel self-adjuster using shear thickening fluid von Nagy-György, P., Bene, J. G., Hős, C. J.

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Structure–activity relationships and key structural feature of pyridyloxybenzene-acylsulfonamides as new, potent, and selective peroxisome proliferator-activated receptor (PPAR) γ... von Rikimaru, Kentaro, Wakabayashi, Takeshi, Abe, Hidenori, Tawaraishi, Taisuke, Imoto, Hiroshi, Yonemori, Jinichi, Hirose, Hideki, Murase, Katsuhito, Matsuo, Takanori, Matsumoto, Mitsuharu, Nomura, Chisako, Tsuge, Hiroko, Arimura, Naoto, Kawakami, Kazutoshi, Sakamoto, Junichi, Funami, Miyuki, Mol, Clifford D., Snell, Gyorgy P., Bragstad, Kenneth A., Sang, Bi-Ching, Dougan, Douglas R., Tanaka, Toshimasa, Katayama, Nozomi, Horiguchi, Yoshiaki, Momose, Yu

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Accommodating Fabrication Defects on Floquet Codes with Minimal Hardware Requirements von Campbell McLauchlan, György P. Gehér, Alexandra E. Moylett

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Compilation of a simple chemistry application to quantum error correction primitives von Blunt, Nick S., Gehér, György P., Moylett, Alexandra E.

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First Indication of Solar ^{8}B Neutrinos via Coherent Elastic Neutrino-Nucleus Scattering with XENONnT von Aprile, E, Aalbers, J, Abe, K, Ahmed Maouloud, S, Althueser, L, Andrieu, B, Angelino, E, Antón Martin, D, Arneodo, F, Baudis, L, Bazyk, M, Bellagamba, L, Biondi, R, Bismark, A, Boese, K, Brown, A, Bruno, G, Budnik, R, Cai, C, Capelli, C, Cardoso, J M R, Cimental Chávez, A P, Colijn, A P, Conrad, J, Cuenca-García, J J, D'Andrea, V, Daniel Garcia, L C, Decowski, M P, Deisting, A, Di Donato, C, Di Gangi, P, Diglio, S, Eitel, K, Elykov, A, Ferella, A D, Ferrari, C, Fischer, H, Flehmke, T, Flierman, M, Fulgione, W, Fuselli, C, Gaemers, P, Gaior, R, Galloway, M, Gao, F, Ghosh, S, Giacomobono, R, Glade-Beucke, R, Grandi, L, Grigat, J, Guan, H, Guida, M, Gyorgy, P, Hammann, R, Higuera, A, Hils, C, Hoetzsch, L, Hood, N F, Iacovacci, M, Itow, Y, Jakob, J, Joerg, F, Kaminaga, Y, Kara, M, Kavrigin, P, Kazama, S, Kobayashi, M, Koke, D, Kopec, A, Kuger, F, Landsman, H, Lang, R F, Levinson, L, Li, I, Li, S, Liang, S, Lin, Y-T, Lindemann, S, Lindner, M, Liu, K, Liu, M, Loizeau, J, Lombardi, F, Long, J, Lopes, J A M, Luce, T, Ma, Y, Macolino, C, Mahlstedt, J, Mancuso, A, Manenti, L, Marignetti, F, Marrodán Undagoitia, T, Martens, K, Masbou, J, Masson, E, Mastroianni, S, Melchiorre, A, Merz, J, Messina, M

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Error-corrected Hadamard gate simulated at the circuit level von Gehér, György P., McLauchlan, Campbell, Campbell, Earl T., Moylett, Alexandra E., Crawford, Ophelia

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First Indication of Solar B 8 Neutrinos via Coherent Elastic Neutrino-Nucleus Scattering with XENONnT von Aprile, E., Aalbers, J., Abe, K., Ahmed Maouloud, S., Althueser, L., Andrieu, B., Angelino, E., Antón Martin, D., Arneodo, F., Baudis, L., Bazyk, M., Bellagamba, L., Biondi, R., Bismark, A., Boese, K., Brown, A., Bruno, G., Budnik, R., Cai, C., Capelli, C., Cardoso, J. M. R., Cimental Chávez, A. P., Colijn, A. P., Conrad, J., Cuenca-García, J. J., D’Andrea, V., Daniel Garcia, L. C., Decowski, M. P., Deisting, A., Di Donato, C., Di Gangi, P., Diglio, S., Eitel, K., Elykov, A., Ferella, A. D., Ferrari, C., Fischer, H., Flehmke, T., Flierman, M., Fulgione, W., Fuselli, C., Gaemers, P., Gaior, R., Galloway, M., Gao, F., Ghosh, S., Giacomobono, R., Glade-Beucke, R., Grandi, L., Grigat, J., Guan, H., Guida, M., Gyorgy, P., Hammann, R., Higuera, A., Hils, C., Hoetzsch, L., Hood, N. F., Iacovacci, M., Itow, Y., Jakob, J., Joerg, F., Kaminaga, Y., Kara, M., Kavrigin, P., Kazama, S., Kobayashi, M., Koke, D., Kopec, A., Kuger, F., Landsman, H., Lang, R. F., Levinson, L., Li, I., Li, S., Liang, S., Lin, Y.-T., Lindemann, S., Lindner, M., Liu, K., Liu, M., Loizeau, J., Lombardi, F., Long, J., Lopes, J. A. M., Luce, T., Ma, Y., Macolino, C., Mahlstedt, J., Mancuso, A., Manenti, L., Marignetti, F., Marrodán Undagoitia, T., Martens, K., Masbou, J., Masson, E., Mastroianni, S., Melchiorre, A., Merz, J., Messina, M.

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Next-Generation Sequencing–Based Genomic Profiling of Children with Acute Myeloid Leukemia von Krizsán, Szilvia, Péterffy, Borbála, Egyed, Bálint, Nagy, Tibor, Sebestyén, Endre, Hegyi, Lajos László, Jakab, Zsuzsanna, Erdélyi, Dániel J., Müller, Judit, Péter, György, Csanádi, Krisztina, Kállay, Krisztián, Kriván, Gergely, Barna, Gábor, Bedics, Gábor, Haltrich, Irén, Ottóffy, Gábor, Csernus, Katalin, Vojcek, Ágnes, Tiszlavicz, Lilla Györgyi, Gábor, Krisztina Mita, Kelemen, Ágnes, Hauser, Péter, Gaál, Zsuzsanna, Szegedi, István, Ujfalusi, Anikó, Kajtár, Béla, Kiss, Csongor, Matolcsy, András, Tímár, Botond, Kovács, Gábor, Alpár, Donát, Bödör, Csaba

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Conformational Flexibility in Crystal Structures of Human 11β-Hydroxysteroid Dehydrogenase Type I Provide Insights into Glucocorticoid Interconversion and Enzyme Regulation von Hosfield, David J., Wu, Yiqin, Skene, Robert J., Hilgers, Mark, Jennings, Andy, Snell, Gyorgy P., Aertgeerts, Kathleen

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Tangling schedules eases hardware connectivity requirements for quantum error correction von Geher, Gyorgy P, Crawford, Ophelia, Campbell, Earl T

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