In Vitro Study of Biological Activity of Tanacetum vulgare Extracts von Babich, Olga, Larina, Viktoria, Krol, Olesia, Ulrikh, Elena, Sukhikh, Stanislav, Gureev, Maxim A, Prosekov, Alexander, Ivanova, Svetlana

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π-π Noncovalent Interaction Involving 1,2,4- and 1,3,4-Oxadiazole Systems: The Combined Experimental, Theoretical, and Database Study von Baykov, Sergey V, Mikherdov, Alexander S, Novikov, Alexander S, Geyl, Kirill K, Tarasenko, Marina V, Gureev, Maxim A, Boyarskiy, Vadim P

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Dual PTP1B/TC-PTP Inhibitors: Biological Evaluation of 3-(Hydroxymethyl)cinnoline-4( 1H )-Ones von Derkach, Kira V, Gureev, Maxim A, Babushkina, Anastasia A, Mikhaylov, Vladimir N, Zakharova, Irina O, Bakhtyukov, Andrey A, Sorokoumov, Viktor N, Novikov, Alexander S, Krasavin, Mikhail, Shpakov, Alexander O, Balova, Irina A

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Functionalized 10-Membered Aza- and Oxaenediynes through the Nicholas Reaction von Danilkina, Natalia A, Khmelevskaya, Ekaterina A, Lyapunova, Anna G, D’yachenko, Alexander S, Bunev, Alexander S, Gasanov, Rovshan E, Gureev, Maxim A, Balova, Irina A

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Novel [1,2,4]triazolo[3,4- b ][1,3,4]thiadiazine and [1,2,4]triazolo[3,4- b ][1,3,4]thiadiazepine Derivatives: Synthesis, Anti-Viral In Vitro Study and Target Validation Activity von Khramchikhin, Andrey V, Skryl'nikova, Mariya A, Esaulkova, Iana L, Sinegubova, Ekaterina O, Zarubaev, Vladimir V, Gureev, Maxim A, Puzyk, Aleksandra M, Ostrovskii, Vladimir A

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5-Nitrofuran-Tagged Oxazolyl Pyrazolopiperidines: Synthesis and Activity against ESKAPE Pathogens von Rogacheva, Elizaveta, Kraeva, Lyudmila, Lukin, Alexey, Vinogradova, Lyubov, Komarova, Kristina, Chudinov, Mikhail, Gureev, Maxim, Chupakhin, Evgeny

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Naphthyl-Substituted Indole and Pyrrole Carboxylic Acids as Effective Antibiotic Potentiators—Inhibitors of Bacterial Cystathionine γ-Lyase von Kuzovlev, Andrey S, Zybalov, Mikhail D, Golovin, Andrey V, Gureev, Maxim A, Kasatkina, Mariia A, Biryukov, Mikhail V, Belik, Albina R, Silonov, Sergey A, Yunin, Maxim A, Zigangirova, Nailya A, Reshetnikov, Vasiliy V, Isakova, Yulia E, Porozov, Yuri B, Ivanov, Roman A

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Molecular Periphery Design Allows Control of the New Nitrofurans Antimicrobial Selectivity von Vinogradova, Lyubov, Lukin, Alexey, Komarova, Kristina, Zhuravlev, Maxim, Fadeev, Artem, Chudinov, Mikhail, Rogacheva, Elizaveta, Kraeva, Lyudmila, Gureev, Maxim, Porozov, Yuri, Dogonadze, Marine, Vinogradova, Tatiana

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The Nitrofuran-Warhead-Equipped Spirocyclic Azetidines Show Excellent Activity against Mycobacterium tuberculosis von Komarova, Kristina, Vinogradova, Lyubov, Lukin, Alexey, Zhuravlev, Maxim, Deniskin, Dmitry, Chudinov, Mikhail, Gureev, Maxim, Dogonadze, Marine, Zabolotnykh, Natalia, Vinogradova, Tatiana, Lavrova, Anastasia, Yablonskiy, Petr

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Novel 1,2,4-Triazole- and Tetrazole-Containing 4H-Thiopyrano[2,3-b]quinolines: Synthesis Based on the Thio-Michael/aza-Morita–Baylis–Hillman Tandem Reaction and Investigation of An... von Khramchikhin, Andrey V., Skryl’nikova, Mariya A., Gureev, Maxim A., Zarubaev, Vladimir V., Esaulkova, Iana L., Ilyina, Polina A., Mammeri, Oussama Abdelhamid, Spiridonova, Dar’ya V., Porozov, Yuri B., Ostrovskii, Vladimir A.

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Simulation of MDM2 N-terminal domain conformational lability in the presence of imidazoline based inhibitors of MDM2-p53 protein–protein interaction von Gureev, Maxim, Novikova, Daria, Grigoreva, Tatyana, Vorona, Svetlana, Garabadzhiu, Alexander, Tribulovich, Vyacheslav

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Comparative Study of the Steroidogenic Effects of Human Chorionic Gonadotropin and Thieno[2,3-D]pyrimidine-Based Allosteric Agonist of Luteinizing Hormone Receptor in Young Adult,... von Bakhtyukov, Andrey A, Derkach, Kira V, Gureev, Maxim A, Dar'in, Dmitry V, Sorokoumov, Viktor N, Romanova, Irina V, Morina, Irina Yu, Stepochkina, Anna M, Shpakov, Alexander O

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Borneol Ester Derivatives as Entry Inhibitors of a Wide Spectrum of SARS-CoV-2 Viruses von Yarovaya, Olga I, Shcherbakov, Dmitriy N, Borisevich, Sophia S, Sokolova, Anastasiya S, Gureev, Maxim A, Khamitov, Edward M, Rudometova, Nadezda B, Zybkina, Anastasiya V, Mordvinova, Ekaterina D, Zaykovskaya, Anna V, Rogachev, Artem D, Pyankov, Oleg V, Maksyutov, Rinat A, Salakhutdinov, Nariman F

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5-(Sulfamoyl)thien-2-yl 1,3-oxazole inhibitors of carbonic anhydrase II with hydrophilic periphery von Kalinin, Stanislav, Kovalenko, Alexander, Valtari, Annika, Nocentini, Alessio, Gureev, Maxim, Urtti, Arto, Korsakov, Mikhail, Supuran, Claudiu T, Krasavin, Mikhail

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Enhanced electromechanical response of ferroelectrics due to charged domain walls von Sluka, Tomas, Tagantsev, Alexander K., Damjanovic, Dragan, Gureev, Maxim, Setter, Nava

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The Potential of Usnic-Acid-Based Thiazolo-Thiophenes as Inhibitors of the Main Protease of SARS-CoV-2 Viruses von Yarovaya, Olga I, Filimonov, Aleksandr S, Baev, Dmitriy S, Borisevich, Sophia S, Zaykovskaya, Anna V, Chirkova, Varvara Yu, Marenina, Mariya K, Meshkova, Yulia V, Belenkaya, Svetlana V, Shcherbakov, Dmitriy N, Gureev, Maxim A, Luzina, Olga A, Pyankov, Oleg V, Salakhutdinov, Nariman F, Khvostov, Mikhail V

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Simulation of Molecular Dynamics of SARS-CoV-2 S-Protein in the Presence of Multiple Arbidol Molecules: Interactions and Binding Mode Insights von Borisevich, Sophia S, Khamitov, Edward M, Gureev, Maxim A, Yarovaya, Olga I, Rudometova, Nadezhda B, Zybkina, Anastasiya V, Mordvinova, Ekaterina D, Shcherbakov, Dmitriy N, Maksyutov, Rinat A, Salakhutdinov, Nariman F

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Three-component Castagnoli-Cushman reaction with ammonium acetate delivers 2-unsubstituted isoquinol-1-ones as potent inhibitors of poly(ADP-ribose) polymerase (PARP) von Safrygin, Alexander, Zhmurov, Petr, Dar'in, Dmitry, Silonov, Sergey, Kasatkina, Mariia, Zonis, Yulia, Gureev, Maxim, Krasavin, Mikhail

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Proapoptotic modification of substituted isoindolinones as MDM2-p53 inhibitors von Grigoreva, Tatyana A., Novikova, Daria S., Petukhov, Alexey V., Gureev, Maxim A., Garabadzhiu, Alexander V., Melino, Gerry, Barlev, Nickolai A., Tribulovich, Vyacheslav G.

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The synthesis of 1-oxa-9-azaspiro[5.5]undecane derivatives and optimization of antituberculosis activity thereof von Komarova, Kristina Yu, Lukin, Alexey Yu, Vinogradova, Lyubov V., Zhuravlev, Maxim E., Dogonadze, Marine Z., Vinogradova, Tatiana I., Gureev, Maxim A., Chudinov, Mikhail V., Dar’in, Dmitry V.

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