Naphthol derivatives as TRPV1 inhibitors for the treatment of urinary incontinence von Urbahns, Klaus, Yura, Takeshi, Mogi, Muneto, Tajimi, Masaomi, Fujishima, Hiroshi, Masuda, Tsutomu, Yoshida, Nagahiro, Moriwaki, Toshiya, Lowinger, Timothy B., Meier, Heinrich, Chan, Fiona, Madge, David, Gupta, Jang B.

Volltext

Tetrahydro-naphthols as orally available TRPV1 inhibitors von Urbahns, Klaus, Yura, Takeshi, Gupta, Jang B., Tajimi, Masaomi, Fujishima, Hiroshi, Masuda, Tsutomu, Yamamoto, Noriyuki, Ikegami, Yuka, Marumo, Makiko, Yasoshima, Kayo, Yoshida, Nagahiro, Moriwaki, Toshiya, Madge, David, Chan, Fiona, Mogi, Muneto

Volltext

Functional role of prostacyclin receptor in rat dorsal root ganglion neurons von Nakae, Koichi, Hayashi, Fumihiko, Hayashi, Mayumi, Yamamoto, Noriyuki, Iino, Takashi, Yoshikawa, Satoru, Gupta, Jang

Volltext

Synthesis and optimization of novel and selective muscarinic M3 receptor antagonists von KUMAR, Naresh, KAUR, Kirandeep, PALLE, Venkata P, CLIFLE, Ian A, AERON, Shelly, DHARMARAJAN, Sankaranarayanan, SILAMKOTI, Arun D. V, MEHTA, Anita, GUPTA, Suman, CHUGH, Anita, GUPTA, Jang B, SALMAN, Mohammad

Volltext

Design, synthesis and activity of novel derivatives of Oxybutynin and Tolterodine von Kaur, Kirandeep, Aeron, Shelly, Bruhaspathy, Miriyala, Shetty, Shankar J., Gupta, Suman, Hegde, Laxminarayan H., Silamkoti, Arun D.V., Mehta, Anita, Chugh, Anita, Gupta, Jang B., Sarma, P.K.S., Kumar, Naresh

Volltext

Benzimidazole derivatives as novel nonpeptide luteinizing hormone-releasing hormone (LHRH) antagonists. Part 2: Benzimidazole-5-sulfonamides von Li, Yingfu, Kataoka, Mikayo, Tatsuta, Miyuki, Yasoshima, Kayo, Yura, Takeshi, Urbahns, Klaus, Kiba, Atsushi, Yamamoto, Noriyuki, Gupta, Jang B., Hashimoto, Kentaro

Volltext

Benzimidazole derivatives as novel nonpeptide luteinizing hormone-releasing hormone (LHRH) antagonists. Part 1: Benzimidazole-5-sulfonamides von Hashimoto, Kentaro, Tatsuta, Miyuki, Kataoka, Mikayo, Yasoshima, Kayo, Shogase, Yuka, Shimazaki, Makoto, Yura, Takeshi, Li, Yingfu, Yamamoto, Noriyuki, Gupta, Jang B., Urbahns, Klaus

Volltext

Endothelin-receptor antagonists: current and future perspectives von Ray, Abhijit, Hegde, Laxminarayan G, Chugh, Anita, Gupta, Jang B

Volltext

Abstract 2643: Discovery and characterization of a selective TrkA inhibitor for the treatment of TrkA-driven cancers von Tirunagaru, Vijaya G., Nagaswamy, Kumaragurubaran, Mitra, Sayan, Maddi, Srinivas, Adluri, Ram Sudheer, Joshi, Hemant, Gupta, Jang B.

Volltext

Abstract 373: Discovery of selective PI3Kb inhibitors for PTEN-deficient tumors and other indications von Chowdhury, Arnab R., Athisayamani, Jeyaraj D., Mitra, Sayan, Maddi, Srinivas, Adluri, Ram Sudheer, Bethi, Sridhar R., Joshi, Hemant, Tirunagaru, Vijaya G., Gupta, Jang B.

Volltext

Relaxant Effect of Oxygen Free Radicals on Rabbit Tracheal Smooth Muscle von Prasad, Kailash, Gupta, Jang B.

Volltext

Benzimidazole-5-sulfonamides as Novel Nonpeptide Luteinizing Hormone Releasing Hormone (LHRH) Antagonists: Minimization of Mechanism-Based CYP3A4 Inhibition von Hashimoto, Kentaro, Kataoka, Mikayo, Tatsuta, Miyuki, Yasoshima, Kayo, Yamamoto, Mako, Yura, Takeshi, Yamamoto, Noriyuki, Urbahns, Klaus, Gupta, Jang Bahadur, Li, Yingfu

Volltext

Abstract 1661: Development of lipid-based nanosuspension formulation of first-in-class PLK2 inhibitor GBO-006 to treat triple-negative breast cancer von Tirunagaru, Vijaya G., Roy Chowdhury, Arnab, Duraiswamy, Jeyaraj Athisayamani, Maddi, Srinivasa Rao, Mitra, Sayan, Deb, Chandra, Adluri, Ram Sudheer, Gupta, Jang B.

Volltext

Preclinical formulation for the pharmacokinetics and efficacy of GBO-006, a selective polo like kinase 2 (PLK2) inhibitor for the treatment of triple negative breast cancer von Maddi, Srinivas, Akkireddy, Ravi, Lenkalapelly, Srinivas, Srivastava, Pratima, Boruwa, Joshodeep, Deb, Chandra, Chowdhury, Arnab Roy, Jeyaraj, Duraiswamy A., Reddy, Ramana, Reddy, Premkumar, Maniar, Manoj, Bansal, Sachin, Gupta, Jang B.

Volltext

Benzimidazoles as non-peptide luteinizing hormone-releasing hormone (LHRH) antagonists. Part 3: Discovery of 1-(1 H-benzimidazol-5-yl)-3- tert-butylurea derivatives von Tatsuta, Miyuki, Kataoka, Mikayo, Yasoshima, Kayo, Sakakibara, Sachiko, Shogase, Yuka, Shimazaki, Makoto, Yura, Takeshi, Li, Yingfu, Yamamoto, Noriyuki, Gupta, Jang, Urbahns, Klaus

Volltext

Effects of platelet-activating factor on cardiovascular function, oxygen free radical status, and blood chemistry von Prasad, Kailash, Gupta, Jang B., Kalra, Jawahar

Volltext

Synthesis and optimization of novel and selective muscarinic M 3 receptor antagonists von Kumar, Naresh, Kaur, Kirandeep, Aeron, Shelly, Dharmarajan, Sankaranarayanan, Silamkoti, Arun D.V., Mehta, Anita, Gupta, Suman, Chugh, Anita, Gupta, Jang B., Salman, Mohammad, Palle, Venkata P., Cliffe, Ian A.

Volltext

Synthesis and optimization of novel and selective muscarinic M(3) receptor antagonists von Kumar, Naresh, Kaur, Kirandeep, Aeron, Shelly, Dharmarajan, Sankaranarayanan, Silamkoti, Arun D V, Mehta, Anita, Gupta, Suman, Chugh, Anita, Gupta, Jang B, Salman, Mohammad, Palle, Venkata P, Cliffe, Ian A

Volltext

Oxidative Stress as a Mechanism of Cardiac Failure in Chronic Volume Overload in Canine Model von Prasad, Kailash, Gupta, Jang B., Kalra, Jawahar, Lee, P., Mantha, Subrahmanyam V., Bharadwaj, Baikunth

Volltext

Corrigendum to “Benzimidazoles as non-peptide luteinizing hormone-releasing hormone (LHRH) antagonists. Part 3: Discovery of 1-(1 H-benzimidazol-5-yl)-3- tert-butylurea derivatives... von Tatsuta, Miyuki, Kataoka, Mikayo, Yasoshima, Kayo, Sakakibara, Sachiko, Shogase, Yaka, Shimazaki, Makoto, Yura, Takeshi, Li, Yingfu, Yamamoto, Noriyuki, Gupta, Jang, Urbahns, Klaus

Volltext