From Inhibition to Degradation: Targeting the Antiapoptotic Protein Myeloid Cell Leukemia 1 (MCL1) von Papatzimas, James W, Gorobets, Evgueni, Maity, Ranjan, Muniyat, Mir Ishruna, MacCallum, Justin L, Neri, Paola, Bahlis, Nizar J, Derksen, Darren J

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Rapid synthesis of pomalidomide-conjugates for the development of protein degrader libraries von Brownsey, Duncan K, Rowley, Ben C, Gorobets, Evgueni, Gelfand, Benjamin S, Derksen, Darren J

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Beyond geminal diesters: increasing the scope of metal-mediated vinylcyclopropane annulations while decreasing pre-activation von Brownsey, Duncan K, Gorobets, Evgueni, Derksen, Darren J

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Pannexin-1 channel inhibition alleviates opioid withdrawal in rodents by modulating locus coeruleus to spinal cord circuitry von Kwok, Charlie H. T., Harding, Erika K., Burma, Nicole E., Markovic, Tamara, Massaly, Nicolas, van den Hoogen, Nynke J., Stokes-Heck, Sierra, Gambeta, Eder, Komarek, Kristina, Yoon, Hye Jean, Navis, Kathleen E., McAllister, Brendan B., Canet-Pons, Julia, Fan, Churmy, Dalgarno, Rebecca, Gorobets, Evgueni, Papatzimas, James W., Zhang, Zizhen, Kohro, Yuta, Anderson, Connor L., Thompson, Roger J., Derksen, Darren J., Morón, Jose A., Zamponi, Gerald W., Trang, Tuan

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Generation of Benzyne Species from Diphenylphosphoryl Derivatives: Simultaneous Exchange of Three Functional Groups von Gorobets, Evgueni, Parvez, Masood, Derksen, Darren J., Keay, Brian A.

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Natural-Product-Derived Transient Receptor Potential Melastatin 8 (TRPM8) Channel Modulators von LeGay, Christina M, Gorobets, Evgueni, Iftinca, Mircea, Ramachandran, Rithwik, Altier, Christophe, Derksen, Darren J

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Metformin Prevents Hyperglycemia-Associated, Oxidative Stress-Induced Vascular Endothelial Dysfunction: Essential Role for the Orphan Nuclear Receptor Human Nuclear Receptor 4A1 (N... von Venu, Vivek Krishna Pulakazhi, Saifeddine, Mahmoud, Mihara, Koichiro, Faiza, Muniba, Gorobets, Evgueni, Flewelling, Andrew J., Derksen, Darren J., Hirota, Simon A., Marei, Isra, Al-Majid, Dana, Motahhary, Majid, Ding, Hong, Triggle, Chris R., Hollenberg, Morley D.

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Leveraging Pyrazolium Ylide Reactivity to Access Indolizine and 1,2‐Dihydropyrimidine Derivatives von Tran, Ricky, Brownsey, Duncan K., O'Sullivan, Leonie, Brandow, Connor M. J., Chang, Emily S., Zhou, Wen, Patel, Ketul V., Gorobets, Evgueni, Derksen, Darren J.

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Regioselective Synthesis of C3-Hydroxyarylated Pyrazoles von O'Sullivan, Leonie, Patel, Ketul V, Rowley, Ben C, Brownsey, Duncan K, Gorobets, Evgueni, Gelfand, Benjamin S, Van Humbeck, Jeffrey F, Derksen, Darren J

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A vinylogous Norrish reaction as a strategy for light-mediated ring expansion von Gorobets, Evgueni, Papatzimas, James W, Dourado, Jorge, Yousefalizadeh, Goonay, Lee, JinGyu, Brownsey, Duncan K, Stamplecoskie, Kevin, Davis, Rebecca, Derksen, Darren J

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Utilising the intrinsic fluorescence of pomalidomide for imaging applications von Brownsey, Duncan K, Gafuik, Christopher J, Kim, Dae-Sun, O'Sullivan, Leonie, Gorobets, Evgueni, Krukowski, Samuel, Turk, Madison, Jenne, Craig N, Mahoney, Douglas J, Derksen, Darren J

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Divergent Photocyclization/1,4-Sigmatropic Rearrangements for the Synthesis of Sesquiterpenoid Derivatives von Gorobets, Evgueni, Wong, Norman E, Paton, Robert S, Derksen, Darren J

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Thiaporphyrin-mediated photocatalysis using red light von Lee, JinGyu, Papatzimas, James W, Bromby, Ashley D, Gorobets, Evgueni, Derksen, Darren J

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Identification of ligand linkage vectors for the development of p300/CBP degraders von Brownsey, Duncan K, Rowley, Ben C, Gorobets, Evgueni, Mihara, Koichiro, Maity, Ranjan, Papatzimas, James W, Gelfand, Benjamin S, Hollenberg, Morley D, Bahlis, Nizar J, Derksen, Darren J

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Avoiding the classical resolution during the synthesis of MeO-BIPHEP and 3,3′-disubstituted derivatives von Gorobets, Evgueni, Wheatley, Bronwen M.M., Hopkins, J. Matthew, McDonald, Robert, Keay, Brian A.

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Synthesis, resolution and applications of 3,3′-bis(RO)-MeO-BIPHEP derivatives von Gorobets, Evgueni, Sun, Guang-Ri, Wheatley, Bronwen M.M., Parvez, Masood, Keay, Brian A.

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Enantioselective Total Synthesis of a trans-Hydrindane Rings/Side-Chain Building-Block of Vitamin D − Asymmetric Induction in an Acid-Catalyzed Conjugate-Addition Reaction von Gorobets, Evgueni, Stepanenko, Viatcheslav, Wicha, Jerzy

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Applications of 3,3′-Disubstituted BINAP Derivatives in Inter- and Intramolecular Heck/Mizoroki Reactions von Hopkins, J. Matthew, Gorobets, Evgueni, Wheatley, Bronwen M., Parvez, Masood, Keay, Brian A.

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Synthesis of tacamonine von Ho, Tse-Lok, Gorobets, Evgueni

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SULFAMOYL BENZENE DERIVATIVES AND USES THEREOF von TRANG, Tuan, NAVIS, Kathleen, PAPATZIMAS, James, DERKSEN, Darren Jason, GOROBETS, Evgueni

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