Synthesis and pharmacological evaluation of thieno[2,3- b]pyridine derivatives as novel c-Src inhibitors von Pevet, Isabelle, Brulé, Cédric, Tizot, André, Gohier, Arnaud, Cruzalegui, Francisco, Boutin, Jean A., Goldstein, Solo

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Productive Syntheses of Privileged Scaffolds Inspired by the Recognition of a Diels–Alder Pattern Common to Three Classes of Natural Products von Badarau, Eduard, Reddy, K. Harsha Vardhan, Loudet, Aurore, Simon, Charles, Trembleau, Laurent, Claerhout, Stijn, Pair, Etienne, Massip, Stéphane, Breton, Philippe, Lesur, Brigitte, Goldstein, Solo, Fourquez, Jean‐Marie, Henlin, Jean Michel, Ghosez, Léon

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Comparison of the pharmacological profile of an olivacine derivative and a potential prodrug von KRAUS-BERTHIER, Laurence, GUILBAUD, Nicolas, LEONCE, Stéphane, PARKER, Tracy, GENISSEL, Patrick, GUILLONNEAU, Claude, GOLDSTEIN, Solo, ATASSI, Ghanem, PIERRE, Alain

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S 50131 and S 51434, two novel small molecule glucokinase activators, lack chronic efficacy despite potent acute antihyperglycaemic activity in diabetic mice von De Ceuninck, Frédéric, Kargar, Catherine, Charton, Yves, Goldstein, Solo, Perron‐Sierra, Françoise, Ilic, Catherine, Caliez, Audrey, Rolin, Jean‐Olivier, Sadlo, Marjorie, Harley, Elizabeth, Vinson, Cédric, Ktorza, Alain

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Preparation and affinity profile of novel nicotinic ligands von Charton, Yves, Guillonneau, Claude, Lockhart, Brian, Lestage, Pierre, Goldstein, Solo

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Synthesis, Structure, and Neuroprotective Properties of Novel Imidazolyl Nitrones von Dhainaut, Alain, Tizot, André, Raimbaud, Eric, Lockhart, Brian, Lestage, Pierre, Goldstein, Solo

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Conformational analysis of pseudo-peptides: The case of FK888, a potent and selective substance P receptor antagonist von Moureau, Florence, Neuwels, Michel, Dogimont, Charles, Goldstein, Solo, Massingham, R.

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Cytotoxic and antitumoral properties in a series of new, ring D modified, olivacine analogues von Guillonneau, Claude, Nault, Annette, Raimbaud, Eric, Léonce, Stéphane, Kraus-Berthier, Laurence, Pierré, Alain, Goldstein, Solo

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Characterization of phospholipase C activity at h5-HT2C compared with h5-HT2B receptors: influence of novel ligands upon membrane-bound levels of [3H]phosphatidylinositols von Cussac, Didier, Newman-Tancredi, Adrian, Quentric, Yann, Carpentier, Nathalie, Poissonnet, Guillaume, Parmentier, Jean-Gilles, Goldstein, Solo, Millan, Mark J

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In vivo neuroprotective effects of the novel imidazolyl nitrone free-radical scavenger (Z)-α-[2-thiazol-2-ylimidazol-4-yl]-N-tert-butylnitrone (S34176) von LOCKHART, Brian, ROGER, Anita, BONHOMME, Norbert, GOLDSTEIN, Solo, LESTAGE, Pierre

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In vivo neuroprotective effects of the novel imidazolyl nitrone free-radical scavenger ( Z)-α-[2-thiazol-2-yl)imidazol-4-yl]- N- tert-butylnitrone (S34176 von Lockhart, Brian, Roger, Anita, Bonhomme, Norbert, Goldstein, Solo, Lestage, Pierre

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IAM retention and blood brain barrier penetration von Ducarme, André, Neuwels, Michel, Goldstein, Solo, Massingham, Roy

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Radical trapping properties of imidazolyl nitrones von Reybier, Karine, Boyer, Jeremie, Farines, Vincent, Camus, Fabrice, Souchard, Jean-Pierre, Monje, Marie-Carmen, Bernardes-Genisson, Vania, Goldstein, Solo, Nepveu, Francoise

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Stereocontrolled construction of 1,7-dimethyl A.B.C.[6.6.6] tricycles. Part II. Transannular Diels-Alder reaction of 14-membered macrocycles containing cis-dienophiles von Xu, Yao-Chang, Roughton, Andrew L, Soucy, Pierre, Goldstein, Solo, Deslongchamps, Pierre

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Stereocontrolled construction of 1,7-dimethyl A.B.C.[6.6.6] tricycles. Part I. Transannular Diels-Alder reactions of 14-membered macrocycles containing trans-dienophiles von Xu, Yao-Chang, Roughton, Andrew L, Plante, Raymond, Goldstein, Solo, Deslongchamps, Pierre

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Synthesis and pharmacological evaluation of new 1,2-dithiolane based antioxidants von Guillonneau, Claude, Charton, Yves, Ginot, Yves-Michel, Fouquier-d'Hérouël, Marie-Victoire, Bertrand, Marc, Lockhart, Brian, Lestage, Pierre, Goldstein, Solo

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Cyclization of Hydroxyenol Ethers into Spiroacetals. Evidence for the position of the transition state and its implication on the stereoelectronic effects in acetal formation von Pothier, Normand, Goldstein, Solo, Deslongchamps, Pierre

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Characterization of phospholipase C activity at h5-HT 2C compared with h5-HT 2B receptors: influence of novel ligands upon membrane-bound levels of [ 3 H]phosphatidylinositols von Cussac, Didier, Newman-Tancredi, Adrian, Quentric, Yann, Carpentier, Nathalie, Poissonnet, Guillaume, Parmentier, Jean-Gilles, Goldstein, Solo, Millan, Mark

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Jean - Luc Fauchere (1941-2003) von Boutin, Jean A., Henlin, Jean-Michel, Goldstein, Solo, Kucharczyk, Nathalie, Ortuno, Jean-Claude

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NEW POLYSUBSTITUTED PYRIDINYLAMINOALKYLENE- AND PYRIDINYLOXYALKYLENE-CYCLOPROPANAMINE COMPOUNDS,A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM von CHARTON, YVES, LOCKHART, BRIAN, GUILLONNEAU, CLAUDE, LESTAGE, PIERRE, GOLDSTEIN, SOLO

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