Structure Activity of 3-Aryl-1,3-diketo-Containing Compounds as HIV-1 Integrase Inhibitors von Pais, Godwin C. G, Zhang, Xuechun, Marchand, Christophe, Neamati, Nouri, Cowansage, Kiriana, Svarovskaia, Evguenia S, Pathak, Vinay K, Tang, Yun, Nicklaus, Marc, Pommier, Yves, Burke, Terrence R

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Metal-dependent inhibition of HIV-1 integrase by beta-diketo acids and resistance of the soluble double-mutant (F185K/C280S) von Marchand, Christophe, Johnson, Allison A, Karki, Rajeshri G, Pais, Godwin C G, Zhang, Xuechun, Cowansage, Kiriana, Patel, Tapan A, Nicklaus, Marc C, Burke, Jr, Terrence R, Pommier, Yves

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Metal-Dependent Inhibition of HIV-1 Integrase von Neamati, Nouri, Lin, Zhaiwei, Karki, Rajeshri G, Orr, Ann, Cowansage, Kiriana, Strumberg, Dirk, Pais, Godwin C. G, Voigt, Johannes H, Nicklaus, Marc C, Winslow, Heather E, Zhao, He, Turpin, Jim A, Yi, Jizu, Skalka, Anna Marie, Burke, Terrence R, Pommier, Yves

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Azido-Containing Diketo Acid Derivatives Inhibit Human Immunodeficiency Virus Type 1 Integrase In Vivo and Influence the Frequency of Deletions at Two-Long-Terminal-Repeat-Circle J... von Svarovskaia, Evguenia S, Barr, Rebekah, Zhang, Xuechun, Pais, Godwin C G, Marchand, Christophe, Pommier, Yves, Burke, Jr, Terrence R, Pathak, Vinay K

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Exploration of the Activity of 7-Pyrrolidino-8-methoxyisothiazoloquinolones against Methicillin-Resistant Staphylococcus aureus (MRSA) von Kim, Ha Young, Wiles, Jason A, Wang, Qiuping, Pais, Godwin C. G, Lucien, Edlaine, Hashimoto, Akihiro, Nelson, David M, Thanassi, Jane A, Podos, Steven D, Deshpande, Milind, Pucci, Michael J, Bradbury, Barton J

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Integration Requires a Specific Interaction of the Donor DNA Terminal 5′-Cytosine with Glutamine 148 of the HIV-1 Integrase Flexible Loop von Johnson, Allison A., Santos, Webster, Pais, Godwin C.G., Marchand, Christophe, Amin, Ronak, Burke, Terrence R., Verdine, Gregory, Pommier, Yves

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Isothiazoloquinolones with Enhanced Antistaphylococcal Activities against Multidrug-Resistant Strains:  Effects of Structural Modifications at the 6-, 7-, and 8-Positions von Wang, Qiuping, Lucien, Edlaine, Hashimoto, Akihiro, Pais, Godwin C. G., Nelson, David M., Song, Yongsheng, Thanassi, Jane A., Marlor, Christopher W., Thoma, Christy L., Cheng, Jijun, Podos, Steven D., Ou, Yangsi, Deshpande, Milind, Pucci, Michael J., Buechter, Douglas D., Bradbury, Barton J., Wiles, Jason A.

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Efficient Synthesis of the γ-Amino-β-hydroxy Acid Subunit of Hapalosin von Pais, Godwin C. G, Maier, Martin E

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Structural Determinants for HIV-1 Integrase Inhibition by β-Diketo Acids von Marchand, Christophe, Zhang, Xuechun, Pais, Godwin C.G., Cowansage, Kiriana, Neamati, Nouri, Burke, Terrence R., Pommier, Yves

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Azido-Containing aryl β-Diketo acid HIV-1 integrase inhibitors von Zhang, Xuechun, Pais, Godwin C.G, Svarovskaia, Evguenia S, Marchand, Christophe, Johnson, Allison A, Karki, Rajeshri G, Nicklaus, Marc C, Pathak, Vinay K, Pommier, Yves, Burke, Terrence R

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Practical Synthesis and Molecular Structure of a Potent Broad-Spectrum Antibacterial Isothiazoloquinolone von Hashimoto, Akihiro, Pais, Godwin C. G, Wang, Qiuping, Lucien, Edlaine, Incarvito, Christopher D, Deshpande, Milind, Bradbury, Barton J, Wiles, Jason A

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Inhibition of Human Immunodeficiency Virus Type 1 Integration by Diketo Derivatives von PLUYMERS, Wim, PAIS, Godwin, VAN MAELE, Bénédicte, PANNECOUQUE, Christophe, FIKKERT, Valery, BURKE, Terrence R, DE CLERCQ, Erik, WITVROUW, Myriam, NEAMATI, Nouri, DEBYSER, Zeger

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Effect of HIV Integrase Inhibitors on the RAG1/2 Recombinase von Melek, Meni, Jones, Jessica M., O'Dea, Mary H., Pais, Godwin, Burke, Terrence R., Pommier, Yves, Neamati, Nouri, Gellert, Martin

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Total Synthesis of Hapalosin and Two Ring Expanded Analogs von Hermann, Christoph, Pais, Godwin C.G, Geyer, Armin, Kühnert, Sven M, Maier, Martin E

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Asymmetric synthesis of ( S) - Massoialactone von Pais, Godwin C.G., Fernandes, Rodney A., Kumar, Pradeep

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Utilization of a Peptide Lead for the Discovery of a Novel PTP1B-Binding Motif von Gao, Yang, Voigt, Johannes, Zhao, He, Pais, Godwin C. G, Zhang, Xuechun, Wu, Li, Zhang, Zhong-Yin, Burke, Terrence R

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METHODS FOR PREPARING (-)-EPICATECHIN von PAIS, Godwin

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Hydroxy-assisted chemo- and stereo-selective epoxidation catalysed by a titanium silicate molecular sieve (TS-1)/H2O2 system von Kumar, Rajiv, Pais, Godwin C. G., Pandey, Bipin, Kumar, Pradeep

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Preclinical Evaluation of Orally Bioavailable Small-Molecule Inhibitors of Complement Factor D As a Potential Treatment for Paroxysmal Nocturnal Hemoglobinuria von Wiles, Jason, Podos, Steven, Thanassi, Jane, Phadke, Avinash, Gadhachanda, Venkat, Pais, Godwin, Hashimoto, Akihiro, Wang, Qiuping, Chen, Dawei, Wang, Xiangzhu, Agarwal, Atul, Rivera, Jose, Elliot, Michael, Marlor, Christopher, Zhang, Jay, Deshpande, Milind, Huang, Mingjun, Huang, Yongqing

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Novel Small-Molecule Inhibitors Targeting Complement Factor D for Therapy of Paroxysmal Nocturnal Hemoglobinuria von Morgan, B. Paul, Thanassi, Jane, Podos, Steven, Phadke, Avinash, Gadhachanda, Venkat, Pais, Godwin, Hashimoto, Akihiro, Wang, Qiuping, Chen, Dawei, Wang, Xiangzhu, Agarwal, Atul, Deshpande, Milind, Huang, Yongqing, Wiles, Jason, Huang, Mingjun

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