Recent encounters with atropisomerism in drug discovery von Glunz, Peter W.

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P2Y6 receptor potentiates pro-inflammatory responses in macrophages and exhibits differential roles in atherosclerotic lesion development von Garcia, Ricardo A, Yan, Mujing, Search, Debra, Zhang, Rongan, Carson, Nancy L, Ryan, Carol S, Smith-Monroy, Constance, Zheng, Joanna, Chen, Jian, Kong, Yan, Tang, Huaping, Hellings, Samuel E, Wardwell-Swanson, Judith, Dinchuk, Joseph E, Psaltis, George C, Gordon, David A, Glunz, Peter W, Gargalovic, Peter S

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Phthalazinone-based lactams and cyclic ureas as ROCK2 selective inhibitors von Hu, Zilun, Sitkoff, Doree, Glunz, Peter W., Zou, Yan, Wang, Cailan, Muckelbauer, Jodi K., Adam, Leonard P., Wexler, Ruth R., Quan, Mimi L.

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Atropisomer Control in Macrocyclic Factor VIIa Inhibitors von Glunz, Peter W, Mueller, Luciano, Cheney, Daniel L, Ladziata, Vladimir, Zou, Yan, Wurtz, Nicholas R, Wei, Anzhi, Wong, Pancras C, Wexler, Ruth R, Priestley, E. Scott

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Discovery of a phenylpyrazole amide ROCK inhibitor as a tool molecule for in vivo studies von Hu, Zilun, Wang, Cailan, Glunz, Peter W., Li, Julia, Cheadle, Nathan L., Chen, Alice Y., Chen, Xue-Qing, Myers, Joseph E., Guarino, Victor R., Rose, Anne, Sack, John S., Sitkoff, Doree, Taylor, David S., Xu, Songmei, Yan, Chunhong, Zhang, Hongwei, Zhang, Lisa, Hennan, James, Adam, Leonard P., Wexler, Ruth R., Quan, Mimi L.

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Discovery of a Highly Potent, Selective, and Orally Bioavailable Macrocyclic Inhibitor of Blood Coagulation Factor VIIa–Tissue Factor Complex von Zhang, Xiaojun, Glunz, Peter W, Johnson, James A, Jiang, Wen, Jacutin-Porte, Swanee, Ladziata, Vladimir, Zou, Yan, Phillips, Monique S, Wurtz, Nicholas R, Parkhurst, Brandon, Rendina, Alan R, Harper, Timothy M, Cheney, Daniel L, Luettgen, Joseph M, Wong, Pancras C, Seiffert, Dietmar, Wexler, Ruth R, Priestley, E. Scott

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Correction to “Atropisomer Control in Macrocyclic Factor VIIa Inhibitors” von Glunz, Peter W, Mueller, Luciano, Cheney, Daniel L, Ladziata, Vladimir, Zou, Yan, Wurtz, Nicholas R, Wei, Anzhi, Wong, Pancras C, Wexler, Ruth R, Priestley, E. Scott

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Neutral macrocyclic factor VIIa inhibitors von Wurtz, Nicholas R., Parkhurst, Brandon L., DeLucca, Indawati, Glunz, Peter W., Jiang, Wen, Zhang, Xiaojun, Cheney, Daniel L., Bozarth, Jeffrey M., Rendina, Alan R., Wei, Anzhi, Harper, Tim, Luettgen, Joseph M., Wu, Yiming, Wong, Pancras C., Seiffert, Dietmar A., Wexler, Ruth R., Priestley, E. Scott

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Synthesis and P1′ SAR exploration of potent macrocyclic tissue factor-factor VIIa inhibitors von Ladziata, Vladimir (Uladzimir), Glunz, Peter W., Zou, Yan, Zhang, Xiaojun, Jiang, Wen, Jacutin-Porte, Swanee, Cheney, Daniel L., Wei, Anzhi, Luettgen, Joseph M., Harper, Timothy M., Wong, Pancras C., Seiffert, Dietmar, Wexler, Ruth R., Priestley, E. Scott

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On the Power of Chemical Synthesis: Immunological Evaluation of Models for Multiantigenic Carbohydrate-Based Cancer Vaccines von Ragupathi, Govindaswami, Coltart, Don M., Williams, Lawrence J., Koide, Fusataka, Kagan, Ella, Allen, Jennifer, Harris, Christina, Glunz, Peter W., Livingston, Philip O., Danishefsky, Samuel J.

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Design and synthesis of potent, selective phenylimidazole-based FVIIa inhibitors von Glunz, Peter W., Cheng, Xuhong, Cheney, Daniel L., Weigelt, Carolyn A., Wei, Anzhi, Luettgen, Joseph M., Wong, Pancras C., Wexler, Ruth R., Priestley, E. Scott

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Principles of Mucin Architecture:  Structural Studies on Synthetic Glycopeptides Bearing Clustered Mono-, Di-, Tri-, and Hexasaccharide Glycodomains von Coltart, Don M, Royyuru, Ajay K, Williams, Lawrence J, Glunz, Peter W, Sames, Dalibor, Kuduk, Scott D, Schwarz, Jacob B, Chen, Xiao-Tao, Danishefsky, Samuel J, Live, David H

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Nonbenzamidine acylsulfonamide tissue factor–factor VIIa inhibitors von Glunz, Peter W., Zhang, Xiaojun, Zou, Yan, Delucca, Indawati, Nirschl, Alexandra H., Cheng, Xuhong, Weigelt, Carolyn A., Cheney, Daniel L., Wei, Anzhi, Anumula, Rushith, Luettgen, Joseph M., Rendina, Alan R., Harpel, Mark, Luo, Gang, Knabb, Robert, Wong, Pancras C., Wexler, Ruth R., Priestley, E. Scott

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Synthetic and Immunological Studies on Clustered Modes of Mucin-Related Tn and TF O-Linked Antigens:  The Preparation of a Glycopeptide-Based Vaccine for Clinical Trials against Pr... von Kuduk, Scott D, Schwarz, Jacob B, Chen, Xiao-Tao, Glunz, Peter W, Sames, Dalibor, Ragupathi, Govindaswami, Livingston, Philip O, Danishefsky, Samuel J

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Design and synthesis of bicyclic pyrazinone and pyrimidinone amides as potent TF–FVIIa inhibitors von Zhang, Xiaojun, Glunz, Peter W., Jiang, Wen, Schmitt, Aaron, Newman, Makenzie, Barbera, Frank A., Bozarth, Jeffery M., Rendina, Alan R., Wei, Anzhi, Wen, Xiao, Rossi, Karen A., Luettgen, Joseph M., Wong, Pancras C., Knabb, Robert M., Wexler, Ruth R., Scott Priestley, E.

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Design and Synthesis of Phenylpyrrolidine Phenylglycinamides As Highly Potent and Selective TF-FVIIa Inhibitors von Zhang, Xiaojun, Jiang, Wen, Jacutin-Porte, Swanee, Glunz, Peter W, Zou, Yan, Cheng, Xuhong, Nirschl, Alexandra H, Wurtz, Nicholas R, Luettgen, Joseph M, Rendina, Alan R, Luo, Gang, Harper, Timothy M, Wei, Anzhi, Anumula, Rushith, Cheney, Daniel L, Knabb, Robert M, Wong, Pancras C, Wexler, Ruth R, Priestley, E. Scott

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A Broadly Applicable Method for the Efficient Synthesis of α-O-Linked Glycopeptides and Clustered Sialic Acid Residues von Schwarz, Jacob B, Kuduk, Scott D, Chen, Xiao-Tao, Sames, Dalibor, Glunz, Peter W, Danishefsky, Samuel J

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New Chemical Synthesis of the Promising Cancer Chemotherapeutic Agent 12,13-Desoxyepothilone B: Discovery of a Surprising Long-Range Effect on the Diastereoselectivity of an Aldol... von Harris, Christina R, Kuduk, Scott D, Balog, Aaron, Savin, Ken, Glunz, Peter W, Danishefsky, Samuel J

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Design and synthesis of bicyclic pyrimidinone-based HCV NS3 protease inhibitors von Glunz, Peter W, Douty, Brent D, Decicco, Carl P

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A mild and readily scalable procedure for the N-1-difluoromethylation of ethyl 6-((tert-butyldiphenylsilyl)oxy)-1H-indazole-3-carboxylate and its applications to the N-difluorometh... von Hong, Zhenqiu, Hou, Xiaoping, Zhao, Rulin, Li, Jianqing, Pawluczyk, Joseph, Wang, Bei, Kempson, James, Khandelwal, Purnima, Smith, Leon M., Glunz, Peter, Mathur, Arvind

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