Structural basis for PPAR partial or full activation revealed by a novel ligand binding mode von Capelli, Davide, Cerchia, Carmen, Montanari, Roberta, Loiodice, Fulvio, Tortorella, Paolo, Laghezza, Antonio, Cervoni, Laura, Pochetti, Giorgio, Lavecchia, Antonio

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Resveratrol and Its Metabolites Bind to PPARs von Calleri, Enrica, Pochetti, Giorgio, Dossou, Katina S. S., Laghezza, Antonio, Montanari, Roberta, Capelli, Davide, Prada, Ellen, Loiodice, Fulvio, Massolini, Gabriella, Bernier, Michel, Moaddel, Ruin

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PHA-680626 Is an Effective Inhibitor of the Interaction between Aurora-A and N-Myc von Boi, Dalila, Souvalidou, Fani, Capelli, Davide, Polverino, Federica, Marini, Grazia, Montanari, Roberta, Pochetti, Giorgio, Tramonti, Angela, Contestabile, Roberto, Trisciuoglio, Daniela, Carpinelli, Patrizia, Ascanelli, Camilla, Lindon, Catherine, De Leo, Alessandro, Saviano, Michele, Di Santo, Roberto, Costi, Roberta, Guarguaglini, Giulia, Paiardini, Alessandro

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Discovery of Novel Chemical Series of OXA-48 β-Lactamase Inhibitors by High-Throughput Screening von Garofalo, Barbara, Prati, Federica, Buonfiglio, Rosa, Coletta, Isabella, D’Atanasio, Noemi, Molteni, Angela, Carettoni, Daniele, Wanke, Valeria, Pochetti, Giorgio, Montanari, Roberta, Capelli, Davide, Milanese, Claudio, Di Giorgio, Francesco Paolo, Ombrato, Rosella

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Surface Plasmon Resonance as a Tool for Ligand Binding Investigation of Engineered GPR17 Receptor, a G Protein Coupled Receptor Involved in Myelination von Capelli, Davide, Parravicini, Chiara, Pochetti, Giorgio, Montanari, Roberta, Temporini, Caterina, Rabuffetti, Marco, Trincavelli, Maria Letizia, Daniele, Simona, Fumagalli, Marta, Saporiti, Simona, Bonfanti, Elisabetta, Abbracchio, Maria P, Eberini, Ivano, Ceruti, Stefania, Calleri, Enrica, Capaldi, Stefano

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Bone-Seeking Matrix Metalloproteinase Inhibitors for the Treatment of Skeletal Malignancy von Laghezza, Antonio, Piemontese, Luca, Brunetti, Leonardo, Caradonna, Alessia, Agamennone, Mariangela, Di Pizio, Antonella, Pochetti, Giorgio, Montanari, Roberta, Capelli, Davide, Tauro, Marilena, Loiodice, Fulvio, Tortorella, Paolo

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Betulinic acid is a PPARγ antagonist that improves glucose uptake, promotes osteogenesis and inhibits adipogenesis von Brusotti, Gloria, Montanari, Roberta, Capelli, Davide, Cattaneo, Giulia, Laghezza, Antonio, Tortorella, Paolo, Loiodice, Fulvio, Peiretti, Franck, Bonardo, Bernadette, Paiardini, Alessandro, Calleri, Enrica, Pochetti, Giorgio

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Affinity-based separation methods for the study of biological interactions: The case of peroxisome proliferator-activated receptors in drug discovery von Temporini, Caterina, Brusotti, Gloria, Pochetti, Giorgio, Massolini, Gabriella, Calleri, Enrica

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Identification of the First PPARα/γ Dual Agonist Able To Bind to Canonical and Alternative Sites of PPARγ and To Inhibit Its Cdk5-Mediated Phosphorylation von Laghezza, Antonio, Piemontese, Luca, Cerchia, Carmen, Montanari, Roberta, Capelli, Davide, Giudici, Marco, Crestani, Maurizio, Tortorella, Paolo, Peiretti, Franck, Pochetti, Giorgio, Lavecchia, Antonio, Loiodice, Fulvio

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Cytosolic localization and in vitro assembly of human de novo thymidylate synthesis complex von Spizzichino, Sharon, Boi, Dalila, Boumis, Giovanna, Lucchi, Roberta, Liberati, Francesca Romana, Capelli, Davide, Montanari, Roberta, Pochetti, Giorgio, Piacentini, Roberta, Parisi, Giacomo, Paone, Alessio, Rinaldo, Serena, Contestabile, Roberto, Tramonti, Angela, Paiardini, Alessandro, Giardina, Giorgio, Cutruzzolà, Francesca

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Screening of saponins and sapogenins from Medicago species as potential PPARγ agonists and X-ray structure of the complex PPARγ/caulophyllogenin von Montanari, Roberta, Capelli, Davide, Tava, Aldo, Galli, Andrea, Laghezza, Antonio, Tortorella, Paolo, Loiodice, Fulvio, Pochetti, Giorgio

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A Novel N‑Substituted Valine Derivative with Unique Peroxisome Proliferator-Activated Receptor γ Binding Properties and Biological Activities von Peiretti, Franck, Montanari, Roberta, Capelli, Davide, Bonardo, Bernadette, Colson, Cécilia, Amri, Ez-Zoubir, Grimaldi, Marina, Balaguer, Patrick, Ito, Keiichi, Roeder, Robert G, Pochetti, Giorgio, Brunel, Jean Michel

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Cytosolic localization and invitro assembly of human denovo thymidylate synthesis complex von Spizzichino, Sharon, Boi, Dalila, Boumis, Giovanna, Lucchi, Roberta, Liberati, Francesca Romana, Capelli, Davide, Montanari, Roberta, Pochetti, Giorgio, Piacentini, Roberta, Parisi, Giacomo, Paone, Alessio, Rinaldo, Serena, Contestabile, Roberto, Tramonti, Angela, Paiardini, Alessandro, Giardina, Giorgio, Cutruzzolà, Francesca

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Insights into PPARγ Phosphorylation and Its Inhibition Mechanism von Montanari, Roberta, Capelli, Davide, Yamamoto, Keiko, Awaishima, Hirono, Nishikata, Kimina, Barendregt, Arjan, Heck, Albert J. R, Loiodice, Fulvio, Altieri, Fabio, Paiardini, Alessandro, Grottesi, Alessandro, Pirone, Luciano, Pedone, Emilia, Peiretti, Franck, Brunel, Jean Michel, Itoh, Toshimasa, Pochetti, Giorgio

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A novel N-substituted valine derivative with unique PPARy binding properties and biological activities von Peiretti, Franck, Montanari, Roberta, Capelli, Davide, Bonardo, Bernadette, Colson, Cécilia, Amri, Ez Zoubir, Grimaldi, Marina, Balaguer, Patrick, Pochetti, Giorgio, Brunel, Jean Michel

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A novel N-substituted valine derivative with unique PPARγ binding properties and biological activities von Peiretti, Franck, Montanari, Roberta, Capelli, Davide, Bonardo, Bernadette, Colson, Cécilia, Amri, Ez-Zoubir, Grimaldi, Marina, Balaguer, Patrick, Ito, Keiichi, Roeder, Robert G., Pochetti, Giorgio, Brunel, Jean Michel

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Extra Binding Region Induced by Non-Zinc Chelating Inhibitors into the S 1 ′ Subsite of Matrix Metalloproteinase 8 (MMP-8) von Pochetti, Giorgio, Montanari, Roberta, Gege, Christian, Chevrier, Carine, Taveras, Arthur G., Mazza, Fernando

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Insights into PPARγ phosphorylation and its inhibition mechanism von Montanari, Roberta, Capelli, Davide, Yamamoto, Keiko, Awaishima, Hirono, Nishikata, Kimina, Barendregt, Arjan, Heck, Albert J R, Loiodice, Fulvio, Altieri, Fabio, Paiardini, Alessandro, Grotessi, Alessandro, Pirone, Luciano, Pedone, Emilia Maria, Peiretti, Franck, Brunel, Jean Michel, Itoh, Toshimasa, Pochetti, Giorgio

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Catechol-based matrix metalloproteinase inhibitors with additional antioxidative activity von Tauro, Marilena, Laghezza, Antonio, Loiodice, Fulvio, Piemontese, Luca, Caradonna, Alessia, Capelli, Davide, Montanari, Roberta, Pochetti, Giorgio, Di Pizio, Antonella, Agamennone, Mariangela, Campestre, Cristina, Tortorella, Paolo

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Insights into the Mechanism of Partial Agonism von Pochetti, Giorgio, Godio, Cristina, Mitro, Nico, Caruso, Donatella, Galmozzi, Andrea, Scurati, Samuele, Loiodice, Fulvio, Fracchiolla, Giuseppe, Tortorella, Paolo, Laghezza, Antonio, Lavecchia, Antonio, Novellino, Ettore, Mazza, Fernando, Crestani, Maurizio

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