Apoptosis-inducing factor: vital and lethal von Modjtahedi, Nazanine, Giordanetto, Fabrizio, Madeo, Frank, Kroemer, Guido

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Structural basis of AMPK regulation by small molecule activators von Xiao, Bing, Sanders, Matthew J., Carmena, David, Bright, Nicola J., Haire, Lesley F., Underwood, Elizabeth, Patel, Bhakti R., Heath, Richard B., Walker, Philip A., Hallen, Stefan, Giordanetto, Fabrizio, Martin, Stephen R., Carling, David, Gamblin, Steven J.

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Stabilization of protein–protein interactions by small molecules von Giordanetto, Fabrizio, Schäfer, Anja, Ottmann, Christian

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Macrocyclic Drugs and Clinical Candidates: What Can Medicinal Chemists Learn from Their Properties? von Giordanetto, Fabrizio, Kihlberg, Jan

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Expansion of chemical space for collaborative lead generation and drug discovery: the European Lead Factory Perspective von Karawajczyk, Anna, Giordanetto, Fabrizio, Benningshof, Jorg, Hamza, Daniel, Kalliokoski, Tuomo, Pouwer, Kees, Morgentin, Remy, Nelson, Adam, Müller, Gerhard, Piechot, Alexander, Tzalis, Dimitrios

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High-Throughput Screening of Drug−Brain Tissue Binding and in Silico Prediction for Assessment of Central Nervous System Drug Delivery von Wan, Hong, Rehngren, Mikael, Giordanetto, Fabrizio, Bergström, Fredrik, Tunek, Anders

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A Versatile Strategy for the Synthesis of 4,5-Dihydroxy-2,3-Pentanedione (DPD) and Related Compounds as Potential Modulators of Bacterial Quorum Sensing von Stotani, Silvia, Gatta, Viviana, Medda, Federico, Padmanaban, Mohan, Karawajczyk, Anna, Tammela, Päivi, Giordanetto, Fabrizio, Tzalis, Dimitrios, Collina, Simona

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On Evaluating Molecular-Docking Methods for Pose Prediction and Enrichment Factors von Chen, Hongming, Lyne, Paul D, Giordanetto, Fabrizio, Lovell, Timothy, Li, Jin

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AIF and cyclophilin A cooperate in apoptosis-associated chromatinolysis von CANDE, Céline, VAHSEN, Nicola, PENNINGER, Josef M, KROEMER, Guido, KOURANTI, Ilektra, SCHMITT, Elise, DAUGAS, Eric, SPAHR, Chris, LUBAN, Jeremy, KROEMER, Romano T, GIORDANETTO, Fabrizio, GARRIDO, Carmen

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Impact of Stereospecific Intramolecular Hydrogen Bonding on Cell Permeability and Physicochemical Properties von Over, Björn, McCarren, Patrick, Artursson, Per, Foley, Michael, Giordanetto, Fabrizio, Grönberg, Gunnar, Hilgendorf, Constanze, Lee, Maurice D, Matsson, Pär, Muncipinto, Giovanni, Pellisson, Mélanie, Perry, Matthew W. D, Svensson, Richard, Duvall, Jeremy R, Kihlberg, Jan

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Structure-Based Discovery of Allosteric Modulators of Two Related Class B G-Protein-Coupled Receptors von de Graaf, Chris, Rein, Chantal, Piwnica, David, Giordanetto, Fabrizio, Rognan, Didier

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2‐Sulfonylpyrimidines Target the Kinesin HSET via Cysteine Alkylation von Förster, Tim, Shang, Erchang, Shimizu, Kenshiro, Sanada, Emiko, Schölermann, Beate, Huebecker, Mylene, Hahne, Gernot, López‐Alberca, Maria Pascual, Janning, Petra, Watanabe, Nobumoto, Sievers, Sonja, Giordanetto, Fabrizio, Shimizu, Takeshi, Ziegler, Slava, Osada, Hiroyuki, Waldmann, Herbert

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Small molecule inhibitors of ebola virus infection von Picazo, Edwige, Giordanetto, Fabrizio

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Discovery of AZD2716: A Novel Secreted Phospholipase A2 (sPLA2) Inhibitor for the Treatment of Coronary Artery Disease von Giordanetto, Fabrizio, Pettersen, Daniel, Starke, Ingemar, Nordberg, Peter, Dahlström, Mikael, Knerr, Laurent, Selmi, Nidhal, Rosengren, Birgitta, Larsson, Lars-Olof, Sandmark, Jenny, Castaldo, Marie, Dekker, Niek, Karlsson, Ulla, Hurt-Camejo, Eva

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Lead Optimization of Ethyl 6‑Aminonicotinate Acyl Sulfonamides as Antagonists of the P2Y12 Receptor. Separation of the Antithrombotic Effect and Bleeding for Candidate Drug AZD1283... von Bach, Peter, Antonsson, Thomas, Bylund, Ruth, Björkman, Jan-Arne, Österlund, Krister, Giordanetto, Fabrizio, van Giezen, J. J. J, Andersen, Søren M, Zachrisson, Helen, Zetterberg, Fredrik

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Oral Druggable Space beyond the Rule of 5: Insights from Drugs and Clinical Candidates von Doak, Bradley Croy, Over, Bjӧrn, Giordanetto, Fabrizio, Kihlberg, Jan

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Discovery of 4-hydroxy-1,6-naphthyridine-3-carbonitrile derivatives as novel PDE10A inhibitors von Bauer, Udo, Giordanetto, Fabrizio, Bauer, Martin, O’Mahony, Gavin, Johansson, Kjell E., Knecht, Wolfgang, Hartleib-Geschwindner, Judith, Carlsson, Eva Töppner, Enroth, Cristofer

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Disruption of the PP1/GADD34 complex induces calreticulin exposure von Kepp, Oliver, Galluzzi, Lorenzo, Giordanetto, Fabrizio, Tesniere, Antoine, Vitale, Ilio, Martins, Isabelle, Schlemmer, Frèdèric, Adjemian, Sandy, Zitvogel, Laurence, Kroemer, Guido

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DYRK1A inhibition as potential treatment for Alzheimer's disease von Stotani, Silvia, Giordanetto, Fabrizio, Medda, Federico

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Intramolecular Hydrogen Bond Expectations in Medicinal Chemistry von Giordanetto, Fabrizio, Tyrchan, Christian, Ulander, Johan

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