Tirbanibulin 1% Ointment Significantly Reduces the Actinic Keratosis Area and Severity Index in Patients with Actinic Keratosis: Results from a Real-World Study von Kirchberger, Michael Constantin, Gfesser, Michael, Erdmann, Michael, Schliep, Stefan, Berking, Carola, Heppt, Markus Vincent

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Transonychial water loss in healthy and diseased nails von KRÖNAUER, Christine, GFESSER, Michael, RING, Johannes, ABECK, Dietrich

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SEASONAL VARIATIONS IN THE SEVERITY OF ACNE VULGARIS von GFESSER, MICHAEL, WORRET, WOLF‐INGO

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Multiple Primary Miliary Osteoma Cutis von Gfesser, Michael, Worret, Wolf-Ingo, Hein, Rüdiger, Ring, Johannes

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SEASONAL VARIATIONS IN THE SEVERITY OF ACNE VULGARIS von GFESSER, MICHAEL, WORRET, WOLF-INGO

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Discovery of ABBV/GLPG-3221, a Potent Corrector of CFTR for the Treatment of Cystic Fibrosis von Scanio, Marc J. C, Searle, Xenia B, Liu, Bo, Koenig, John R, Altenbach, Robert, Gfesser, Gregory A, Bogdan, Andrew, Greszler, Stephen, Zhao, Gang, Singh, Ashvani, Fan, Yihong, Swensen, Andrew M, Vortherms, Timothy, Manelli, Arlene, Balut, Corina, Jia, Ying, Gao, Wenqing, Yong, Hong, Schrimpf, Michael, Tse, Chris, Kym, Philip, Wang, Xueqing

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Synthesis and Pharmacology of (Pyridin-2-yl)methanol Derivatives as Novel and Selective Transient Receptor Potential Vanilloid 3 Antagonists von Gomtsyan, Arthur, Schmidt, Robert G, Bayburt, Erol K, Gfesser, Gregory A, Voight, Eric A, Daanen, Jerome F, Schmidt, Diana L, Cowart, Marlon D, Liu, Huaqing, Altenbach, Robert J, Kort, Michael E, Clapham, Bruce, Cox, Phil B, Shrestha, Anurupa, Henry, Rodger, Whittern, David N, Reilly, Regina M, Puttfarcken, Pamela S, Brederson, Jill-Desiree, Song, Ping, Li, Bin, Huang, Susan M, McDonald, Heath A, Neelands, Torben R, McGaraughty, Steve P, Gauvin, Donna M, Joshi, Shailen K, Banfor, Patricia N, Segreti, Jason A, Shebley, Mohamad, Faltynek, Connie R, Dart, Michael J, Kym, Philip R

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Discovery and SAR of 4-aminopyrrolidine-2-carboxylic acid correctors of CFTR for the treatment of cystic fibrosis von Scanio, Marc J.C., Searle, Xenia B., Liu, Bo, Koenig, John R., Altenbach, Robert J., Gfesser, Gregory A., Bogdan, Andrew, Greszler, Stephen, Zhao, Gang, Singh, Ashvani, Fan, Yihong, Swensen, Andrew M., Vortherms, Timothy, Manelli, Arlene, Balut, Corina, Gao, Wenqing, Yong, Hong, Schrimpf, Michael, Tse, Chris, Kym, Philip, Wang, Xueqing

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4-(2-[2-(2(R)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl)benzonitrile and Related 2-Aminoethylbenzofuran H3 Receptor Antagonists Potently Enhance Cognition and Attention von Cowart, Marlon, Faghih, Ramin, Curtis, Michael P, Gfesser, Gregory A, Bennani, Youssef L, Black, Lawrence A, Pan, Liping, Marsh, Kennan C, Sullivan, James P, Esbenshade, Timothy A, Fox, Gerard B, Hancock, Arthur A

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Discovery of 4-(5-(4-Chlorophenyl)-2-methyl-3-propionyl-1H-pyrrol-1-yl)benzenesulfonamide (A-867744) as a Novel Positive Allosteric Modulator of the α7 Nicotinic Acetylcholine Rece... von Faghih, Ramin, Gopalakrishnan, Sujatha M, Gronlien, Jens Halvard, Malysz, John, Briggs, Clark A, Wetterstrand, Caroline, Ween, Hilde, Curtis, Michael P, Sarris, Kathy A, Gfesser, Gregory A, El-Kouhen, Rachid, Robb, Holly M, Radek, Richard J, Marsh, Kennan C, Bunnelle, William H, Gopalakrishnan, Murali

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4-(2-[2-(2( R )-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl)benzonitrile and Related 2-Aminoethylbenzofuran H 3 Receptor Antagonists Potently Enhance Cognition and Attention von Cowart, Marlon, Faghih, Ramin, Curtis, Michael P., Gfesser, Gregory A., Bennani, Youssef L., Black, Lawrence A., Pan, Liping, Marsh, Kennan C., Sullivan, James P., Esbenshade, Timothy A., Fox, Gerard B., Hancock, Arthur A.

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Structure–activity relationships of arylbenzofuran H3 receptor antagonists von Gfesser, Gregory A., Faghih, Ramin, Bennani, Youssef L., Curtis, Michael P., Esbenshade, Timothy A., Hancock, Arthur A., Cowart, Marlon D.

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Synthesis and SAR of 5-Amino- and 5-(Aminomethyl)benzofuran Histamine H 3 Receptor Antagonists with Improved Potency von Sun, Minghua, Zhao, Chen, Gfesser, Gregory A., Thiffault, Christine, Miller, Thomas R., Marsh, Kennan, Wetter, Jill, Curtis, Michael, Faghih, Ramin, Esbenshade, Timothy A., Hancock, Arthur A., Cowart, Marlon

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Synthesis and SAR of 5-Amino- and 5-(Aminomethyl)benzofuran Histamine H3 Receptor Antagonists with Improved Potency von Sun, Minghua, Zhao, Chen, Gfesser, Gregory A, Thiffault, Christine, Miller, Thomas R, Marsh, Kennan, Wetter, Jill, Curtis, Michael, Faghih, Ramin, Esbenshade, Timothy A, Hancock, Arthur A, Cowart, Marlon

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Novel heterocyclic-substituted benzofuran histamine H3 receptor antagonists: in vitro properties, drug-likeness, and behavioral activity von Cowart, Marlon, Gfesser, Gregory A, Browman, Kaitlin E, Faghih, Ramin, Miller, Thomas R, Milicic, Ivan, Baranowski, John L, Krueger, Kathleen M, Witte, David G, Molesky, Angela L, Komater, Victoria A, Buckley, Michael J, Diaz, Gilbert J, Gagne, Gerard D, Zhou, Deliang, Deng, Xiaoqing, Pan, Liping, Roberts, Ellen M, Diehl, Marilyn S, Wetter, Jill M, Marsh, Kennan C, Fox, Gerard B, Brioni, Jorge D, Esbenshade, Timothy A, Hancock, Arthur A

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5-(3-Bromophenyl)-7-(6-morpholin-4-ylpyridin-3-yl)pyrido[2,3-d]pyrimidin-4-ylamine: structure–activity relationships of 7-substituted heteroaryl analogs as non-nucleoside adenosine... von Matulenko, Mark A., Lee, Chih-Hung, Jiang, Meiqun, Frey, Robin R., Cowart, Marlon D., Bayburt, Erol K., DiDomenico, Stanley, Gfesser, Gregory A., Gomtsyan, Arthur, Zheng, Guo Zhu, McKie, Jeffery A., Stewart, Andrew O., Yu, Haixia, Kohlhaas, Kathy L., Alexander, Karen M., McGaraughty, Steve, Wismer, Carol T., Mikusa, Joseph, Marsh, Kennan C., Snyder, Ronald D., Diehl, Marilyn S., Kowaluk, Elizabeth A., Jarvis, Michael F., Bhagwat, Shripad S.

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Discovery of 4-Amino-5-(3-bromophenyl)-7-(6-morpholino-pyridin- 3-yl)pyrido[2,3-d]pyrimidine, an Orally Active, Non-Nucleoside Adenosine Kinase Inhibitor von Lee, Chih-Hung, Jiang, Meiqun, Cowart, Marlon, Gfesser, Greg, Perner, Richard, Kim, Ki Hwan, Gu, Yu Gui, Williams, Michael, Jarvis, Michael F, Kowaluk, Elizabeth A, Stewart, Andrew O, Bhagwat, Shripad S

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Synthesis and structure-activity relationships of 5-heteroatom-substituted pyridopyrimidines as adenosine kinase inhibitors von Gfesser, Gregory A, Bayburt, Erol K, Cowart, Marlon, DiDomenico, Stanley, Gomtsyan, Arthur, Lee, Chih-Hung, Stewart, Andrew O, Jarvis, Michael F, Kowaluk, Elizabeth A, Bhagwat, Shripad S

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Adenosine kinase inhibitors: polar 7-Substitutent of pyridopyrimidine derivatives improving their locomotor selectivity von Zheng, Guo Zhu, Mao, Yue, Lee, Chih-Hung, Pratt, John K., Koenig, John R., Perner, Richard J., Cowart, Marlon D., Gfesser, Gregory A., McGaraughty, Steve, Chu, Katharine L., Zhu, Chang, Yu, Haixia, Kohlhaas, Kathy, Alexander, Karen M., Wismer, Carol T., Mikusa, Joseph, Jarvis, Michael F., Kowaluk, Elizabeth A., Stewart, Andrew O.

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Correction to Synthesis and SAR of 5-Amino- and 5-(Aminomethyl)benzofuran Histamine H 3 Receptor Antagonists with Improved Potency von Sun, Minghua, Zhao, Chen, Gfesser, Gregory A., Thiffault, Christine, Miller, Thomas R., Marsh, Kennan, Wetter, Jill, Curtis, Michael, Faghih, Ramin, Esbenshade, Timothy A., Hancock, Arthur A., Cowart, Marlon

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