Synthesis and pharmacological properties of 5H,10H-imidazo[1,2-a]indeno[1,2-e]pyrazine-4-one, a new competitive AMPA/KA receptor antagonist von Mignani, Serge, Aloup, Jean-Claude, Barreau, Michel, Blanchard, Jean Charles, Böhme, Georg Andrees, Boireau, Alain, Damour, Dominique, Debono, Marc-Williams, Dubroeucq, Marie-Christine, Genevois-Borella, Arielle, Imperato, Assunta, Jimonet, Patrick, Pratt, Jeremy, Randle, John C.R., Reibaud, Michel, Ribeill, Yves, Stutzmann, Jean-Marie

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Abstract 130: Pharmacological effects of selective xCT inhibition in ARID1A mutated cancer models von Henry, Christophe, Péron, Philippe, Blanchet, Anne-Marie, Genevois-Borella, Arielle, Trellu, Marc, Bourges, Dorothée, Lienard, Philippe, Basset, Alexandra, Jouannot, Erwan, Philippo, Christophe, Debussche, Laurent, Moll, Jürgen

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In vitro and in vivo characterization of TC-1827, a novel brain α4β2 nicotinic receptor agonist with pro-cognitive activity von Bohme, Georg Andrees, Letchworth, Sharon R., Piot-Grosjean, Odile, Gatto, Gregory J., Obinu, Marie-Carmen, Caldwell, William S., Laville, Michel, Brunel, Pascale, Pellerin, Rachel, Leconte, Jean-Pierre, Genevois-Borella, Arielle, Dubedat, Pierre, Mazadier, Martine, Pradier, Laurent, Bencherif, Merouane, Benavides, Jesus

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PYRAZOLOPYRAZINONE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND THERAPEUTIC USES THEREOF von GENEVOIS-BORELLA, Arielle, OBINU-REIBAUD, Maria-Carmen

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A convenient one-pot synthesis of phosphino-dipeptide analogs von Cristau, Henri-Jean, Coulombeau, Agnès, Genevois-Borella, Arielle, Pirat, Jean-Luc

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Preparation of phosphinodipeptide analogs as building blocks for pseudopeptides synthesis von Cristau, Henri-Jean, Coulombeau, Agnès, Genevois-Borella, Arielle, Sanchez, Frédéric, Pirat, Jean-Luc

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ChemInform Abstract: A Preparative Route to Fused 4-Hydroxy-3-phenylindeno(benzothieno)pyridin-2-ones von Genevois-Borella, Arielle, Vuilhorgne, Marc, Mignani, Serge

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9-Carboxymethyl-5H, 10H-imidazo[1,2-a]indeno[1,2-e]pyrazin-4-one-2-carbocylic acid (RPR117824): Selective anticonvulsive and neuroprotective AMPA antagonist von MIGNANI, Serge, BOHME, Georg Andrees, WAHL, Florence, STUTZMANN, Jean-Marie, BIRRAUX, Guillaume, BOIREAU, T. Alain, JIMONET, Patrick, DAMOUR, Dominique, GENEVOIS-BORELLA, Arielle, DEBONO, Marc-Williams, PRATT, Jeremy, VUILHORGNE, Marc

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PYRAZOLOPYRAZINE COMPOUNDS AS SHP2 INHIBITORS von KARLSSON, Andreas, DEVILLERS, Ingrid, GENEVOIS-BORELLA, Arielle, BEGIS, Guillaume, FORICHER, Yann, GILL, Adrian L, BIANCIOTTO, Marc, KOLTUN, Elena S

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PYRAZOLOPYRAZINE COMPOUNDS AS SHP2 INHIBITORS von KARLSSON, Andreas, DEVILLERS, Ingrid, GENEVOIS-BORELLA, Arielle, BEGIS, Guillaume, FORICHER, Yann, GILL, Adrian L, BIANCIOTTO, Marc, KOLTUN, Elena S

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ChemInform Abstract: A Preparative Route to Fused Indeno[1,2-e][1,2,4]triazolo[4,3-a]pyrazin-4-ones von Ribeill, Yves, Genevois-Borella, Arielle, Vuilhorgne, Marc, Mignani, Serge

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ChemInform Abstract: A Convenient One-Pot Synthesis of Phosphino-Dipeptide Analogues von Cristau, Henri-Jean, Coulombeau, Agnes, Genevois-Borella, Arielle, Pirat, Jean-Luc

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Indeno[1,2-b]pyrazin-2,3-diones: A New Class of Antagonists at the Glycine Site of the NMDA Receptor with Potent in Vivo Activity von Jimonet, Patrick, Ribeill, Yves, Bohme, Georg Andrees, Boireau, Alain, Chevé, Michel, Damour, Dominique, Doble, Adam, Genevois-Borella, Arielle, Herman, Frédéric, Imperato, Assunta, Le Guern, Sylvain, Manfré, Franco, Pratt, Jeremy, Randle, John C. R, Stutzmann, Jean-Marie, Mignani, Serge

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Enantioselective synthesis of (+)-3-isorauniticine via a catalytic tandem palladium-ene/carbonylation reaction von Oppolzer, Wolfgang, Bienayme, Hugues, Genevois-Borella, Arielle

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MACROCYCLIC COMPOUNDS, COMPOSITIONS, AND METHODS OF USING THEREOF von BORCHERDING, David, GUESSREGEN, Stefan, GAO, Zhongli, CAUSSANEL, Franck, GOOD, Andrew, DEVILLERS, Ingrid, SCHWINK, Lothar, RACKELMANN, Nils, THURAIRATNAM, Sukanthini, HIRTH, Brad, LIU, Jinyu, HURLBUT, Greg, GENEVOIS-BORELLA, Arielle, TOPALOV, George, THOMPSON, Fabienne, RUF, Sven, MACOR, John, VAZ, Roy, LI, Yi, BERNARDELLI, Patrick, LIAO, Junkai, GLOMBIK, Heiner, NICOLAI, Eric, RUVINSKY, Anatoly, MUNSON, Mark, KOTHE, Michael, PODESCHWA, Michael, SLOWINSKI, Franck

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MACROCYCLIC COMPOUNDS, COMPOSITIONS AND METHODS OF USING THEREOF von BORCHERDING, David, GUESSREGEN, Stefan, GAO, Zhongli, CAUSSANEL, Franck, GOOD, Andrew, BERNADELLI, Patrick, DEVILLERS, Ingrid, SCHWINK, Lothar, RACKELMANN, Nils, THURAIRATNAM, Sukanthini, HIRTH, Brad, LIU, Jinyu, HURLBUT, Greg, GENEVOIS-BORELLA, Arielle, TOPALOV, George, THOMPSON, Fabienne, RUF, Sven, MACOR, John, VAZ, Roy, LI, Yi, LIAO, Junkai, GLOMBIK, Heiner, NICOLAI, Eric, RUVINSKY, Anatoly, MUNSON, Mark, KOTHE, Michael, PODESCHWA, Michael, SLOWINSKI, Franck

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4,10-Dihydro-4-oxo-4H-imidazo[1,2-a]indeno[1,2-e]pyrazin-2-carboxylic acid derivatives: highly potent and selective AMPA receptors antagonists with in vivo activity von Stutzmann, J M, Bohme, G A, Boireau, A, Damour, D, Debono, M W, Genevois-Borella, A, Imperato, A, Jimonet, P, Pratt, J, Randle, J C, Ribeill, Y, Vuilhorgne, M, Mignani, S

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Spiro-imidazo[1,2-a]indeno[1,2-e]pyrazine-4-one derivatives are mixed AMPA and NMDA glycine-site antagonists active in vivo von Jimonet, Patrick, Boireau, Alain, Chevé, Michel, Damour, Dominique, Genevois-Borella, Arielle, Imperato, Assunta, Pratt, Jeremy, Randle, John C.R., Ribeill, Yves, Stutzmann, Jean-Marie, Mignani, Serge

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Synthesis and potent anticonvulsant activities of 4-oxo-imidazo[1,2- a]indeno[1,2- e]pyrazin-8- and -9-carboxylic (acetic) acid AMPA antagonists von Pratt, Jeremy, Jimonet, Patrick, Bohme, Georg Andrees, Boireau, Alain, Damour, Dominique, Debono, Marc Williams, Genevois-Borella, Arielle, Randle, John C.R, Ribeill, Yves, Stutzmann, Jean-Marie, Vuilhorgne, Marc, Mignani, Serge

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9-Carboxymethyl-5 H ,10 H -imidazo[1,2- a ]indeno[1,2- e ]pyrazin-4-one-2-carbocylic Acid (RPR117824): Selective Anticonvulsive and Neuroprotective AMPA Antagonist von Mignani, Serge, Bohme, Georg Andrees, Birraux, Guillaume, Boireau, Alain, Jimonet, Patrick, Damour, Dominique, Genevois-Borella, Arielle, Debono, Marc-Williams, Pratt, Jeremy, Vuilhorgne, Marc, Wahl, Florence, Stutzmann, Jean-Marie

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