Characterization and isolation of an 18-crown-6 complex of potassium hydroxide prepared by milling: application to mechanochemical organic synthesis von Vugrin, Leonarda, Halasz, Ivan, Geneste, Hervé

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One-step hydroxylation of aryl and heteroaryl fluorides using mechanochemistry von Rodrigo, Eduardo, Wiechert, Rainer, Walter, Magnus W, Braje, Wilfried, Geneste, Hervé

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Parallel mechanochemical optimization - Buchwald-Hartwig C-N coupling as a test case von Lemesre, Quentin, Wiesner, Thomas, Wiechert, Rainer, Rodrigo, Eduardo, Triebel, Sonja, Geneste, Hervé

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Investigation of Mechanochemical Sonogashira CouplingsFrom Batch Solution to Continuous Reactive Extrusion through Ball-Milling Optimization von Hastings, Riley H., Mokhtar, Mennatullah M., Ruggles, Alexander, Schmidt, Constanze, Bourdeau, David, Haibach, Michael C., Geneste, Hervé, Mack, James, Co, Sarah S., Speight, Isaiah R.

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Investigation of Mechanochemical Thianthrene-Mediated Aryl C−H Functionalization von Vugrin, Leonarda, Cvrtila, Ivica, Geneste, Hervé, Halasz, Ivan

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Novel, potent, selective, and brain penetrant phosphodiesterase 10A inhibitors von Geneste, Hervé, Drescher, Karla, Jakob, Clarissa, Laplanche, Loïc, Ochse, Michael, Torrent, Maricel

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Multi-faceted reactivity of N -fluorobenzenesulfonimide (NFSI) under mechanochemical conditions: fluorination, fluorodemethylation, sulfonylation, and amidation reactions von Hernández, José G, Ardila-Fierro, Karen J, Barišić, Dajana, Geneste, Hervé

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Novel, potent, selective and brain penetrant vasopressin 1b receptor antagonists von Geneste, Hervé, Bhowmik, Swati, van Gaalen, Marcel M., Hornberger, Wilfried, Hutchins, Charles W., Netz, Astrid, Oost, Thorsten, Unger, Liliane

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Potent and selective oxindole-based vasopressin 1b receptor antagonists with improved pharmacokinetic properties von Oost, Thorsten, Backfisch, Gisela, Bhowmik, Swati, van Gaalen, Marcel M., Geneste, Hervé, Hornberger, Wilfried, Lubisch, Wilfried, Netz, Astrid, Unger, Liliane, Wernet, Wolfgang

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2-Substituted 4-(Trifluoromethyl)phenols by Directed ortho-Lithiation von Geneste, Hervé, Schäfer, Bernd

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Design and synthesis of 1,5- and 2,5-substituted tetrahydrobenzazepinones as novel potent and selective integrin αvβ3antagonists von KLING, Andreas, BACKFISCH, Gisela, DELZER, Jürgen, GENESTE, Herve, GRAEF, Claudia, HORNBERGER, Wilfried, LANGE, Udo E. W, LAUTERBACH, Arnulf, SEITZ, Werner, SUBKOWSKI, Thomas

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Mononuclear Tetraamineplatinum(II) Complexes: Synthesis, Anticancer Activity, DNA Binding, and Cellular Uptake von Robillard, Marc S., Jansen, Bart A. J., Lochner, Martin, Geneste, Hervé, Li, Yi, Brouwer, Jaap, Hesse, Manfred, Reedijk, Jan

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Design and synthesis of novel potent and selective integrin αvβ3 antagonists—Novel synthetic routes to isoquinolinone, benzoxazinone, and quinazolinone acetates von Seitz, Werner, Geneste, Hervé, Backfisch, Gisela, Delzer, Jürgen, Graef, Claudia, Hornberger, Wilfried, Kling, Andreas, Subkowski, Thomas, Zimmermann, Norbert

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Synthesis and SAR of highly potent and selective dopamine D 3-receptor antagonists: Quinolin(di)one and benzazepin(di)one derivatives von Geneste, Hervé, Backfisch, Gisela, Braje, Wilfried, Delzer, Jürgen, Haupt, Andreas, Hutchins, Charles W., King, Linda L., Lubisch, Wilfried, Steiner, Gerd, Teschendorf, Hans-Jürgen, Unger, Liliane, Wernet, Wolfgang

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Design and synthesis of novel potent and selective integrin α v β 3 antagonists—Novel synthetic routes to isoquinolinone, benzoxazinone, and quinazolinone acetates von Seitz, Werner, Geneste, Hervé, Backfisch, Gisela, Delzer, Jürgen, Graef, Claudia, Hornberger, Wilfried, Kling, Andreas, Subkowski, Thomas, Zimmermann, Norbert

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Design and synthesis of novel potent and selective integrin ανβ3 antagonists : Novel synthetic routes to isoquinolinone, benzoxazinone, and quinazolinone acetates von SEITZ, Werner, GENESTE, Hervé, BACKFISCH, Gisela, DELZER, Jürgen, GRAEF, Claudia, HORNBERGER, Wilfried, KLING, Andreas, SUBKOWSKI, Thomas, ZIMMERMANN, Norbert

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Synthesis of 13C-dilabeled 4-coumaroylspermidines von Geneste, Hervé, Hesse, Manfred

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The Superbase Approach to Flurbiprofen: An Exercise in Optionally Site-Selective Metalation von Schlosser, Manfred, Geneste, Hervé

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Synthesis and SAR of N-substituted dibenzazepinone derivatives as novel potent and selective alpha(V)beta(3) antagonists von Kling, Andreas, Backfisch, Gisela, Delzer, Jürgen, Geneste, Hervé, Graef, Claudia, Holzenkamp, Uta, Hornberger, Wilfried, Lange, Udo E W, Lauterbach, Arnulf, Mack, Helmut, Seitz, Werner, Subkowski, Thomas

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Synthesis and SAR of N-substituted dibenzazepinone derivatives as novel potent and selective αVβ3 antagonists von KLING, Andreas, BACKFISCH, Gisela, SEITZ, Werner, SUBKOWSKI, Thomas, DELZER, Jürgen, GENESTE, Hervé, GRAEF, Claudia, HOLZENKAMP, Uta, HORNBERGER, Wilfried, LANGE, Udo E. W, LAUTERBACH, Arnulf, MACK, Helmut

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