Solution-phase library generation: methods and applications in drug discovery von Gayo, L.M

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Inhibitors of NF-κB and AP-1 Gene Expression:  SAR Studies on the Pyrimidine Portion of 2-Chloro-4-trifluoromethylpyrimidine-5-[N-(3‘,5‘-bis(trifluoromethyl)phenyl)carboxamide]... von Palanki, Moorthy S. S, Erdman, Paul E, Gayo-Fung, Leah M, Shevlin, Graziella I, Sullivan, Robert W, Goldman, Mark E, Ransone, Lynn J, Bennett, Brydon L, Manning, Anthony M, Suto, Mark J

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Effects of SP500263, a novel, potent antiestrogen, on breast cancer cells and in xenograft models von BRADY, Helen, DESAI, Sonal, STEIN, Bernd, GAYO-FUNG, Leah M, KHAMMUNGKHUNE, Sak, MCKIE, Jeffrey A, O'LEARY, Eoin, PASCASIO, Laura, SUTHERLAND, May Kung, ANDERSON, David W, BHAGWAT, Shripad S

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Ion-exchange resins for solution phase parallel synthesis of chemical libraries von Gayo, Leah M., Suto, Mark J.

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Differential response of estrogen receptors alpha and beta to SP500263, a novel potent selective estrogen receptor modulator von Brady, Helen, Doubleday, Mary, Gayo-Fung, Leah M, Hickman, Matt, Khammungkhune, Sak, Kois, Adam, Lipps, Stephanie, Pierce, Steve, Richard, Normand, Shevlin, Graciella, Sutherland, May Kung, Anderson, David W, Bhagwat, Shripad S, Stein, Bernd

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Traceless linker: Oxidative activation and displacement of a sulfur-based linker von Gayo, Leah M., Suto, Mark J.

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Synthetic Utility of Alkenylcyclobutenedione Monoketals. Michael Additions and the Synthesis of a Natural Benzofuranosesquiterpenequinone von Liu, Hui, Gayo, Leah M, Sullivan, Robert W, Choi, Angela Y. H, Moore, Harold W

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SP500263, a novel SERM, blocks osteoclastogenesis in a human bone cell model: role of IL-6 and GM-CSF von Sutherland, May S.Kung, Lipps, Stephanie G, Patnaik, Nandita, Gayo-Fung, Leah M, Khammungkune, Sak, Xie, Weilin, Brady, Helen A, Barbosa, Miguel S, Anderson, David W, Stein, Bernd

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Lead identification of a potent benzopyranone selective estrogen receptor modulator von McKie, Jeffrey A., Bhagwat, Shripad S., Brady, Helen, Doubleday, Mary, Gayo, Leah, Hickman, Mathew, Jalluri, Ravi K., Khammungkhune, Sak, Kois, Adam, Mortensen, Deborah, Richard, Normand, Sapienza, John, Shevlin, Graziella, Stein, Bernd, Sutherland, May

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A potentially general regiospecific synthesis of substituted quinones from dimethyl squarate von Gayo, Leah M, Winters, Michael P, Moore, Harold W

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Use of pentafluorophenyl esters for one-pot protection/activation of amino and thiol carboxylic acids von Gayo, Leah M., Suto, Mark J.

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Structure–Activity Relationship Studies of Ethyl 2-[(3-Methyl-2,5-dioxo(3-pyrrolinyl))amino]-4-(trifluoromethyl)pyrimidine-5-carboxylate: An Inhibitor of AP-1 and NF-κB Mediated Ge... von Palanki, Moorthy S.S., Gayo-Fung, Leah M., Shevlin, Graziella I., Erdman, Paul, Sato, Mark, Goldman, Mark, Ransone, Lynn J., Spooner, Cheryl

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Solution-phase parallel synthesis using ion-exchange resins von Suto, Mark J., Gayo-Fung, Leah M., Palanki, Moorthy S.S., Sullivan, Robert

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Structure-activity relationship studies of ethyl 2-[(3-methyl-2,5-dioxo(3-pyrrolinyl))amino]-4-(trifluoromethyl)pyrimidine-5-carboxylate: an inhibitor of AP-1 and NF-kappaB mediate... von Palanki, Moorthy S S, Gayo-Fung, Leah M, Shevlin, Graziella I, Erdman, Paul, Sato, Mark, Goldman, Mark, Ransone, Lynn J, Spooner, Cheryl

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Structure-Activity Relationship Studies of Ethyl 2-[(3-Methyl-2,5-dioxo(3-pyrrolinyl))amino] -4-(trifluoromethyl)pyrimidine-5-carboxylate: An Inhibitor of AP-1 and NF-ϰB Mediated G... von Palanki, Moorthy S. S., Gayo-Fung, Leah M., Shevlin, Graziella I., Erdman, Paul, Sato, Mark, Goldman, Mark, Ransone, Lynn J., Spooner, Cheryl

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Structure-activity relationship studies of ethyl 2-[(3-methyl-2,5-dioxo(3-pyrrolinyl))amino]-4-(trifluoromethyl)pyrimidine-5-carb oxylate: An inhibitor of AP-1 and NF-kB mediated g... von PALANKI, Moorthy S. S, GAYO-FUNG, Leah M, SHEVLIN, Graziella I, ERDMAN, Paul, SATO, Mark, GOLDMAN, Mark, RANSONE, Lynn J, SPOONER, Cheryl

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Differential Response of Estrogen Receptors α and β to SP500263, a Novel Potent Selective Estrogen Receptor Modulator von Helen Brady, Mary Doubleday, Leah M. Gayo-Fung, Matt Hickman, Sak Khammungkhune, Adam Kois, Stephanie Lipps, Steve Pierce, Normand Richard, Graciella Shevlin, May Kung Sutherland, David W. Anderson, Shripad S. Bhagwat, Bernd Stein

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Differential Response of Estrogen Receptors α and β to SP500263, a Novel Potent Selective Estrogen Receptor Modulator von Brady, Helen, Doubleday, Mary, Gayo-Fung, Leah M., Hickman, Matt, Khammungkhune, Sak, Kois, Adam, Lipps, Stephanie, Pierce, Steve, Richard, Normand, Shevlin, Graciella, Sutherland, May Kung, Anderson, David W., Bhagwat, Shripad S., Stein, Bernd

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Compounds and methods for modulation of estrogen receptors von STEIN BERND M, GAYO-FUNG LEAH MARIE

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Compounds and methods for modulation of estrogen receptors von Gayo-Fung, Leah Marie, Stein, Bernd M

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