Highly Enantioselective Rhodium-Catalyzed Transfer Hydrogenation of Tetrasubstituted Olefins: Application toward the Synthesis of GPR40 Agonist MK-2305 von Zhong, Yong-Li, Ji, Yining, Wang, Heather, Wang, Xiao, Gauthier, Donald R

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A metal-catalysed functional group metathesis approach to the carbon isotope labelling of carboxylic acids von Kinney, R. Garrison, Zgheib, José, Lagueux-Tremblay, Pierre-Louis, Zhou, Cuihan, Yang, Haifeng, Li, Jingwei, Gauthier, Donald R., Arndtsen, Bruce A.

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A General, One-Pot Method for the Synthesis of Sulfinic Acids from Methyl Sulfones von Gauthier, Donald R, Yoshikawa, Naoki

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Total Synthesis of Darobactin A von Nesic, Marko, Ryffel, David B., Maturano, Jonathan, Shevlin, Michael, Pollack, Scott R., Gauthier, Donald R., Trigo-Mouriño, Pablo, Zhang, Li-Kang, Schultz, Danielle M., McCabe Dunn, Jamie M., Campeau, Louis-Charles, Patel, Niki R., Petrone, David A., Sarlah, David

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Palladium-Catalyzed Carbon Isotope Exchange on Aliphatic and Benzoic Acid Chlorides von Gauthier, Donald R, Rivera, Nelo R, Yang, Haifeng, Schultz, Danielle M, Shultz, C. Scott

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Characterization of impurities of HIV NNRTI Doravirine by UHPLC-high resolution MS and tandem MS analysis von Zhang, Li-Kang, Yang, Ross, Sheng, Huaming, Helmy, Roy, Zheng, Jinjian, Cao, Yang, Gauthier Jr, Donald R.

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Highly Efficient Synthesis of HIV NNRTI Doravirine von Gauthier, Donald R, Sherry, Benjamin D, Cao, Yang, Journet, Michel, Humphrey, Guy, Itoh, Tetsuji, Mangion, Ian, Tschaen, David M

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Potassium isopropyl xanthate (PIX): an ultra-efficient palladium scavenger von Ren, Hong, Strulson, Christopher A., Humphrey, Guy, Xiang, Rong, Li, Guangtao, Gauthier, Donald R., Maloney, Kevin M.

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Development of a Commercial Manufacturing Route to 2‑Fluoroadenine, The Key Unnatural Nucleobase of Islatravir von Hong, Cynthia M, Xu, Yingju, Chung, John Y. L, Schultz, Danielle M, Weisel, Mark, Varsolona, Richard J, Zhong, Yong-Li, Purohit, Akasha K, He, Cyndi Q, Gauthier, Donald R, Humphrey, Guy R, Maloney, Kevin M, Lévesque, François, Wang, Zhixun, Whittaker, Aaron M, Sirota, Eric, McMullen, Jonathan P

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A chemoenzymatic strategy for site-selective functionalization of native peptides and proteins von Fryszkowska, Anna, An, Chihui, Alvizo, Oscar, Banerjee, Goutami, Canada, Keith A., Cao, Yang, DeMong, Duane, Devine, Paul N., Duan, Da, Elgart, David M., Farasat, Iman, Gauthier, Donald R., Guidry, Erin N., Jia, Xiujuan, Kong, Jongrock, Kruse, Nikki, Lexa, Katrina W., Makarov, Alexey A., Mann, Benjamin F., Milczek, Erika M., Mitchell, Vesna, Nazor, Jovana, Neri, Claudia, Orr, Robert K., Orth, Peter, Phillips, Eric M., Riggins, James N., Schafer, Wes A., Silverman, Steven M., Strulson, Christopher A., Subramanian, Nandhitha, Voladri, Rama, Yang, Hao, Yang, Jie, Yi, Xiang, Zhang, Xiyun, Zhong, Wendy

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Mechanistic Understanding of a Robust and Scalable Synthesis of Per(6-deoxy-6-halo)cyclodextrins, Versatile Intermediates for Cyclodextrin Modification von Zultanski, Susan L, Kuhl, Nadine, Zhong, Wendy, Cohen, Ryan D, Reibarkh, Mikhail, Jurica, Jon, Kim, Jungchul, Weisel, Lauren, Ekkati, Anil R, Klapars, Artis, Gauthier, Donald R, McCabe Dunn, Jamie M

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An efficient synthesis of 4-chromanones von Zhong, Yong-Li, Boruta, David T., Gauthier, Donald R., Askin, David

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Synthesis of Antifungal Glucan Synthase Inhibitors from Enfumafungin von Zhong, Yong-Li, Gauthier, Donald R, Shi, Yao-Jun, McLaughlin, Mark, Chung, John Y. L, Dagneau, Philippe, Marcune, Benjamin, Krska, Shane W, Ball, Richard G, Reamer, Robert A, Yasuda, Nobuyoshi

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Rapid End-Game Process Development and First GMP Production of MK-7845: An Experimental Antiviral Treatment for COVID-19 von Deprez, Nicholas R., Hughes, Jonathan M. E., Badir, Shorouk O., Popov, Stasik, Andreani, Teresa, Bade, Rachel S., Hartmanshenn, Clara, Kwok, Thomas Tai-min, Gauthier, Donald R., Salehi Marzijarani, Nastaran, Sakhaei, Zeinab, Drout, Riki, Castro, Steve, Schenk, David J., Wolstenholme, Charles, Padivitage, Nilusha, Welch, Cody, Kowalski, Jason R., Kassim, Brittany, Liu, Yong, Cohen, Ryan D., Confer, Alex M., Dal Poggetto, Guilherme, Brunskill, Andrew P. J., Peng, Feng, Qi, Ji, Xu, Jing, Lin, Mingxiang, McCabe Dunn, Jamie M.

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13 C NMR-Based Approaches for Solving Challenging Stereochemical Problems von Ndukwe, Ikenna E, Brunskill, Andrew, Gauthier, Jr, Donald R, Zhong, Yong-Li, Martin, Gary E, Williamson, R Thomas, Reibarkh, Mikhail, Liu, Yizhou

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A Concise Synthesis of (S)-N-Ethoxycarbonyl-α-methylvaline von Kuethe, Jeffrey T, Gauthier, Donald R, Beutner, Gregory L, Yasuda, Nobuyoshi

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Facile Synthesis of 2-Bromo-3-fluorobenzonitrile:  An Application and Study of the Halodeboronation of Aryl Boronic Acids von Szumigala, Ronald H, Devine, Paul N, Gauthier, Donald R, Volante, R. P

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Palladium-Catalyzed Regioselective Arylation of Imidazo[1,2-b][1,2,4]triazine:  Synthesis of an α2/ 3-Selective GABA Agonist von Gauthier, Donald R, Limanto, John, Devine, Paul N, Desmond, Richard A, Szumigala, Ronald H, Foster, Bruce S, Volante, R. P

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An Efficient Chemoenzymatic Approach to (S)-γ-Fluoroleucine Ethyl Ester von Limanto, John, Shafiee, Ali, Devine, Paul N., Upadhyay, Veena, Desmond, Richard A., Foster, Bruce R., Gauthier, Donald R., Reamer, Robert A., Volante, R. P.

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Design Procedure of a Novel Microturbine Low NOx Conical Wire-Mesh Duct Burner von Ramadan, Omar B, Gauthier, J. E. Donald, Hughes, Patrick M, Brandon, Robert

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