Adenosine A2A receptor antagonists: from caffeine to selective non‐xanthines von Jacobson, Kenneth A., Gao, Zhan‐Guo, Matricon, Pierre, Eddy, Matthew T., Carlsson, Jens

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Historical and Current Adenosine Receptor Agonists in Preclinical and Clinical Development von Jacobson, Kenneth A, Tosh, Dilip K, Jain, Shanu, Gao, Zhan-Guo

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A3 Adenosine Receptors as Modulators of Inflammation: From Medicinal Chemistry to Therapy von Jacobson, Kenneth A., Merighi, Stefania, Varani, Katia, Borea, Pier Andrea, Baraldi, Stefania, Aghazadeh Tabrizi, Mojgan, Romagnoli, Romeo, Baraldi, Pier Giovanni, Ciancetta, Antonella, Tosh, Dilip K., Gao, Zhan‐Guo, Gessi, Stefania

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A2B Adenosine Receptor and Cancer von Gao, Zhan-Guo, Jacobson, Kenneth A.

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Structure of an Agonist-Bound Human A2A Adenosine Receptor von FEI XU, HUIXIAN WU, KATRITCH, Vsevolod, GYE WON HAN, JACOBSON, Kenneth A, GAO, Zhan-Guo, CHEREZOV, Vadim, STEVENS, Raymond C

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Structural Connection between Activation Microswitch and Allosteric Sodium Site in GPCR Signaling von White, Kate L., Eddy, Matthew T., Gao, Zhan-Guo, Han, Gye Won, Lian, Tiffany, Deary, Alexander, Patel, Nilkanth, Jacobson, Kenneth A., Katritch, Vsevolod, Stevens, Raymond C.

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Allosteric Coupling of Drug Binding and Intracellular Signaling in the A2A Adenosine Receptor von Eddy, Matthew T., Lee, Ming-Yue, Gao, Zhan-Guo, White, Kate L., Didenko, Tatiana, Horst, Reto, Audet, Martin, Stanczak, Pawel, McClary, Kyle M., Han, Gye Won, Jacobson, Kenneth A., Stevens, Raymond C., Wüthrich, Kurt

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Two disparate ligand-binding sites in the human P2Y1 receptor von Zhang, Dandan, Gao, Zhan-Guo, Zhang, Kaihua, Kiselev, Evgeny, Crane, Steven, Wang, Jiang, Paoletta, Silvia, Yi, Cuiying, Ma, Limin, Zhang, Wenru, Han, Gye Won, Liu, Hong, Cherezov, Vadim, Katritch, Vsevolod, Jiang, Hualiang, Stevens, Raymond C., Jacobson, Kenneth A., Zhao, Qiang, Wu, Beili

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Fragment-based design of selective GPCR ligands guided by free energy simulations von Matricon, Pierre, Vo, Duc Duy, Gao, Zhan-Guo, Kihlberg, Jan, Jacobson, Kenneth A, Carlsson, Jens

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Adenosine receptors as therapeutic targets von Jacobson, Kenneth A, Gao, Zhan-Guo

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On the G protein-coupling selectivity of the native A2B adenosine receptor von Gao, Zhan-Guo, Inoue, Asuka, Jacobson, Kenneth A.

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Agonist-bound structure of the human P2Y12 receptor von Zhang, Jin, Zhang, Kaihua, Gao, Zhan-Guo, Paoletta, Silvia, Zhang, Dandan, Han, Gye Won, Li, Tingting, Ma, Limin, Zhang, Wenru, Müller, Christa E., Yang, Huaiyu, Jiang, Hualiang, Cherezov, Vadim, Katritch, Vsevolod, Jacobson, Kenneth A., Stevens, Raymond C., Wu, Beili, Zhao, Qiang

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Purinergic Signaling in Mast Cell Degranulation and Asthma von Gao, Zhan-Guo, Jacobson, Kenneth A

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Ligand design by targeting a binding site water von Matricon, Pierre, Suresh, R. Rama, Gao, Zhan-Guo, Panel, Nicolas, Jacobson, Kenneth A, Carlsson, Jens

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Species dependence of A3 adenosine receptor pharmacology and function von Gao, Zhan-Guo, Auchampach, John A., Jacobson, Kenneth A.

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Anionic phospholipids control mechanisms of GPCR-G protein recognition von Thakur, Naveen, Ray, Arka P., Sharp, Liam, Jin, Beining, Duong, Alexander, Pour, Niloofar Gopal, Obeng, Samuel, Wijesekara, Anuradha V., Gao, Zhan-Guo, McCurdy, Christopher R., Jacobson, Kenneth A., Lyman, Edward, Eddy, Matthew T.

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Salvianolic acids from antithrombotic Traditional Chinese Medicine Danshen are antagonists of human P2Y1 and P2Y12 receptors von Liu, Xuyang, Gao, Zhan-Guo, Wu, Yiran, Stevens, Raymond C., Jacobson, Kenneth A., Zhao, Suwen

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Nucleotides Acting at P2Y Receptors: Connecting Structure and Function von Jacobson, Kenneth A., Paoletta, Silvia, Katritch, Vsevolod, Wu, Beili, Gao, Zhan-Guo, Zhao, Qiang, Stevens, Raymond C., Kiselev, Evgeny

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Novel alendronate-CGS21680 conjugate reduces bone resorption and induces new bone formation in post-menopausal osteoporosis and inflammatory osteolysis mouse models von Larrañaga-Vera, Ane, Toti, Kiran S, Flatow, James S, Haraczy, Alexandra J, Warnick, Eugene, Rao, Harsha, Gao, Zhan-Guo, Sussman, Sarah M, Mediero, Aranzazu, Leucht, Philipp, Jacobson, Kenneth A, Cronstein, Bruce N

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Genetic and functional modulation by agonist MRS5698 and allosteric enhancer LUF6000 at the native A3 adenosine receptor in HL-60 cells von Gao, Zhan-Guo, Chen, Weiping, Gao, Ray R., Li, Jonathan, Tosh, Dilip K., Hanover, John A., Jacobson, Kenneth A.

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