syn-1,2-Amino Alcohols via Diastereoselective Allylic C−H Amination von Fraunhoffer, Kenneth J, White, M. Christina

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Macrolactonization via Hydrocarbon Oxidation von FRAUNHOFFER, Kenneth J., PRABAGARAN, Narayanasamy, SIROIS, Lauren E., WHITE, M. Christina

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Hydrocarbon Oxidation vs C−C Bond-Forming Approaches for Efficient Syntheses of Oxygenated Molecules von Fraunhoffer, Kenneth J, Bachovchin, Daniel A, White, M. Christina

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Development of a Practical Synthesis of Functionalized Azaxanthene-Derived Nonsteroidal Glucocorticoid Receptor Modulators von Conlon, David A, Natalie, Kenneth J, Cuniere, Nicolas, Razler, Thomas M, Zhu, Jason, de Mas, Nuria, Tymonko, Steven, Fraunhoffer, Kenneth J, Sortore, Eric, Rosso, Victor W, Xu, Zhongmin, Adams, Monica L, Patel, Anisha, Huang, Jun, Gong, Hua, Weinstein, David S, Quiroz, Fernando, Chen, Doris C

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Sustainable Pd(OAc)2/Hydroquinone Cocatalyst System for Cis‐Selective Dibenzoyloxylation of 1,3‐Cyclohexadiene von Stamoulis, Alexios G., Geng, Peng, Schmidt, Michael A., Eastgate, Martin D., Borovika, Alina, Fraunhoffer, Kenneth J., Stahl, Shannon S.

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Utilizing Native Directing Groups: Synthesis of a Selective IKur Inhibitor, BMS-919373, via a Regioselective C–H Arylation von Wisniewski, Steven R, Stevens, Jason M, Yu, Miao, Fraunhoffer, Kenneth J, Romero, Evan O, Savage, Scott A

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The First Kilogram Synthesis of Beclabuvir, an HCV NS5B Polymerase Inhibitor von Bien, Jeffrey, Davulcu, Akin, DelMonte, Albert J, Fraunhoffer, Kenneth J, Gao, Zhinong, Hang, Chao, Hsiao, Yi, Hu, Wenhao, Katipally, Kishta, Littke, Adam, Pedro, Aghogho, Qiu, Yuping, Sandoval, Maria, Schild, Richard, Soltani, Michelle, Tedesco, Anthony, Vanyo, Dale, Vemishetti, Purushotham, Waltermire, Robert E

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Revisiting the Cleavage of Evans Oxazolidinones with LiOH/H2O2 von Beutner, Gregory L, Cohen, Benjamin M, DelMonte, Albert J, Dixon, Darryl D, Fraunhoffer, Kenneth J, Glace, Andrew W, Lo, Ehrlic, Stevens, Jason M, Vanyo, Dale, Wilbert, Christopher

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Rapid Development of a Commercial Process for Linrodostat, an Indoleamine 2,3-Dioxygenase (IDO) Inhibitor von Fraunhoffer, Kenneth J, DelMonte, Albert J, Beutner, Gregory L, Bultman, Michael S, Camacho, Kathryn, Cohen, Benjamin, Dixon, Darryl D, Fan, Yu, Fanfair, Dayne, Freitag, Adam J, Glace, Andrew W, Gonzalez-Bobes, Francisco, Gujjar, Manjunath, Haley, Matthew W, Hickey, Matthew R, Ho, Jeanne, Iyer, Vidya, Maity, Prantik, Patel, Sunil, Rosso, Victor W, Schmidt, Michael A, Stevens, Jason M, Tan, Yichen, Wilbert, Christopher, Young, Ian S, Yu, Miao

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Utilizing Native Directing Groups: Synthesis of a Selective I Kur Inhibitor, BMS-919373, via a Regioselective C-H Arylation von Wisniewski, Steven R, Stevens, Jason M, Yu, Miao, Fraunhoffer, Kenneth J, Romero, Evan O, Savage, Scott A

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Safe Scale-up of an Oxygen-Releasing Cleavage of Evans Oxazolidinone with Hydrogen Peroxide von Glace, Andrew W, Cohen, Benjamin M, Dixon, Darryl D, Beutner, Gregory L, Vanyo, Dale, Akpinar, Fulya, Rosso, Victor, Fraunhoffer, Kenneth J, DelMonte, Albert J, Santana, Edgar, Wilbert, Christopher, Gallo, Frank, Bartels, William

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Synthesis of Fmoc-Protected Arylphenylalanines (Bip Derivatives) via Nonaqueous Suzuki-Miyaura Cross-Coupling Reactions von Qiao, Jennifer X, Fraunhoffer, Kenneth J, Hsiao, Yi, Li, Yi-Xin, Wang, Chunlei, Wang, Tammy C, Poss, Michael A

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A Scalable Synthesis of 2‑(1,2,4-Oxadiazol-3-yl)propan-2-amine Hydrobromide Using a Process Safety-Driven Protecting Group Strategy von Likhite, Nachiket, Lakshminarasimhan, Thirumalai, Rao, Mallem H. V. Ramana, Shekarappa, Vijaykumar, Sidar, Somprabha, Subramanian, Varadharajan, Fraunhoffer, Kenneth J, Leung, Simon, Vaidyanathan, Rajappa

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Sustainable Pd(OAc)2/Hydroquinone Cocatalyst System for Cis‐Selective Dibenzoyloxylation of 1,3‐Cyclohexadiene von Stamoulis, Alexios G., Geng, Peng, Schmidt, Michael A., Eastgate, Martin D., Borovika, Alina, Fraunhoffer, Kenneth J., Stahl, Shannon S.

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Improving Robustness: In Situ Generation of a Pd(0) Catalyst for the Cyanation of Aryl Bromides von Coombs, John R, Fraunhoffer, Kenneth J, Simmons, Eric M, Stevens, Jason M, Wisniewski, Steven R, Yu, Miao

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Advancing Base Metal Catalysis through Data Science: Insight and Predictive Models for Ni-Catalyzed Borylation through Supervised Machine Learning von Stevens, Jason M., Li, Jun, Simmons, Eric M., Wisniewski, Steven R., DiSomma, Stacey, Fraunhoffer, Kenneth J., Geng, Peng, Hao, Bo, Jackson, Erika W.

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Impact of ICH Q11 Questions and Answers on the Outcome of Active Pharmaceutical Ingredient Starting Material Proposal Acceptance by ICH Regulatory Members von Tymonko, Steven, Burke, Brenda J., Crochard, Jean-Philippe, Dirat, Olivier, Fraunhoffer, Kenneth J., Harrison, Cristian, Kramer, Timothy, Lee, Heewon, Liberman, Vlad, Sidhu, Kanwar P. S., Smith, Randi, Strotman, Neil A., Tandogan, Nil, Triman, Alan, Zhang, Haitao

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Revisiting the Cleavage of Evans Oxazolidinones with LiOH/H 2 O 2 von Beutner, Gregory L., Cohen, Benjamin M., DelMonte, Albert J., Dixon, Darryl D., Fraunhoffer, Kenneth J., Glace, Andrew W., Lo, Ehrlic, Stevens, Jason M., Vanyo, Dale, Wilbert, Christopher

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syn-1,2-Amino Alcohols via Diastereoselective Allylic C-H Amination von Fraunhoffer, Kenneth J., White, M. Christina

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Methods and intermediates for the preparation of (4bS,5aR)-12-cyclohexyl-N-(N,N-dimethylsulfamoyl)-3-methoxy-5a-((1R,5S)-3-methyl-3,8-diazabicyclo [3.2.1]octane-8-carbonyl)-4b,5,5a... von Hang Chao, Natalie, Jr. Kenneth J, Davulcu Akin H, Fraunhoffer Kenneth J, Gao Zhinong, Risatti Christina Ann, Hu Wenhao, DelMonte Albert J

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