Four-Membered Ring-Containing Spirocycles: Synthetic Strategies and Opportunities von Carreira, Erick M, Fessard, Thomas C

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[2]-Ladderanes as isosteres for meta-substituted aromatic rings and rigidified cyclohexanes von Epplin, Rachel C., Paul, Shashwati, Herter, Loïc, Salome, Christophe, Hancock, Erin N., Larrow, Jay F., Baum, Erich W., Dunstan, David R., Ginsburg-Moraff, Carol, Fessard, Thomas C., Brown, M. Kevin

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Improving Nonspecific Binding and Solubility: Bicycloalkyl Groups and Cubanes as para‐Phenyl Bioisosteres von Auberson, Yves P., Brocklehurst, Cara, Furegati, Markus, Fessard, Thomas C., Koch, Guido, Decker, Andrea, La Vecchia, Luigi, Briard, Emmanuelle

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Pushing the Frontiers of Accessible Chemical Space to Unleash Design Creativity and Accelerate Drug Discovery von Fessard, Thomas C., Goncharenko, Kristina, Lefebvre, Quentin, Salomé, Christophe

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Enantioselective Preparation of 1,1-Diarylethanes: Aldehydes as Removable Steering Groups for Asymmetric Synthesis von Fessard, Thomas C, Andrews, Stephen P, Motoyoshi, Hajime, Carreira, Erick M

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Accelerating fragment-based library generation by coupling high-performance photoreactors with benchtop analysis von Lefebvre, Quentin, Salomé, Christophe, Fessard, Thomas C

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Strain-Release [2π + 2σ] Cycloadditions for the Synthesis of Bicyclo[2.1.1]hexanes Initiated by Energy Transfer von Guo, Renyu, Chang, Yu-Che, Herter, Loic, Salome, Christophe, Braley, Sarah E., Fessard, Thomas C., Brown, M. Kevin

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Synthesis of Undecachlorosulfolipid A: Re-evaluation of the Nominal Structure von Nilewski, Christian, Deprez, Nicholas R., Fessard, Thomas C., Li, Dong Bo, Geisser, Roger W., Carreira, Erick M.

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Oxetanyl Peptides: Novel Peptidomimetic Modules for Medicinal Chemistry von McLaughlin, Martin, Yazaki, Ryo, Fessard, Thomas C, Carreira, Erick M

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Nickel‐Photoredox‐Catalyzed Synthesis of sp2−sp3 Fragments and the Impact of Bicycloalkane Isosteric Replacement on Their Physical‐Chemical Properties von Lefebvre, Quentin, Bocu, Mina, Giorgiutti, Christophe, Fessard, Thomas C.

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Synthesis of Borylated Carbocycles by [2 + 2]-Cycloadditions and Photo-Ene Reactions von Posz, Jarett M., Sharma, Neetu, Royalty, Paige A., Liu, Yanyao, Salome, Christophe, Fessard, Thomas C., Brown, M. Kevin

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Diversification of Simple Arenes into Complex (Amino)cyclitols von Angelini, Elisa, Martinelli, Matteo, Roà, Eugenio, Ungarean, Chad N., Salome, Christophe, Lefebvre, Quentin, Bournez, Colin, Fessard, Thomas C., Sarlah, David

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Pd-Catalyzed Cleavage of Benzylic Nitro Bonds: New Opportunities for Asymmetric Synthesis von Fessard, Thomas C., Motoyoshi, Hajime, Carreira, Erick M.

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Reactivity and Selectivity of Azaspirocycles in Radical C–H Functionalization von Ungarean, Chad N., Larin, Egor M., Egger, Dominic T., Ziegler, Philipp, Lefebvre, Quentin, Fessard, Thomas C., Morandi, Bill

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A GAP Replacement, Part 2: Preparation of Poly(3-azidooxetane) via Azidation of Poly(3-tosyloxyoxetane) and Poly(3-mesyloxyoxetane) von Born, Max, Fessard, Thomas C, Göttemann, Lucas, Plank, Jakob, Klapötke, Thomas M

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A Concise and Stereoselective Synthesis of the A-Ring Fragment of the Gambieric Acids von Clark, J. Stephen, Fessard, Thomas C, Wilson, Claire

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3,3-Dinitratooxetane - an important leap towards energetic oxygen-rich monomers and polymers von Born, Max, Fessard, Thomas C, Göttemann, Lucas, Klapötke, Thomas M, Stierstorfer, Jörg, Voggenreiter, Michael

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Energetic but insensitive spiro‐tetrahydrotetrazines based on oxetane‐3‐one von Fessard, Thomas C., Gospodinov, Ivan, Klapötke, Thomas M., Stierstorfer, Jörg, Voggenreiter, Michael

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Identification Of Key Residues For Interaction Of Vasoactive Intestinal Peptide With Human Vpac(1) And Vpac(2) Receptors And Development Of A Highly Selective Vpac(1) Receptor Agon... von Nicole, P., Lins, Laurence, Rouyer-Fessard, C., Drouot, C., Fulcrand, P., Thomas, Annick, Couvineau, A., Martinez, J., Brasseur, Robert, Laburthe, M.

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3-(Nitromethylene)oxetane: a very versatile and promising building block for energetic oxetane based monomers von Born, Max, Fessard, Thomas C, Göttemann, Lucas, Karaghiosoff, Konstantin, Plank, Jakob, Klapötke, Thomas M

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