Thieno[3,2‑b]pyrrole-5-carboxamides as New Reversible Inhibitors of Histone Lysine Demethylase KDM1A/LSD1. Part 2: Structure-Based Drug Design and Structure–Activity Relationship... von Vianello, Paola, Sartori, Luca, Amigoni, Federica, Cappa, Anna, Fagá, Giovanni, Fattori, Raimondo, Legnaghi, Elena, Ciossani, Giuseppe, Mattevi, Andrea, Meroni, Giuseppe, Moretti, Loris, Cecatiello, Valentina, Pasqualato, Sebastiano, Romussi, Alessia, Thaler, Florian, Trifiró, Paolo, Villa, Manuela, Botrugno, Oronza A, Dessanti, Paola, Minucci, Saverio, Vultaggio, Stefania, Zagarrí, Elisa, Varasi, Mario, Mercurio, Ciro

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Thieno[3,2‑b]pyrrole-5-carboxamides as New Reversible Inhibitors of Histone Lysine Demethylase KDM1A/LSD1. Part 1: High-Throughput Screening and Preliminary Exploration von Sartori, Luca, Mercurio, Ciro, Amigoni, Federica, Cappa, Anna, Fagá, Giovanni, Fattori, Raimondo, Legnaghi, Elena, Ciossani, Giuseppe, Mattevi, Andrea, Meroni, Giuseppe, Moretti, Loris, Cecatiello, Valentina, Pasqualato, Sebastiano, Romussi, Alessia, Thaler, Florian, Trifiró, Paolo, Villa, Manuela, Vultaggio, Stefania, Botrugno, Oronza A, Dessanti, Paola, Minucci, Saverio, Zagarrí, Elisa, Carettoni, Daniele, Iuzzolino, Lucia, Varasi, Mario, Vianello, Paola

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Pathogenic Effects of Human Herpesvirus 6 in Human Lymphoid Tissue Ex Vivo von Grivel, Jean-Charles, Santoro, Fabio, Chen, Silvia, Fagá, Giovanni, Malnati, Mauro S, Ito, Yoshinori, Margolis, Leonid, Lusso, Paolo

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Selective transcriptional regulation by Myc in cellular growth control and lymphomagenesis von Sabò, Arianna, Kress, Theresia R., Pelizzola, Mattia, de Pretis, Stefano, Gorski, Marcin M., Tesi, Alessandra, Morelli, Marco J., Bora, Pranami, Doni, Mirko, Verrecchia, Alessandro, Tonelli, Claudia, Fagà, Giovanni, Bianchi, Valerio, Ronchi, Alberto, Low, Diana, Müller, Heiko, Guccione, Ernesto, Campaner, Stefano, Amati, Bruno

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Novel selective inhibitors of macropinocytosis-dependent growth in pancreatic ductal carcinoma von Brambillasca, Silvia, Cera, Maria Rosaria, Andronache, Adrian, Dey, Sumit Kumar, Fagá, Giovanni, Fancelli, Daniele, Frittoli, Emanuela, Pasi, Maurizio, Robusto, Michela, Varasi, Mario, Scita, Giorgio, Mercurio, Ciro

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A multiparametric screen uncovers FDA-approved small molecules that potentiate the nuclear mechano-dysfunctions in ATR-defective cells von Cera, Maria Rosaria, Bastianello, Giulia, Purushothaman, Divya, Andronache, Adrian, Ascione, Flora, Robusto, Michela, Fagà, Giovanni, Pasi, Maurizio, Meroni, Giuseppe, Li, Qingsen, Choudhary, Ramveer, Varasi, Mario, Foiani, Marco, Mercurio, Ciro

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ATR expands embryonic stem cell fate potential in response to replication stress von Atashpaz, Sina, Samadi Shams, Sara, Gonzalez, Javier Martin, Sebestyén, Endre, Arghavanifard, Negar, Gnocchi, Andrea, Albers, Eliene, Minardi, Simone, Faga, Giovanni, Soffientini, Paolo, Allievi, Elisa, Cancila, Valeria, Bachi, Angela, Fernández-Capetillo, Óscar, Tripodo, Claudio, Ferrari, Francesco, López-Contreras, Andrés Joaquin, Costanzo, Vincenzo

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Discovery of Reversible Inhibitors of KDM1A Efficacious in Acute Myeloid Leukemia Models von Romussi, Alessia, Cappa, Anna, Vianello, Paola, Brambillasca, Silvia, Cera, Maria Rosaria, Dal Zuffo, Roberto, Fagà, Giovanni, Fattori, Raimondo, Moretti, Loris, Trifirò, Paolo, Villa, Manuela, Vultaggio, Stefania, Cecatiello, Valentina, Pasqualato, Sebastiano, Dondio, Giulio, So, Chi Wai Eric, Minucci, Saverio, Sartori, Luca, Varasi, Mario, Mercurio, Ciro

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High-throughput screening identifies histone deacetylase inhibitors that modulate GTF2I expression in 7q11.23 microduplication autism spectrum disorder patient-derived cortical neu... von Cavallo, Francesca, Troglio, Flavia, Fagà, Giovanni, Fancelli, Daniele, Shyti, Reinald, Trattaro, Sebastiano, Zanella, Matteo, D'Agostino, Giuseppe, Hughes, James M, Cera, Maria Rosaria, Pasi, Maurizio, Gabriele, Michele, Lazzarin, Maddalena, Mihailovich, Marija, Kooy, Frank, Rosa, Alessandro, Mercurio, Ciro, Varasi, Mario, Testa, Giuseppe

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A high-throughput screening identifies MCM chromatin loading inhibitors targeting cells with increased replication origins von Falbo, Lucia, Técher, Hervé, Sannino, Vincenzo, Robusto, Michela, Fagà, Giovanni, Pezzimenti, Federica, Romeo, Francesco, Colombo, Luca Gabriele, Vultaggio, Stefania, Fancelli, Daniele, Monzani, Silvia, Cecatiello, Valentina, Pasqualato, Sebastiano, Varasi, Mario, Mercurio, Ciro, Costanzo, Vincenzo

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Myc, Cdk2 and cellular senescence: Old players, new game von Campaner, Stefano, Doni, Mirko, Verrecchia, Alessandro, Fagà, Giovanni, Bianchi, Lucia, Amati, Bruno

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Suppression of CCR5- but not CXCR4-tropic HIV-1 in lymphoid tissue by human herpesvirus 6 von Grivel, Jean-Charles, Ito, Yoshinori, Fagà, Giovanni, Santoro, Fabio, Shaheen, Farida, Malnati, Mauro S., Fitzgerald, Wendy, Lusso, Paolo, Margolis, Leonid

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Development of Reverse Transcriptase PCR Assays for Detection of Active Human Herpesvirus 6 Infection von VAN DEN BOSCH, Glenn, LOCATELLI, Giuseppe, GEERTS, Lieve, FAGA, Giovanni, IEVEN, Margareta, GOOSSENS, Herman, BOTTIGER, Disa, ÖBERG, Bo, LUSSO, Paolo, BERNEMAN, Zwi N

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Optimized and Scalable Precoating‐Free Reprogramming of Human Peripheral Blood Mononuclear Cells into iPSCs von Fiacco, Elisabetta, Landi, Sara, Zasso, Jacopo, Ambrosini, Chiara, Faga, Giovanni

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TGFβ-dependent gene expression shows that senescence correlates with abortive differentiation along several lineages in Myc-induced lymphomas von Müller, Judith, Samans, Birgit, van Riggelen, Jan, Fagà, Giovanni, Peh K.N., Raquel, Wei, Chia-Lin, Müller, Heiko, Amati, Bruno, Felsher, Dean, Eilers, Martin

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Dual regulation of Myc by Abl von Sanchez-Arévalo Lobo, V J, Doni, M, Verrecchia, A, Sanulli, S, Fagà, G, Piontini, A, Bianchi, M, Conacci-Sorrell, M, Mazzarol, G, Peg, V, Losa, J H, Ronchi, P, Ponzoni, M, Eisenman, R N, Doglioni, C, Amati, B

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Abstract A44: Selective transcriptional regulation by Myc in growth control and tumorigenesis von Sabò, Arianna, Kress, Theresia K., Pelizzola, Mattia, Pretis, Stefano de, Gorski, Marcin, Tesi, Alessandra, Morelli, Marco J., Bora, Pranami, Doni, Mirko, Verrecchia, Alessandro, Tonelli, Claudia, Fagà, Giovanni, Bianchi, Valerio, Ronchi, Alberto, Low, Diana, Muller, Heiko, Guccione, Ernesto, Campaner, Stefano, Amati, Bruno

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They're not funding government von Faga, Giovanni

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HISTONE DEACETYLASE INHIBITORS AND USES THEREOF von FAGA, Giovanni, TESTA, Giuseppe, FANCELLI, Daniele, CAVALLO, Francesca, TROGLIO, Flavia

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HISTONE DEACETYLASE INHIBITORS AND USES THEREOF von FAGA, Giovanni, TESTA, Giuseppe, FANCELLI, Daniele, CAVALLO, Francesca, TROGLIO, Flavia

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