Improving Nonspecific Binding and Solubility: Bicycloalkyl Groups and Cubanes as para‐Phenyl Bioisosteres von Auberson, Yves P., Brocklehurst, Cara, Furegati, Markus, Fessard, Thomas C., Koch, Guido, Decker, Andrea, La Vecchia, Luigi, Briard, Emmanuelle

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Synthesis of the 3-Aza-[7]-paracyclophane Core of Haouamine A and B von Wipf, Peter, Furegati, Markus

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Practical Isolation of the (1R,2R)‑Enantiomer from a Racemic cis/trans Mixture of 2‑Methyl-1-cyclohexanamine von Furegati, Markus, Nocito, Sandro

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Graphitic Carbon Nitride as a Photocatalyst for Decarboxylative C(sp2)−C(sp3) Couplings via Nickel Catalysis von Lukas, Florian, Findlay, Michael T., Fillols, Méritxell, Templ, Johanna, Savino, Elia, Martin, Benjamin, Allmendinger, Simon, Furegati, Markus, Noël, Timothy

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Scale-Up Synthesis of IID572: A New β‑Lactamase Inhibitor von Furegati, Markus, Nocito, Sandro, Reck, Folkert, Casarez, Anthony, Simmons, Robert, Schuetz, Heiner, Koch, Guido

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Graphitisches Kohlenstoffnitrid als Photokatalysator für die decarboxylative C(sp2)−C(sp3) Kupplung mittels Nickelkatalyse von Lukas, Florian, Findlay, Michael T., Fillols, Méritxell, Templ, Johanna, Savino, Elia, Martin, Benjamin, Allmendinger, Simon, Furegati, Markus, Noël, Timothy

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Synthesis of All Four Stereoisomers of 3‑(tert-Butoxycarbonyl)-3-azabicyclo[3.1.0]hexane-2-carboxylic Acid von Bakonyi, Bettina, Furegati, Markus, Kramer, Christian, La Vecchia, Luigi, Ossola, Flavio

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Potent Nonimmunosuppressive Cyclophilin Inhibitors With Improved Pharmaceutical Properties and Decreased Transporter Inhibition von Fu, Jiping, Tjandra, Meiliana, Becker, Christopher, Bednarczyk, Dallas, Capparelli, Michael, Elling, Robert, Hanna, Imad, Fujimoto, Roger, Furegati, Markus, Karur, Subramanian, Kasprzyk, Theresa, Knapp, Mark, Leung, Kwan, Li, Xiaolin, Lu, Peichao, Mergo, Wosenu, Miault, Charlotte, Ng, Simon, Parker, David, Peng, Yunshan, Roggo, Silvio, Rivkin, Alexey, Simmons, Robert L, Wang, Michael, Wiedmann, Brigitte, Weiss, Andrew H, Xiao, Linda, Xie, Lili, Xu, Wenjian, Yifru, Aregahegn, Yang, Shengtian, Zhou, Bo, Sweeney, Zachary K

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IID572: A New Potentially Best-In-Class β‑Lactamase Inhibitor von Reck, Folkert, Bermingham, Alun, Blais, Johanne, Casarez, Anthony, Colvin, Richard, Dean, Charles R, Furegati, Markus, Gamboa, Luis, Growcott, Ellena, Li, Cindy, Lopez, Sara, Metzger, Louis, Nocito, Sandro, Ossola, Flavio, Phizackerley, Kaci, Rasper, Dita, Shaul, Jacob, Shen, Xiaoyu, Simmons, Robert L, Tang, Dazhi, Tashiro, Kyuto, Yue, Qin

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Discovery of Potent and Selective Antibody–Drug Conjugates with Eg5 Inhibitors through Linker and Payload Optimization von Karpov, Alexei S, Nieto-Oberhuber, Cristina M, Abrams, Tinya, Beng-Louka, Edwige, Blanco, Enrique, Chamoin, Sylvie, Chene, Patrick, Dacquignies, Isabelle, Daniel, Dylan, Dillon, Michael P, Doumampouom-Metoul, Lionel, Drosos, Nikolaos, Fedoseev, Pavel, Furegati, Markus, Granda, Brian, Grotzfeld, Robert M, Hess Clark, Suzanna, Joly, Emilie, Jones, Darryl, Lacaud-Baumlin, Marion, Lagasse-Guerro, Stephanie, Lorenzana, Edward G, Mallet, William, Martyniuk, Piotr, Marzinzik, Andreas L, Mesrouze, Yannick, Nocito, Sandro, Oei, Yoko, Perruccio, Francesca, Piizzi, Grazia, Richard, Etienne, Rudewicz, Patrick J, Schindler, Patrick, Velay, Mélanie, Venstrom, Kristine, Wang, Peiyin, Zurini, Mauro, Lafrance, Marc

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Graphitisches Kohlenstoffnitrid als Photokatalysator für die decarboxylative C(sp 2 )−C(sp 3 ) Kupplung mittels Nickelkatalyse von Lukas, Florian, Findlay, Michael T., Fillols, Méritxell, Templ, Johanna, Savino, Elia, Martin, Benjamin, Allmendinger, Simon, Furegati, Markus, Noël, Timothy

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7-Azaindole-3-acetic acid derivatives: Potent and selective CRTh2 receptor antagonists von Sandham, David A., Adcock, Claire, Bala, Kamlesh, Barker, Lucy, Brown, Zarin, Dubois, Gerald, Budd, David, Cox, Brian, Fairhurst, Robin A., Furegati, Markus, Leblanc, Catherine, Manini, Jodie, Profit, Rachael, Reilly, John, Stringer, Rowan, Schmidt, Alfred, Turner, Katharine L., Watson, Simon J., Willis, Jennifer, Williams, Gareth, Wilson, Caroline

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Unusual base dependent enantioselectivity in a transfer hydrogenation using axially chiral Ir(III)-catalysts von Furegati, Markus, Rippert, Andreas J.

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Benzyl N ‐[(Benzyloxy)methyl]carbamate: An Improved Aminomethylation Electrophile for the Synthesis of (Benzyloxy)carbonyl (Cbz)‐Protected Chiral β 2 ‐Amino Acids von Brocklehurst, Cara E., Furegati, Markus, Müller‐Hartwieg, J. Constanze D., Ossola, Flavio, La Vecchia, Luigi

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Benzyl N-[(Benzyloxy)methyl]carbamate: An Improved Aminomethylation Electrophile for the Synthesis of (Benzyloxy)carbonyl (Cbz)-Protected Chiral β2-Amino Acids von Brocklehurst, Cara E., Furegati, Markus, Müller-Hartwieg, J. Constanze D., Ossola, Flavio, La Vecchia, Luigi

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Optimized Synthesis of l-m-Tyrosine Suitable for Chemical Scale-Up von Humphrey, Cara E, Furegati, Markus, Laumen, Kurt, La Vecchia, Luigi, Leutert, Thomas, Müller-Hartwieg, J. Constanze D, Vögtle, Markus

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(P,M)-1,2,3,9,10,11-Hexa­methoxy-5,7-di­hydro­dibenz­[c,e]­oxepine and (P,M)-1,11-di­methyl-5,5,7,7-tetra­phenyl-5,7-di­hydro­dibenz­[c,e]­oxepine von Linden, Anthony, Furegati, Markus, Rippert, Andreas J.

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An Approach to New, Axially Chiral ζ-Amino Alcohols Using a Ring Opening Reaction von Furegati, Markus, Rippert, Andreas J.

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BICYCLIC HETEROCYCLES AND THEIR USE AS WRN INHIBITORS von ZECRI, Frederic, MOEBITZ, Henrik, FUREGATI, Markus, NOCITO, Sandro, YU, Huangchao, GONG, Wanben, STRANG, Ross, SCHOEPFER, Joseph, HAMON, Jacques, SCHMIEDEBERG, Niko, HINRICHS, Juergen Hans-Hermann

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(P, M)-1,2,3,9,10,11-hexamethoxy-5,7-dihydrodibenz[c, e]oxepine and (P, M)-1,11-dimethyl-5,5,7,7-tetraphenyl-5,7-dihydrodibenz[c, e]oxepine von LINDEN, Anthony, FUREGATI, Markus, RIPPERT, Andreas J

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