The Dynamic Process of β2-Adrenergic Receptor Activation von Nygaard, Rie, Zou, Yaozhong, Dror, Ron O., Mildorf, Thomas J., Arlow, Daniel H., Manglik, Aashish, Pan, Albert C., Liu, Corey W., Fung, Juan José, Bokoch, Michael P., Thian, Foon Sun, Kobilka, Tong Sun, Shaw, David E., Mueller, Luciano, Prosser, R. Scott, Kobilka, Brian K.

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Ligand-specific regulation of the extracellular surface of a G-protein-coupled receptor von Bokoch, Michael P., Zou, Yaozhong, Rasmussen, Søren G. F., Liu, Corey W., Nygaard, Rie, Rosenbaum, Daniel M., Fung, Juan José, Choi, Hee-Jung, Thian, Foon Sun, Kobilka, Tong Sun, Puglisi, Joseph D., Weis, William I., Pardo, Leonardo, Prosser, R. Scott, Mueller, Luciano, Kobilka, Brian K.

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GPC-100, a novel CXCR4 antagonist, improves in vivo hematopoietic cell mobilization when combined with propranolol von Sukhtankar, Devki D., Fung, Juan José, Kim, Mi-na, Cayton, Thomas, Chiou, Valerie, Caculitan, Niña G., Zalicki, Piotr, Kim, Sujeong, Jo, Yoonjung, Kim, SoHui, Lee, Jae Min, Choi, Junhee, Mun, SeongGyeong, Chin, Ashley, Jang, Yongdae, Lee, Ji Yeong, Kim, Gowoon, Kim, Eun Hee, Huh, Won-Ki, Jeong, Jae-Yeon, Seen, Dong-Seung, Cardarelli, Pina M.

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Allosteric coupling from G protein to the agonist-binding pocket in GPCRs von DeVree, Brian T., Mahoney, Jacob P., Vélez-Ruiz, Gisselle A., Rasmussen, Soren G. F., Kuszak, Adam J., Edwald, Elin, Fung, Juan-Jose, Manglik, Aashish, Masureel, Matthieu, Du, Yang, Matt, Rachel A., Pardon, Els, Steyaert, Jan, Kobilka, Brian K., Sunahara, Roger K.

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Nanoscale high-content analysis using compositional heterogeneities of single proteoliposomes von Mathiasen, Signe, Christensen, Sune M, Fung, Juan José, Rasmussen, Søren G F, Fay, Jonathan F, Jorgensen, Sune K, Veshaguri, Salome, Farrens, David L, Kiskowski, Maria, Kobilka, Brian, Stamou, Dimitrios

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A monoclonal antibody for G protein-coupled receptor crystallography von Kobilka, Tong Sun, Weis, William I, Choi, Hee-Jung, Day, Peter W, Masood, Asna, Parnot, Charles, Rasmussen, Søren G F, Fung, Juan José, Yao, Xiao-Jie, Rohrer, Daniel K, Kobilka, Brian K

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Correction: Replication Study: Inhibition of BET recruitment to chromatin as an effective treatment for MLL-fusion leukaemia von Shan, Xiaochuan, Fung, Juan José, Kosaka, Alan, Danet-Desnoyers, Gwenn

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The dynamic process of β(2)-adrenergic receptor activation von Nygaard, Rie, Zou, Yaozhong, Dror, Ron O, Mildorf, Thomas J, Arlow, Daniel H, Manglik, Aashish, Pan, Albert C, Liu, Corey W, Fung, Juan José, Bokoch, Michael P, Thian, Foon Sun, Kobilka, Tong Sun, Shaw, David E, Mueller, Luciano, Prosser, R Scott, Kobilka, Brian K

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Registered report: Inhibition of BET recruitment to chromatin as an effective treatment for MLL-fusion leukemia von Fung, Juan José, Kosaka, Alan, Shan, Xiaochuan, Danet-Desnoyers, Gwenn, Gormally, Michael, Owen, Kate

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High-resolution crystal structure of human protease-activated receptor 1 von Zhang, Cheng, Srinivasan, Yoga, Arlow, Daniel H., Fung, Juan Jose, Palmer, Daniel, Zheng, Yaowu, Green, Hillary F., Pandey, Anjali, Dror, Ron O., Shaw, David E., Weis, William I., Coughlin, Shaun R., Kobilka, Brian K.

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Structure of a nanobody-stabilized active state of the β2 adrenoceptor von Rasmussen, Søren G. F., Choi, Hee-Jung, Fung, Juan Jose, Pardon, Els, Casarosa, Paola, Chae, Pil Seok, DeVree, Brian T., Rosenbaum, Daniel M., Thian, Foon Sun, Kobilka, Tong Sun, Schnapp, Andreas, Konetzki, Ingo, Sunahara, Roger K., Gellman, Samuel H., Pautsch, Alexander, Steyaert, Jan, Weis, William I., Kobilka, Brian K.

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Registered report: androgen receptor splice variants determine taxane sensitivity in prostate cancer von Shan, Xiaochuan, Danet-Desnoyers, Gwenn, Fung, Juan José, Kosaka, Alan H, Tan, Fraser, Perfito, Nicole, Lomax, Joelle, Iorns, Elizabeth

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Ligand-regulated oligomerization of β2-adrenoceptors in a model lipid bilayer von Fung, Juan José, Deupi, Xavier, Pardo, Leonardo, Yao, Xiao Jie, Velez-Ruiz, Gisselle A, DeVree, Brian T, Sunahara, Roger K, Kobilka, Brian K

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Structure-based discovery of β 2 -adrenergic receptor ligands von Kolb, Peter, Rosenbaum, Daniel M., Irwin, John J., Fung, Juan José, Kobilka, Brian K., Shoichet, Brian K.

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Structure-based discovery of β₂-adrenergic receptor ligands von Kolb, Peter, Rosenbaum, Daniel M, Irwin, John J, Fung, Juan José, Kobilka, Brian K, Shoichet, Brian K

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Replication Study: Inhibition of BET recruitment to chromatin as an effective treatment for MLL-fusion leukaemia von Shan, Xiaochuan, Fung, Juan Jose, Kosaka, Alan, Danet-Desnoyers, Gwenn

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1385 Dual Inhibition of DGKα and DGKζ increases T cell and NK cell activity von Schweickert, Patrick G, Reiner, Gabrielle L, Mitchell, Casey G, Piovesan, Dana, Meleza, Cesar, Fung, Juan Jose, Wang, Ning, Cho, Sean, Fournier, Jeremy, Walters, Matthew J, Sivick Gauthier, Kelsey E

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Structure and Conformational Changes in the C-terminal Domain of the β₂-Adrenoceptor: INSIGHTS FROM FLUORESCENCE RESONANCE ENERGY TRANSFER STUDIES von Granier, Sébastien, Kim, Samuel, Shafer, Aaron M, Ratnala, Venkata R.P, Fung, Juan José, Zare, Richard N, Kobilka, Brian

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FRET-Based Measurement of GPCR Conformational Changes von Granier, Sébastien, Kim, Samuel, Fung, Juan José, Bokoch, Michael P., Parnot, Charles

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GPC-100 Is a Novel CXCR4 Inhibitor That Leads to Improved in Vitro Potency and In Vivo Efficacy in Stem Cell Mobilization When Combined with a Beta-Blocker von Fung, Juan Jose, Chiou, Valerie, Lee, Jaemin, Jang, Yongdae, Choi, Junhee, Zalicki, Piotr, Cayton, Thomas, Chin, Ashley, Caculitan, Niña, Kim, SoHui, Lee, Jiyeong, Sukhtankar, Devki, Kim, Eunhee, Cardarelli, Josephine

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