Lessons from crystal structures of kainate receptors von Møllerud, Stine, Frydenvang, Karla, Pickering, Darryl S., Kastrup, Jette Sandholm

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Structure Elucidation of Prenyl- and Geranyl-Substituted Coumarins in Gerbera piloselloides by NMR Spectroscopy, Electronic Circular Dichroism Calculations, and Single Crystal X-ra... von Li, Tuo, Ma, Xue, Fedotov, Daniil, Kjaerulff, Louise, Frydenvang, Karla, Coriani, Sonia, Hansen, Paul Robert, Kongstad, Kenneth T, Staerk, Dan

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Nanoscale Mobility of the Apo State and TARP Stoichiometry Dictate the Gating Behavior of Alternatively Spliced AMPA Receptors von Dawe, G. Brent, Kadir, Md. Fahim, Venskutonytė, Raminta, Perozzo, Amanda M., Yan, Yuhao, Alexander, Ryan P.D., Navarrete, Camilo, Santander, Eduardo A., Arsenault, Marika, Fuentes, Christian, Aurousseau, Mark R.P., Frydenvang, Karla, Barrera, Nelson P., Kastrup, Jette S., Edwardson, J. Michael, Bowie, Derek

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Structure−Activity Relationship Study of First Selective Inhibitor of Excitatory Amino Acid Transporter Subtype 1: 2-Amino-4-(4-methoxyphenyl)-7-(naphthalen-1-yl)-5-oxo-5,6,7,8-tet... von Erichsen, Mette N, Huynh, Tri H. V, Abrahamsen, Bjarke, Bastlund, Jesper F, Bundgaard, Christoffer, Monrad, Olja, Bekker-Jensen, Anders, Nielsen, Christina W, Frydenvang, Karla, Jensen, Anders A, Bunch, Lennart

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Structural analysis of Cytochrome P450 BM3 mutant M11 in complex with dithiothreitol von Frydenvang, Karla, Verkade-Vreeker, Marlies C A, Dohmen, Floor, Commandeur, Jan N M, Rafiq, Maria, Mirza, Osman, Jørgensen, Flemming Steen, Geerke, Daan P

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Thermodynamics and structural analysis of positive allosteric modulation of the ionotropic glutamate receptor GluA2 von Krintel, Christian, Frydenvang, Karla, Olsen, Lars, Kristensen, Maria T, de Barrios, Oriol, Naur, Peter, Francotte, Pierre, Pirotte, Bernard, Gajhede, Michael, Kastrup, Jette S

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Synthesis and Antitumor Effect in Vitro and in Vivo of Substituted 1,3-Dihydroindole-2-ones von Christensen, Mette K, Erichsen, Kamille D, Trojel-Hansen, Christina, Tjørnelund, Jette, Nielsen, Søren J, Frydenvang, Karla, Johansen, Tommy N, Nielsen, Birgitte, Sehested, Maxwell, Jensen, Peter B, Ikaunieks, Martins, Zaichenko, Andrei, Loza, Einars, Kalvinsh, Ivars, Björkling, Fredrik

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Studies on an (S)‑2-Amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic Acid (AMPA) Receptor Antagonist IKM-159: Asymmetric Synthesis, Neuroactivity, and Structural Characterization... von Juknaitė, Lina, Sugamata, Yutaro, Tokiwa, Kazuya, Ishikawa, Yuichi, Takamizawa, Satoshi, Eng, Andrew, Sakai, Ryuichi, Pickering, Darryl S, Frydenvang, Karla, Swanson, Geoffrey T, Kastrup, Jette S, Oikawa, Masato

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Design and Synthesis of 2,3-trans-Proline Analogues as Ligands for Ionotropic Glutamate Receptors and Excitatory Amino Acid Transporters von Poulie, Christian B. M, Alcaide, Anna, Krell-Jørgensen, Mikkel, Larsen, Younes, Astier, Eloi, Bjørn-Yoshimoto, Walden E, Yi, Feng, Syrenne, Jed T, Storgaard, Morten, Nielsen, Birgitte, Frydenvang, Karla A, Jensen, Anders A, Hansen, Kasper B, Pickering, Darryl S, Bunch, Lennart

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Full Domain Closure of the Ligand-binding Core of the Ionotropic Glutamate Receptor iGluR5 Induced by the High Affinity Agonist Dysiherbaine and the Functional Antagonist 8,9-Dideo... von Frydenvang, Karla, Lash, L. Leanne, Naur, Peter, Postila, Pekka A., Pickering, Darryl S., Smith, Caleb M., Gajhede, Michael, Sasaki, Makoto, Sakai, Ryuichi, Pentikaïnen, Olli T., Swanson, Geoffrey T., Kastrup, Jette S.

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Structure-activity relationships of a small-molecule inhibitor of the PDZ domain of PICK1 von Bach, Anders, Stuhr-Hansen, Nicolai, Thorsen, Thor S, Bork, Nicolai, Moreira, Irina S, Frydenvang, Karla, Padrah, Shahrokh, Christensen, S Brøgger, Madsen, Kenneth L, Weinstein, Harel, Gether, Ulrik, Strømgaard, Kristian

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Structural basis for positive allosteric modulation of AMPA and kainate receptors von Frydenvang, Karla, Pickering, Darryl S., Kastrup, Jette Sandholm

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Psychrophilin A and Cycloaspeptide D, Novel Cyclic Peptides from the Psychrotolerant Fungus Penicillium ribeum von DALSGAARD, Petur Weihe, LARSEN, Thomas Ostenfeld, FRYDENVANG, Karla, CHRISTOPHERSEN, Carsten

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Discovery and Structure–Activity Relationships of 2,5-Dimethoxyphenylpiperidines as Selective Serotonin 5‑HT2A Receptor Agonists von M. Ro̷rsted, Emil, Jensen, Anders A., Smits, Gints, Frydenvang, Karla, Kristensen, Jesper L.

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The positive allosteric modulator BPAM344 and L‐glutamate introduce an active‐like structure of the ligand‐binding domain of GluK2 von Bay, Yasmin, Egeberg Jeppesen, Mie, Frydenvang, Karla, Francotte, Pierre, Pirotte, Bernard, Pickering, Darryl S., Kristensen, Anders Skov, Kastrup, Jette Sandholm

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Discovery and Structure-Activity Relationships of 2,5-Dimethoxyphenylpiperidines as Selective Serotonin 5-HT 2A Receptor Agonists von M Ro Rsted, Emil, Jensen, Anders A, Smits, Gints, Frydenvang, Karla, Kristensen, Jesper L

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A Tetrazolyl-Substituted Subtype-Selective AMPA Receptor Agonist von Vogensen, Stine B, Frydenvang, Karla, Greenwood, Jeremy R, Postorino, Giovanna, Nielsen, Birgitte, Pickering, Darryl S, Ebert, Bjarke, Bølcho, Ulrik, Egebjerg, Jan, Gajhede, Michael, Kastrup, Jette S, Johansen, Tommy N, Clausen, Rasmus P, Krogsgaard-Larsen, Povl

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Lessons from more than 80 structures of the GluA2 ligand-binding domain in complex with agonists, antagonists and allosteric modulators von Pøhlsgaard, Jacob, Frydenvang, Karla, Madsen, Ulf, Kastrup, Jette Sandholm

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Identification and Structure-Function Study of Positive Allosteric Modulators of Kainate Receptors von Larsen, Anja Probst, Fièvre, Sabine, Frydenvang, Karla, Francotte, Pierre, Pirotte, Bernard, Kastrup, Jette Sandholm, Mulle, Christophe

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Functionalized Helical β‑Peptoids von Wellhöfer, Isabelle, Frydenvang, Karla, Kotesova, Simona, Christiansen, Andreas M, Laursen, Jonas S, Olsen, Christian A

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