Evaluation of 1H‑Triazole-1‑[N,N′‑Bis(tert-butoxycarbonyl)]carboxamidine in Solution-Phase and On-Resin Guanidinylation von Wester, Anita, Björkling, Fredrik, Franzyk, Henrik

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Evaluation of the topoisomerase II-inactive bisdioxopiperazine ICRF-161 as a protectant against doxorubicin-induced cardiomyopathy von Martin, Elke, Thougaard, Annemette Vinding, Grauslund, Morten, Jensen, Peter B, Bjorkling, Fredrik, Hasinoff, Brian B, Tjørnelund, Jette, Sehested, Maxwell, Jensen, Lars H

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Non-steroidal CYP17A1 Inhibitors: Discovery and Assessment von Wróbel, Tomasz M., Jørgensen, Flemming Steen, Pandey, Amit V., Grudzińska, Angelika, Sharma, Katyayani, Yakubu, Jibira, Björkling, Fredrik

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Polymyxins with Potent Antibacterial Activity against Colistin-Resistant Pathogens: Fine-Tuning Hydrophobicity with Unnatural Amino Acids von Jørgensen, Johan Storm, Mood, Elnaz Harifi, Knap, Anne Sofie Holst, Nielsen, Simone Eidnes, Nielsen, Peter E., Żabicka, Dorota, Matias, Carina, Domraceva, Ilona, Björkling, Fredrik, Franzyk, Henrik

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Peptide/Peptoid Hybrid Oligomers: The Influence of Hydrophobicity and Relative Side-Chain Length on Antibacterial Activity and Cell Selectivity von Frederiksen, Nicki, Hansen, Paul R, Björkling, Fredrik, Franzyk, Henrik

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Optimized Synthesis of Fmoc/Boc‐Protected PNA Monomers and their Assembly into PNA Oligomers von Shaikh, Ashif Y., Björkling, Fredrik, Nielsen, Peter E., Franzyk, Henrik

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Alternating Cationic‐Hydrophobic Peptide/Peptoid Hybrids: Influence of Hydrophobicity on Antibacterial Activity and Cell Selectivity von Frederiksen, Nicki, Hansen, Paul R., Zabicka, Dorota, Tomczak, Magdalena, Urbas, Malgorzata, Domraceva, Ilona, Björkling, Fredrik, Franzyk, Henrik

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Imitation of β-lactam binding enables broad-spectrum metallo-β-lactamase inhibitors von Brem, Jürgen, Panduwawala, Tharindi, Hansen, Jon Ulf, Hewitt, Joanne, Liepins, Edgars, Donets, Pawel, Espina, Laura, Farley, Alistair J. M., Shubin, Kirill, Campillos, Gonzalo Gomez, Kiuru, Paula, Shishodia, Shifali, Krahn, Daniel, Leśniak, Robert K., Schmidt (Adrian), Juliane, Calvopiña, Karina, Turrientes, María-Carmen, Kavanagh, Madeline E., Lubriks, Dmitrijs, Hinchliffe, Philip, Langley, Gareth W., Aboklaish, Ali F., Eneroth, Anders, Backlund, Maria, Baran, Andrei G., Nielsen, Elisabet I., Speake, Michael, Kuka, Janis, Robinson, John, Grinberga, Solveiga, Robinson, Lindsay, McDonough, Michael A., Rydzik, Anna M., Leissing, Thomas M., Jimenez-Castellanos, Juan Carlos, Avison, Matthew B., Da Silva Pinto, Solange, Pannifer, Andrew D., Martjuga, Marina, Widlake, Emma, Priede, Martins, Hopkins Navratilova, Iva, Gniadkowski, Marek, Belfrage, Anna Karin, Brandt, Peter, Yli-Kauhaluoma, Jari, Bacque, Eric, Page, Malcolm G. P., Björkling, Fredrik, Tyrrell, Jonathan M., Spencer, James, Lang, Pauline A., Baranczewski, Pawel, Cantón, Rafael, McElroy, Stuart P., Jones, Philip S., Baquero, Fernando, Suna, Edgars, Morrison, Angus, Walsh, Timothy R., Schofield, Christopher J.

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Silver carbene complexes: An emerging class of anticancer agents von Kankala, Shravankumar, Thota, Niranjan, Björkling, Fredrik, Taylor, Myles K., Vadde, Ravinder, Balusu, Ramesh

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Structure-activity study of oncocin: On-resin guanidinylation and incorporation of homoarginine, 4-hydroxyproline or 4,4-difluoroproline residues von Shaikh, Ashif Y., Björkling, Fredrik, Zabicka, Dorota, Tomczak, Magdalena, Urbas, Malgorzata, Domraceva, Ilona, Kreicberga, Agrita, Franzyk, Henrik

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Peptide/β-Peptoid Hybrids with Ultrashort PEG-Like Moieties: Effects on Hydrophobicity, Antibacterial Activity and Hemolytic Properties von Frederiksen, Nicki, Louka, Stavroula, Mudaliar, Chirag, Domraceva, Ilona, Kreicberga, Agrita, Pugovics, Osvalds, Żabicka, Dorota, Tomczak, Magdalena, Wygoda, Weronika, Björkling, Fredrik, Franzyk, Henrik

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Anticancer agent CHS-828 inhibits cellular synthesis of NAD von Olesen, Uffe Høgh, Christensen, Mette Knak, Björkling, Fredrik, Jäättelä, Marja, Jensen, Peter Buhl, Sehested, Maxwell, Nielsen, Søren Jensby

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Microwave-assisted solid-phase synthesis of antisense acpP peptide nucleic acid-peptide conjugates active against colistin- and tigecycline-resistant E. coli and K. pneumoniae von Hansen, Anna Mette, Bonke, Gitte, Hogendorf, Wouter Frederik Johan, Björkling, Fredrik, Nielsen, John, Kongstad, Kenneth T., Zabicka, Dorota, Tomczak, Magdalena, Urbas, Malgorzata, Nielsen, Peter E., Franzyk, Henrik

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Discovery of Novel Non-Steroidal Cytochrome P450 17A1 Inhibitors as Potential Prostate Cancer Agents von Wróbel, Tomasz M, Rogova, Oksana, Andersen, Kasper L, Yadav, Rahul, Brixius-Anderko, Simone, Scott, Emily E, Olsen, Lars, Jørgensen, Flemming Steen, Björkling, Fredrik

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Selected strategies to fight pathogenic bacteria von Plotniece, Aiva, Sobolev, Arkadij, Supuran, Claudiu T., Carta, Fabrizio, Björkling, Fredrik, Franzyk, Henrik, Yli-Kauhaluoma, Jari, Augustyns, Koen, Cos, Paul, De Vooght, Linda, Govaerts, Matthias, Aizawa, Juliana, Tammela, Päivi, Žalubovskis, Raivis

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Imaging of treatment response to the combination of carboplatin and paclitaxel in human ovarian cancer xenograft tumors in mice using FDG and FLT PET von Munk Jensen, Mette, Erichsen, Kamille Dumong, Björkling, Fredrik, Madsen, Jacob, Jensen, Peter Buhl, Sehested, Maxwell, Højgaard, Liselotte, Kjær, Andreas

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Structural Basis of Metallo-β-lactamase Inhibition by N‑Sulfamoylpyrrole-2-carboxylates von Farley, Alistair J. M, Ermolovich, Yuri, Calvopiña, Karina, Rabe, Patrick, Panduwawala, Tharindi, Brem, Jürgen, Björkling, Fredrik, Schofield, Christopher J

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Synthesis and Antitumor Effect in Vitro and in Vivo of Substituted 1,3-Dihydroindole-2-ones von Christensen, Mette K, Erichsen, Kamille D, Trojel-Hansen, Christina, Tjørnelund, Jette, Nielsen, Søren J, Frydenvang, Karla, Johansen, Tommy N, Nielsen, Birgitte, Sehested, Maxwell, Jensen, Peter B, Ikaunieks, Martins, Zaichenko, Andrei, Loza, Einars, Kalvinsh, Ivars, Björkling, Fredrik

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Nicotinamide Phosphoribosyltransferase Inhibitors, Design, Preparation, and Structure–Activity Relationship von Christensen, Mette K, Erichsen, Kamille D, Olesen, Uffe H, Tjørnelund, Jette, Fristrup, Peter, Thougaard, Annemette, Nielsen, Søren Jensby, Sehested, Maxwell, Jensen, Peter B, Loza, Einars, Kalvinsh, Ivars, Garten, Antje, Kiess, Wieland, Björkling, Fredrik

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Triphenylcarbenium Tetrafluoroborate as an Efficient Catalyst in the Regioselective Reductive Ring Opening of Benzylidene Acetals of Carbohydrates von Thota, Niranjan, Björkling, Fredrik, Kankala, Shravankumar

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