Pyridylpiperazine-based allosteric inhibitors of RND-type multidrug efflux pumps von Plé, Coline, Tam, Heng-Keat, Vieira Da Cruz, Anais, Compagne, Nina, Jiménez-Castellanos, Juan-Carlos, Müller, Reinke T., Pradel, Elizabeth, Foong, Wuen Ee, Malloci, Giuliano, Ballée, Alexia, Kirchner, Moritz A., Moshfegh, Parisa, Herledan, Adrien, Herrmann, Andrea, Deprez, Benoit, Willand, Nicolas, Vargiu, Attilio Vittorio, Pos, Klaas M., Flipo, Marion, Hartkoorn, Ruben C.

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Combination therapy for tuberculosis treatment: pulmonary administration of ethionamide and booster co-loaded nanoparticles von Costa-Gouveia, Joana, Pancani, Elisabetta, Jouny, Samuel, Machelart, Arnaud, Delorme, Vincent, Salzano, Giuseppina, Iantomasi, Raffaella, Piveteau, Catherine, Queval, Christophe J., Song, Ok-Ryul, Flipo, Marion, Deprez, Benoit, Saint-André, Jean-Paul, Hureaux, José, Majlessi, Laleh, Willand, Nicolas, Baulard, Alain, Brodin, Priscille, Gref, Ruxandra

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Update on the Discovery of Efflux Pump Inhibitors against Critical Priority Gram-Negative Bacteria von Compagne, Nina, Vieira Da Cruz, Anais, Müller, Reinke T, Hartkoorn, Ruben C, Flipo, Marion, Pos, Klaas M

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Molecular Design in Practice: A Review of Selected Projects in a French Research Institute That Illustrates the Link between Chemical Biology and Medicinal Chemistry von Deprez, Benoit, Bosc, Damien, Charton, Julie, Couturier, Cyril, Deprez-Poulain, Rebecca, Flipo, Marion, Leroux, Florence, Villemagne, Baptiste, Willand, Nicolas

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Rapid and Efficient Access to Novel Bio-Inspired 3-Dimensional Tricyclic SpiroLactams as Privileged Structures via Meyers' Lactamization von Tangara, Salia, Faïon, Léo, Piveteau, Catherine, Capet, Frédéric, Godelier, Romain, Michel, Marion, Flipo, Marion, Deprez, Benoit, Willand, Nicolas, Villemagne, Baptiste

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Exploring the Antitubercular Activity of Anthranilic Acid Derivatives: From MabA (FabG1) Inhibition to Intrabacterial Acidification von Faïon, Léo, Djaout, Kamel, Pintiala, Catalin, Piveteau, Catherine, Leroux, Florence, Biela, Alexandre, Slupek, Stéphanie, Antoine, Rudy, Záhorszká, Monika, Cantrelle, Francois-Xavier, Hanoulle, Xavier, Korduláková, Jana, Deprez, Benoit, Willand, Nicolas, Baulard, Alain R, Flipo, Marion

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On the Hunt for Next-Generation Antimicrobial Agents: An Online Symposium Organized Jointly by the French Society for Medicinal Chemistry (Société de Chimie Thérapeutique) and the... von Antraygues, Kevin, Compagne, Nina, Ruggieri, Francesca, Djaout, Kamel, Edoo, Zainab, Eveque, Maxime, Faïon, Léo, Gioia, Bruna, Tangara, Salia, Vieira Da Cruz, Anais, Villemagne, Baptiste, Flipo, Marion, Baulard, Alain, Willand, Nicolas

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Publisher Correction: Combination therapy for tuberculosis treatment: pulmonary administration of ethionamide and booster co-loaded nanoparticles von Costa-Gouveia, Joana, Pancani, Elisabetta, Jouny, Samuel, Machelart, Arnaud, Delorme, Vincent, Salzano, Giuseppina, Iantomasi, Raffaella, Piveteau, Catherine, Queval, Christophe J., Song, Ok-Ryul, Flipo, Marion, Deprez, Benoit, Saint-André, Jean-Paul, Hureaux, José, Majlessi, Laleh, Willand, Nicolas, Baulard, Alain, Brodin, Priscille, Gref, Ruxandra

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Antibiotics with novel mode of action as new weapons to fight antimicrobial resistance von Ruggieri, Francesca, Compagne, Nina, Antraygues, Kevin, Eveque, Maxime, Flipo, Marion, Willand, Nicolas

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Reversion of antibiotic resistance in Mycobacterium tuberculosis by spiroisoxazoline SMARt-420 von Blondiaux, Nicolas, Moune, Martin, Desroses, Matthieu, Frita, Rosangela, Flipo, Marion, Mathys, Vanessa, Soetaert, Karine, Kiass, Mehdi, Delorme, Vincent, Djaout, Kamel, Trebosc, Vincent, Kemmer, Christian, Wintjens, René, Wohlkönig, Alexandre, Antoine, Rudy, Huot, Ludovic, Hot, David, Coscolla, Mireia, Feldmann, Julia, Gagneux, Sebastien, Locht, Camille, Brodin, Priscille, Gitzinger, Marc, Déprez, Benoit, Willand, Nicolas, Baulard, Alain R.

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Tuberculosis: The drug development pipeline at a glance von Villemagne, Baptiste, Crauste, Céline, Flipo, Marion, Baulard, Alain R., Déprez, Benoit, Willand, Nicolas

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Microwave-assisted synthesis of functionalized spirohydantoins as 3-D privileged fragments for scouting the chemical space von Prevet, Hugues, Flipo, Marion, Roussel, Pascal, Deprez, Benoit, Willand, Nicolas

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Synthesis of functionalized 2-isoxazolines as three-dimensional fragments for fragment-based drug discovery von Tran, Ngoc Chau, Dhondt, Heleen, Flipo, Marion, Deprez, Benoit, Willand, Nicolas

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Intrinsic Antibacterial Activity of Nanoparticles Made of β‑Cyclodextrins Potentiates Their Effect as Drug Nanocarriers against Tuberculosis von Machelart, Arnaud, Salzano, Giuseppina, Li, Xue, Demars, Aurore, Debrie, Anne-Sophie, Menendez-Miranda, Mario, Pancani, Elisabetta, Jouny, Samuel, Hoffmann, Eik, Deboosere, Nathalie, Belhaouane, Imène, Rouanet, Carine, Simar, Sophie, Talahari, Smaïl, Giannini, Valerie, Villemagne, Baptiste, Flipo, Marion, Brosch, Roland, Nesslany, Fabrice, Deprez, Benoit, Muraille, Eric, Locht, Camille, Baulard, Alain R, Willand, Nicolas, Majlessi, Laleh, Gref, Ruxandra, Brodin, Priscille

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Tricyclic SpiroLactams Kill Mycobacteria In Vitro and In Vivo by Inhibiting Type II NADH Dehydrogenases von Dam, Sushovan, Tangara, Salia, Hamela, Claire, Hattabi, Theo, Faïon, Léo, Carre, Paul, Antoine, Rudy, Herledan, Adrien, Leroux, Florence, Piveteau, Catherine, Eveque, Maxime, Flipo, Marion, Deprez, Benoit, Kremer, Laurent, Willand, Nicolas, Villemagne, Baptiste, Hartkoorn, Ruben C.

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Hydroxamates: Relationships between Structure and Plasma Stability von Flipo, Marion, Charton, Julie, Hocine, Akila, Dassonneville, Sandrine, Deprez, Benoit, Deprez-Poulain, Rebecca

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Optimization of pyridylpiperazine-based inhibitors of the Escherichia coli AcrAB-TolC efflux pump von Compagne, Nina, Jiménez-Castellanos, Juan-Carlos, Meurillon, Virginie, Pradel, Elizabeth, Vieira Da Cruz, Anais, Piveteau, Catherine, Biela, Alexandre, Eveque, Maxime, Leroux, Florence, Deprez, Benoit, Willand, Nicolas, Hartkoorn, Ruben C., Flipo, Marion

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Discovery of the first Mycobacterium tuberculosis MabA (FabG1) inhibitors through a fragment-based screening von Faïon, Léo, Djaout, Kamel, Frita, Rosangela, Pintiala, Catalin, Cantrelle, Francois-Xavier, Moune, Martin, Vandeputte, Alexandre, Bourbiaux, Kevin, Piveteau, Catherine, Herledan, Adrien, Biela, Alexandre, Leroux, Florence, Kremer, Laurent, Blaise, Mickael, Tanina, Abdalkarim, Wintjens, René, Hanoulle, Xavier, Déprez, Benoit, Willand, Nicolas, Baulard, Alain R., Flipo, Marion

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Ligand Efficiency Driven Design of New Inhibitors of Mycobacterium tuberculosis Transcriptional Repressor EthR Using Fragment Growing, Merging, and Linking Approaches von Villemagne, Baptiste, Flipo, Marion, Blondiaux, Nicolas, Crauste, Céline, Malaquin, Sandra, Leroux, Florence, Piveteau, Catherine, Villeret, Vincent, Brodin, Priscille, Villoutreix, Bruno O, Sperandio, Olivier, Soror, Sameh H, Wohlkönig, Alexandre, Wintjens, René, Deprez, Benoit, Baulard, Alain R, Willand, Nicolas

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Pyridylpiperazine efflux pump inhibitor boosts in vivo antibiotic efficacy against K. pneumoniae von Vieira Da Cruz, Anais, Jiménez-Castellanos, Juan-Carlos, Börnsen, Clara, Van Maele, Laurye, Compagne, Nina, Pradel, Elizabeth, Müller, Reinke T, Meurillon, Virginie, Soulard, Daphnée, Piveteau, Catherine, Biela, Alexandre, Dumont, Julie, Leroux, Florence, Deprez, Benoit, Willand, Nicolas, Pos, Klaas M, Frangakis, Achilleas S, Hartkoorn, Ruben C, Flipo, Marion

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