Crystallographic and electrophilic fragment screening of the SARS-CoV-2 main protease von Douangamath, Alice, Fearon, Daren, Gehrtz, Paul, Krojer, Tobias, Lukacik, Petra, Owen, C. David, Resnick, Efrat, Strain-Damerell, Claire, Aimon, Anthony, Ábrányi-Balogh, Péter, Brandão-Neto, José, Carbery, Anna, Davison, Gemma, Dias, Alexandre, Downes, Thomas D., Dunnett, Louise, Fairhead, Michael, Firth, James D., Jones, S. Paul, Keeley, Aaron, Keserü, György M., Klein, Hanna F., Martin, Mathew P., Noble, Martin E. M., O’Brien, Peter, Powell, Ailsa, Reddi, Rambabu N., Skyner, Rachael, Snee, Matthew, Waring, Michael J., Wild, Conor, London, Nir, von Delft, Frank, Walsh, Martin A.

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Synthesis of Enantiopure Piperazines via Asymmetric Lithiation–Trapping of N‑Boc Piperazines: Unexpected Role of the Electrophile and Distal N‑Substituent von Firth, James D, O’Brien, Peter, Ferris, Leigh

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Deciphering complexity in Pd–catalyzed cross-couplings von Clarke, George E., Firth, James D., Ledingham, Lyndsay A., Horbaczewskyj, Chris S., Bourne, Richard A., Bray, Joshua T. W., Martin, Poppy L., Eastwood, Jonathan B., Campbell, Rebecca, Pagett, Alex, MacQuarrie, Duncan J., Slattery, John M., Lynam, Jason M., Whitwood, Adrian C., Milani, Jessica, Hart, Sam, Wilson, Julie, Fairlamb, Ian J. S.

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An Experimental and in Situ IR Spectroscopic Study of the Lithiation–Substitution of N-Boc-2-phenylpyrrolidine and -piperidine: Controlling the Formation of Quaternary Stereocenter... von Sheikh, Nadeem S, Leonori, Daniele, Barker, Graeme, Firth, James D, Campos, Kevin R, Meijer, Anthony J. H. M, O’Brien, Peter, Coldham, Iain

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A Need for Caution in the Preparation and Application of Synthetically Versatile Aryl Diazonium Tetrafluoroborate Salts von Firth, James D, Fairlamb, Ian J. S

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Gram‐Scale Synthesis of the (−)‐Sparteine Surrogate and (−)‐Sparteine von Firth, James D., Canipa, Steven J., Ferris, Leigh, O'Brien, Peter

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Diastereoselective Synthesis of 4-Hydroxypiperidin-2-ones via Cu(I)-Catalyzed Reductive Aldol Cyclization von Lam, Hon Wai, Murray, Gordon J, Firth, James D

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α‐Functionalisation of Cyclic Sulfides Enabled by Lithiation Trapping von Seling, Nico, Atobe, Masakazu, Kasten, Kevin, Firth, James D., Karadakov, Peter B., Goldberg, Frederick W., O'Brien, Peter

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Lipopolysaccharide-Induced Epithelial Monoamine Oxidase Mediates Alveolar Bone Loss in a Rat Chronic Wound Model von Ekuni, Daisuke, Firth, James D, Nayer, Tarun, Tomofuji, Takaaki, Sanbe, Toshihiro, Irie, Koichiro, Yamamoto, Tatsuo, Oka, Takashi, Liu, Zhenzi, Vielkind, Juergen, Putnins, Edward E

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General Procedures for the Lithiation/Trapping of N‑Boc Piperazines von Firth, James D, O’Brien, Peter, Ferris, Leigh

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Cross-Coupling Knows No Limits: Assessing the Synthetic Potential of the Palladium-Catalysed Cross-Coupling of Organolithiums von Firth, James D., O'Brien, Peter

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Design and Synthesis of 56 Shape‐Diverse 3D Fragments von Downes, Thomas D., Jones, S. Paul, Klein, Hanna F., Wheldon, Mary C., Atobe, Masakazu, Bond, Paul S., Firth, James D., Chan, Ngai S., Waddelove, Laura, Hubbard, Roderick E., Blakemore, David C., De Fusco, Claudia, Roughley, Stephen D., Vidler, Lewis R., Whatton, Maria Ann, Woolford, Alison J.‐A., Wrigley, Gail L., O'Brien, Peter

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Fusobacterium nucleatum Increases Collagenase 3 Production and Migration of Epithelial Cells von Uitto, Veli-Jukka, Baillie, Daniel, Wu, Qiang, Gendron, Renee, Grenier, Daniel, Putnins, Edward E, Kanervo, Arja, Firth, James D

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Revisiting the sparteine surrogate: development of a resolution route to the (-)-sparteine surrogate von Firth, James D, O'Brien, Peter, Ferris, Leigh

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An in vitro analysis of mechanical wounding-induced ligand-independent KGFR activation von Li, Min, Firth, James D, Putnins, Edward E

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Light‐ and Manganese‐Initiated Borylation of Aryl Diazonium Salts: Mechanistic Insight on the Ultrafast Time‐Scale Revealed by Time‐Resolved Spectroscopic Analysis von Firth, James D., Hammarback, L. Anders, Burden, Thomas J., Eastwood, Jonathan B., Donald, James R., Horbaczewskyj, Chris S., McRobie, Matthew T., Tramaseur, Adam, Clark, Ian P., Towrie, Michael, Robinson, Alan, Krieger, Jean‐Philippe, Lynam, Jason M., Fairlamb, Ian J. S.

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Increase of enzyme activity through specific covalent modification with fragments von Darby, John F, Atobe, Masakazu, Firth, James D, Bond, Paul, Davies, Gideon J, O'Brien, Peter, Hubbard, Roderick E

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Mechanical Induction of an Epithelial Cell Chymase Associated with Wound Edge Migration von Firth, James D., Uitto, Veli-Jukka, Putnins, Edward E.

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Fragment-derived modulators of an industrial beta-glucosidase von Makraki, Eleni, Darby, John F., Carneiro, Marta G., Firth, James D., Heyam, Alex, Eiso, A. B., O'Brien, Peter, Siegal, Gregg, Hubbard, Roderick E.

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A biosynthesis-inspired approach to over twenty diverse natural product-like scaffolds von Firth, James D, Craven, Philip G E, Lilburn, Matthew, Pahl, Axel, Marsden, Stephen P, Nelson, Adam

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