A Ring-Closing Metathesis (RCM)-Based Approach to Mycolactones A/B von Gersbach, Philipp, Jantsch, Andrea, Feyen, Fabian, Scherr, Nicole, Dangy, Jean-Pierre, Pluschke, Gerd, Altmann, Karl-Heinz

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Synthesis and evaluation of the antitumor agent TMC-69-6H and a focused library of analogs von Fürstner, Alois, Feyen, Fabian, Prinz, Heino, Waldmann, Herbert

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Making Epothilones Fluoresce: Design, Synthesis, and Biological Characterization of a Fluorescent N12-Aza-Epothilone (Azathilone) von Gertsch, Jürg, Feyen, Fabian, Bützberger, Alexander, Gerber, Barbara, Pfeiffer, Bernhard, Altmann, Karl-Heinz

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Natural products as leads for anticancer drug discovery: discovery of new chemotypes of microtubule stabilizers through reengineering of the epothilone scaffold von Altmann, Karl-Heinz, Cachoux, Frédéric, Feyen, Fabian, Gertsch, Jürg, Kuzniewski, Christian N, Wartmann, Markus

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Synthesis and Biological Activity of 12-Aza-Epothilones (Azathilones) – Non-Natural Natural Products with Potent Antiproliferative Activity von Feyen, Fabian, Gertsch, Jürg, Wartmann, Markus, Altmann, Karl-Heinz

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A Ring-Closing Metathesis (RCM)-Based Approach to MycolactonesA/B von Gersbach, Philipp, Jantsch, Andrea, Feyen, Fabian, Scherr, Nicole, Dangy, Jean-Pierre, Pluschke, Gerd, Altmann, Karl-Heinz

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Epothilones as Lead Structures for the Synthesis-Based Discovery of New Chemotypes for Microtubule Stabilization von Feyen, Fabian, Cachoux, Frédéric, Gertsch, Jürg, Wartmann, Markus, Altmann, Karl-Heinz

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Synthetic Studies on Mycolactones: Synthesis of the Mycolactone Core ­Structure through Ring-Closing Olefin Metathesis von Feyen, Fabian, Jantsch, Andrea, Altmann, Karl-Heinz

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Total Synthesis and Reassessment of the Phosphatase-Inhibitory Activity of the Antitumor Agent TMC-69-6H von Fürstner, Alois, Feyen, Fabian, Prinz, Heino, Waldmann, Herbert

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Synthesis of 12-aza analogs of epothilones and ( E)-9,10-dehydroepothilones von Feyen, Fabian, Jantsch, Andrea, Hauenstein, Kurt, Pfeiffer, Bernhard, Altmann, Karl-Heinz

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Design and Synthesis of 12-Aza-Epothilones (Azathilones)-"Non-Natural" Natural Products with Potent Anticancer Activity von Feyen, Fabian, Gertsch, Jürg, Wartmann, Markus, Altmann, Karl-Heinz

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Cover Picture: Making Epothilones Fluoresce: Design, Synthesis, and Biological Characterization of a Fluorescent N12-Aza-Epothilone (Azathilone) (ChemBioChem 15/2009) von Gertsch , Jürg, Feyen , Fabian, Bützberger, Alexander, Gerber, Barbara, Pfeiffer, Bernhard, Altmann, Karl-Heinz

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PROCESS FOR THE SYNTHESIS OF 4-((R)-2-{[6-((S)-3-METHOXY-PYRROLIDIN-1-YL)-2-PHENYL-PYRIMIDINE-4-CARBONYL]-AMINO}-3-PHOSPHONO-PROPIONYL)-PIPERAZINE-1-CARBOXYLIC ACID BUTYL ESTER von CLAVEAU, Romain, HALL, Leanne, HUGHES, Stephen, REBER, Stefan, FEYEN, Fabian, BLUMER, Nicole

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A PROCESS FOR THE SYNTHESIS OF 4-((R)-2-{[6-((S)-3-METHOXY-PYRROLIDIN-1-YL)-2-PHENYL- PYRIMIDINE-4-CARBONYL]-AMINO}-3-PHOSPHONO-PROPIONYL)-PIPERAZINE-1 -CARBOXYLIC ACID BUTYL ESTER von CLAVEAU, Romain, HALL, Leanne, HUGHES, Stephen, REBER, Stefan, FEYEN, Fabian, BLUMER, Nicole

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A process for the synthesis of 4-((r)-2-{[6-((s)-3-methoxy-pyrrolidin-1-yl)-2-phenyl- pyrimidine-4-carbonyl]-amino}-3-phosphono-propionyl)-piperazine-1 -carboxylic acid butyl ester von CLAVEAU Romain, REBER Stefan, HALL Leanne, FEYEN Fabian, HUGHES Stephen, BLUMER Nicole

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A PROCESS FOR THE SYNTHESIS OF 4-((R)-2-{[6-((S)-3-METHOXY-PYRROL IDIN-1-YL)-2-PHENYL- PYRIMIDINE-4-CARBONYL]-AMINO}-3-PHOSPHONO-PR OPIONYL)-PIPERAZINE-1 -CARBOXYLIC ACID BUTYL EST... von CLAVEAU Romain, REBER Stefan, HALL Leanne, FEYEN Fabian, HUGHES Stephen, BLUMER Nicole

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A PROCESS FOR THE SYNTHESIS OF 4-((R)-2-{[6-((S)-3-METHOXY-PYRROLIDIN-1-YL)-2-PHENYL- PYRIMIDINE-4-CARBONYL]-AMINO}-3-PHOSPHONO-PROPIONYL)-PIPERAZINE-1 -CARBOXYLIC ACID BUTYL ESTER von CLAVEAU, Romain, HALL, Leanne, HUGHES, Stephen, REBER, Stefan, FEYEN, Fabian, BLUMER, Nicole

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A PROCESS FOR THE SYNTHESIS OF 4-((R)-2-{[6-((S)-3-METHOXY-PYRROLIDIN-1-YL)-2-PHENYL- PYRIMIDINE-4-CARBONYL]-AMINO}-3-PHOSPHONO-PROPIONYL)-PIPERAZINE-1 -CARBOXYLIC ACID BUTYL ESTER von CLAVEAU, Romain, HALL, Leanne, HUGHES, Stephen, REBER, Stefan, FEYEN, Fabian, BLUMER, Nicole

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A PROCESS FOR THE SYNTHESIS OF 4-((R)-2-{[6-((S)-3-METHOXY-PYRROLIDIN-1-YL)-2-PHENYL- PYRIMIDINE-4-CARBONYL]-AMINO}-3-PHOSPHONO-PROPIONYL)-PIPERAZINE-1 -CARBOXYLIC ACID BUTYL ESTER von REBER, STEFAN, BLUMER, NICOLE, FEYEN, FABIAN, HALL, LEANNE, HUGHES, STEPHEN, CLAVEAU, ROMAIN

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Entwurf und Synthese von 12-Aza-Epothilonen (Azathilonen) - "nicht-natürliche Naturstoffe" mit potenter Antitumorwirkung von Feyen, Fabian, Gertsch, Jürg, Wartmann, Markus, Altmann, Karl-Heinz

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