Rapid and direct control of target protein levels with VHL-recruiting dTAG molecules von Nabet, Behnam, Ferguson, Fleur M., Seong, Bo Kyung A., Kuljanin, Miljan, Leggett, Alan L., Mohardt, Mikaela L., Robichaud, Amanda, Conway, Amy S., Buckley, Dennis L., Mancias, Joseph D., Bradner, James E., Stegmaier, Kimberly, Gray, Nathanael S.

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A bump-and-hole approach to engineer controlled selectivity of BET bromodomain chemical probes von Baud, Matthias G. J., Lin-Shiao, Enrique, Cardote, Teresa, Tallant, Cynthia, Pschibul, Annica, Chan, Kwok-Ho, Zengerle, Michael, Garcia, Jordi R., Kwan, Terence T.-L., Ferguson, Fleur M., Ciulli, Alessio

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Targeted degradation of aberrant tau in frontotemporal dementia patient-derived neuronal cell models von Silva, M Catarina, Ferguson, Fleur M, Cai, Quan, Donovan, Katherine A, Nandi, Ghata, Patnaik, Debasis, Zhang, Tinghu, Huang, Hai-Tsang, Lucente, Diane E, Dickerson, Bradford C, Mitchison, Timothy J, Fischer, Eric S, Gray, Nathanael S, Haggarty, Stephen J

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Kinase inhibitors: the road ahead von Ferguson, Fleur M., Gray, Nathanael S.

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Molecular Basis of Histone Tail Recognition by Human TIP5 PHD Finger and Bromodomain of the Chromatin Remodeling Complex NoRC von Tallant, Cynthia, Valentini, Erica, Fedorov, Oleg, Overvoorde, Lois, Ferguson, Fleur M., Filippakopoulos, Panagis, Svergun, Dmitri I., Knapp, Stefan, Ciulli, Alessio

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A biotin targeting chimera (BioTAC) system to map small molecule interactomes in situ von Tao, Andrew J., Jiang, Jiewei, Gadbois, Gillian E., Goyal, Pavitra, Boyle, Bridget T., Mumby, Elizabeth J., Myers, Samuel A., English, Justin G., Ferguson, Fleur M.

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Harnessing Antibody-Mimetic Selectivity for Activation-State-Specific Targeted Degradation of Endogenous K‑Ras von Ferguson, Fleur M

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PROTACs reach clinical development in inflammatory skin disease von Ferguson, Fleur M.

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Targeting Low-Druggability Bromodomains: Fragment Based Screening and Inhibitor Design against the BAZ2B Bromodomain von Ferguson, Fleur M, Fedorov, Oleg, Chaikuad, Apirat, Philpott, Martin, Muniz, Joao R. C, Felletar, Ildiko, von Delft, Frank, Heightman, Tom, Knapp, Stefan, Abell, Chris, Ciulli, Alessio

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Discovery and Optimization of Tau Targeted Protein Degraders Enabled by Patient Induced Pluripotent Stem Cells-Derived Neuronal Models of Tauopathy von Silva, M Catarina, Nandi, Ghata, Donovan, Katherine A, Cai, Quan, Berry, Bethany C, Nowak, Radoslaw P, Fischer, Eric S, Gray, Nathanael S, Ferguson, Fleur M, Haggarty, Stephen J

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Tuned out von Ferguson, Fleur M.

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Editorial: E3 ubiquitin ligases: From structure to physiology to therapeutics, Volume II von Licchesi, Julien D F, Laman, Heike, Ikeda, Fumiyo, Ferguson, Fleur M, Bolanos-Garcia, Victor M

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Application of induced proximity for therapeutic discovery von Cacace, Angela, Daniels, Danette, Ferguson, Fleur M., Mayor-Ruiz, Cristina, Woo, Christina

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Mapping the Degradable Kinome Provides a Resource for Expedited Degrader Development von Donovan, Katherine A., Ferguson, Fleur M., Bushman, Jonathan W., Eleuteri, Nicholas A., Bhunia, Debabrata, Ryu, SeongShick, Tan, Li, Shi, Kun, Yue, Hong, Liu, Xiaoxi, Dobrovolsky, Dennis, Jiang, Baishan, Wang, Jinhua, Hao, Mingfeng, You, Inchul, Teng, Mingxing, Liang, Yanke, Hatcher, John, Li, Zhengnian, Manz, Theresa D., Groendyke, Brian, Hu, Wanyi, Nam, Yunju, Sengupta, Sandip, Cho, Hanna, Shin, Injae, Agius, Michael P., Ghobrial, Irene M., Ma, Michelle W., Che, Jianwei, Buhrlage, Sara J., Sim, Taebo, Gray, Nathanael S., Fischer, Eric S.

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Binding Hotspots of BAZ2B Bromodomain: Histone Interaction Revealed by Solution NMR Driven Docking von Ferguson, Fleur M, Dias, David M, Rodrigues, João P. G. L. M, Wienk, Hans, Boelens, Rolf, Bonvin, Alexandre M. J. J, Abell, Chris, Ciulli, Alessio

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Selective Mediator dependence of cell-type-specifying transcription von Jaeger, Martin G., Schwalb, Björn, Mackowiak, Sebastian D., Velychko, Taras, Hanzl, Alexander, Imrichova, Hana, Brand, Matthias, Agerer, Benedikt, Chorn, Someth, Nabet, Behnam, Ferguson, Fleur M., Müller, André C., Bergthaler, Andreas, Gray, Nathanael S., Bradner, James E., Bock, Christoph, Hnisz, Denes, Cramer, Patrick, Winter, Georg E.

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A new avenue for molecular glues: Rapid discovery of a NFKB1 degrader von Fan, Angela T., Boyle, Bridget T., Ferguson, Fleur M.

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Making transient complexes stick von Wang, YiYu, Mouli, M. S. S. Vinod, Ma, Min, Ferguson, Fleur M.

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Assembling a Robust Workflow for Characterizing Endogenous E3 Ligase Substrates von Tao, Andrew J, Ferguson, Fleur M

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TRIM8 modulates the EWS/FLI oncoprotein to promote survival in Ewing sarcoma von Seong, Bo Kyung A., Dharia, Neekesh V., Lin, Shan, Donovan, Katherine A., Chong, Shasha, Robichaud, Amanda, Conway, Amy, Hamze, Amanda, Ross, Linda, Alexe, Gabriela, Adane, Biniam, Nabet, Behnam, Ferguson, Fleur M., Stolte, Björn, Wang, Emily Jue, Sun, Jialin, Darzacq, Xavier, Piccioni, Federica, Gray, Nathanael S., Fischer, Eric S., Stegmaier, Kimberly

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