An update on therapeutic opportunities offered by cancer glycolytic metabolism von Granchi, Carlotta, Fancelli, Daniele, Minutolo, Filippo

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PHA-739358, a potent inhibitor of Aurora kinases with a selective target inhibition profile relevant to cancer von Carpinelli, Patrizia, Ceruti, Roberta, Giorgini, Maria Laura, Cappella, Paolo, Gianellini, Laura, Croci, Valter, Degrassi, Anna, Texido, Gemma, Rocchetti, Maurizio, Vianello, Paola, Rusconi, Luisa, Storici, Paola, Zugnoni, Paola, Arrigoni, Claudio, Soncini, Chiara, Alli, Cristina, Patton, Veronica, Marsiglio, Aurelio, Ballinari, Dario, Pesenti, Enrico, Fancelli, Daniele, Moll, Jürgen

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High-throughput screening identifies histone deacetylase inhibitors that modulate GTF2I expression in 7q11.23 microduplication autism spectrum disorder patient-derived cortical neu... von Cavallo, Francesca, Troglio, Flavia, Fagà, Giovanni, Fancelli, Daniele, Shyti, Reinald, Trattaro, Sebastiano, Zanella, Matteo, D'Agostino, Giuseppe, Hughes, James M, Cera, Maria Rosaria, Pasi, Maurizio, Gabriele, Michele, Lazzarin, Maddalena, Mihailovich, Marija, Kooy, Frank, Rosa, Alessandro, Mercurio, Ciro, Varasi, Mario, Testa, Giuseppe

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PHA-680632, a Novel Aurora Kinase Inhibitor with Potent Antitumoral Activity von Soncini, Chiara, Carpinelli, Patrizia, Gianellini, Laura, Fancelli, Daniele, Vianello, Paola, Rusconi, Luisa, Storici, Paola, Zugnoni, Paola, Pesenti, Enrico, Croci, Valter, Ceruti, Roberta, Giorgini, Maria Laura, Cappella, Paolo, Ballinari, Dario, Sola, Francesco, Varasi, Mario, Bravo, Rodrigo, Moll, Jürgen

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A high-throughput screening identifies MCM chromatin loading inhibitors targeting cells with increased replication origins von Falbo, Lucia, Técher, Hervé, Sannino, Vincenzo, Robusto, Michela, Fagà, Giovanni, Pezzimenti, Federica, Romeo, Francesco, Colombo, Luca Gabriele, Vultaggio, Stefania, Fancelli, Daniele, Monzani, Silvia, Cecatiello, Valentina, Pasqualato, Sebastiano, Varasi, Mario, Mercurio, Ciro, Costanzo, Vincenzo

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Quantitative Chemical Proteomics Identifies Novel Targets of the Anti-cancer Multi-kinase Inhibitor E-3810 von Colzani, Mara, Noberini, Roberta, Romanenghi, Mauro, Colella, Gennaro, Pasi, Maurizio, Fancelli, Daniele, Varasi, Mario, Minucci, Saverio, Bonaldi, Tiziana

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Novel selective inhibitors of macropinocytosis-dependent growth in pancreatic ductal carcinoma von Brambillasca, Silvia, Cera, Maria Rosaria, Andronache, Adrian, Dey, Sumit Kumar, Fagá, Giovanni, Fancelli, Daniele, Frittoli, Emanuela, Pasi, Maurizio, Robusto, Michela, Varasi, Mario, Scita, Giorgio, Mercurio, Ciro

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Cinnamic Anilides as New Mitochondrial Permeability Transition Pore Inhibitors Endowed with Ischemia-Reperfusion Injury Protective Effect in Vivo von Fancelli, Daniele, Abate, Agnese, Amici, Raffaella, Bernardi, Paolo, Ballarini, Marco, Cappa, Anna, Carenzi, Giacomo, Colombo, Andrea, Contursi, Cristina, Di Lisa, Fabio, Dondio, Giulio, Gagliardi, Stefania, Milanesi, Eva, Minucci, Saverio, Pain, Gilles, Pelicci, Pier Giuseppe, Saccani, Alessandra, Storto, Mariangela, Thaler, Florian, Varasi, Mario, Villa, Manuela, Plyte, Simon

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GNX-4728, a novel small molecule drug inhibitor of mitochondrial permeability transition, is therapeutic in a mouse model of amyotrophic lateral sclerosis von Martin, Lee J, Fancelli, Daniele, Wong, Margaret, Niedzwiecki, Mark, Ballarini, Marco, Plyte, Simon, Chang, Qing

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1,4,5,6-Tetrahydropyrrolo[3,4-c]pyrazoles:  Identification of a Potent Aurora Kinase Inhibitor with a Favorable Antitumor Kinase Inhibition Profile von Fancelli, Daniele, Moll, Jürgen, Varasi, Mario, Bravo, Rodrigo, Artico, Roberta, Berta, Daniela, Bindi, Simona, Cameron, Alexander, Candiani, Ilaria, Cappella, Paolo, Carpinelli, Patrizia, Croci, Walter, Forte, Barbara, Giorgini, Maria Laura, Klapwijk, Jan, Marsiglio, Aurelio, Pesenti, Enrico, Rocchetti, Maurizio, Roletto, Fulvia, Severino, Dino, Soncini, Chiara, Storici, Paola, Tonani, Roberto, Zugnoni, Paola, Vianello, Paola

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Crystal structure of the T315I abl mutant in complex with the aurora kinases inhibitor PHA-739358 von MODUGNO, Michele, CASALE, Elena, ISACCHI, Antonella, MOLL, Jürgen, SONCINI, Chiara, ROSETTANI, Pamela, COLOMBO, Riccardo, LUPI, Rosita, RUSCONI, Luisa, FANCELLI, Daniele, CARPINELLI, Patrizia, CAMERON, Alexander D

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Compounds and methods for inhibiting mitotic progression: Millennium Pharmaceuticals Inc.: US20050256102 von Fancelli, Daniele

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Potent and Selective Aurora Inhibitors Identified by the Expansion of a Novel Scaffold for Protein Kinase Inhibition von Fancelli, Daniele, Berta, Daniela, Bindi, Simona, Cameron, Alexander, Cappella, Paolo, Carpinelli, Patrizia, Catana, Cornel, Forte, Barbara, Giordano, Patrizia, Giorgini, Maria Laura, Mantegani, Sergio, Marsiglio, Aurelio, Meroni, Maurizio, Moll, Juergen, Pittalà, Valeria, Roletto, Fulvia, Severino, Dino, Soncini, Chiara, Storici, Paola, Tonani, Roberto, Varasi, Mario, Vulpetti, Anna, Vianello, Paola

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Thieno[3,2- c]pyrazoles: A novel class of Aurora inhibitors with favorable antitumor activity von Bindi, Simona, Fancelli, Daniele, Alli, Cristina, Berta, Daniela, Bertrand, Jay A., Cameron, Alexander D., Cappella, Paolo, Carpinelli, Patrizia, Cervi, Giovanni, Croci, Valter, D’Anello, Matteo, Forte, Barbara, Laura Giorgini, M., Marsiglio, Aurelio, Moll, Juergen, Pesenti, Enrico, Pittalà, Valeria, Pulici, Maurizio, Riccardi-Sirtori, Federico, Roletto, Fulvia, Soncini, Chiara, Storici, Paola, Varasi, Mario, Volpi, Daniele, Zugnoni, Paola, Vianello, Paola

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3-Amino-1,4,5,6-tetrahydropyrrolo[3,4- c]pyrazoles: A new class of CDK2 inhibitors von Pevarello, Paolo, Fancelli, Daniele, Vulpetti, Anna, Amici, Raffaella, Villa, Manuela, Pittalà, Valeria, Vianello, Paola, Cameron, Alexander, Ciomei, Marina, Mercurio, Ciro, Bischoff, James R., Roletto, Fulvia, Varasi, Mario, Brasca, Maria Gabriella

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Manganese(III) acetate-induced cyclization of .alpha.-(arylalkyl) and .alpha.-(aryloxy)alkyl .beta.-dicarbonyl derivatives von Citterio, Attilio, Fancelli, Daniele, Finzi, Claudia, Pesce, Luca, Santi, Roberto

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Inhibitors of Aurora kinases for the treatment of cancer von Fancelli, Daniele, Moll, Jürgen

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Solid phase synthesis of 2-substituted benzofurans via the palladium-catalysed heteroannulation of acetylenes von Fancelli, Daniele, Fagnola, Maria Chiara, Severino, Dino, Bedeschi, Angelo

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6-Substituted Pyrrolo[3,4-c]pyrazoles: An Improved Class of CDK2 Inhibitors von Brasca, Maria Gabriella, Albanese, Clara, Amici, Raffaella, Ballinari, Dario, Corti, Luca, Croci, Valter, Fancelli, Daniele, Fiorentini, Francesco, Nesi, Marcella, Orsini, Paolo, Orzi, Fabrizio, Pastori, Wilma, Perrone, Ettore, Pesenti, Enrico, Pevarello, Paolo, Riccardi-Sirtori, Federico, Roletto, Fulvia, Roussel, Patrick, Varasi, Mario, Vulpetti, Anna, Mercurio, Ciro

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SUBSTITUTED PYRROLO-PYRAZOLE DERIVATIVES AS KINASE INHIBITORS von PEVARELLO PAOLO, ORZI FABRIZIO, ROUSSEL PATRICK, NESI MARCELLA, AMICI RAFFAELLA, FANCELLI DANIELE, VULPETTI ANNA, BRASCA MARIA GABRIELLA, ORSINI PAOLO

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