Discovery and Preclinical Evaluation of [4-[[1-(3-fluorophenyl)methyl]-1H-indazol-5-ylamino]-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yl]carbamic Acid, (3S)-3-Morpholinylmethyl Ester... von Gavai, Ashvinikumar V, Fink, Brian E, Fairfax, David J, Martin, Gregory S, Rossiter, Lana M, Holst, Christian L, Kim, Soong-Hoon, Leavitt, Kenneth J, Mastalerz, Harold, Han, Wen-Ching, Norris, Derek, Goyal, Bindu, Swaminathan, Shankar, Patel, Bharat, Mathur, Arvind, Vyas, Dolatrai M, Tokarski, John S, Yu, Chiang, Oppenheimer, Simone, Zhang, Hongjian, Marathe, Punit, Fargnoli, Joseph, Lee, Francis Y, Wong, Tai W, Vite, Gregory D

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Discovery of 2-substituted benzoxazole carboxamides as 5-HT3 receptor antagonists von Yang, Zhicai, Fairfax, David J., Maeng, Jun-Ho, Masih, Liaqat, Usyatinsky, Alexander, Hassler, Carla, Isaacson, Soshanna, Fitzpatrick, Kevin, DeOrazio, Russell J., Chen, Jianqing, Harding, James P., Isherwood, Matthew, Dobritsa, Svetlana, Christensen, Kevin L., Wierschke, Jonathan D., Bliss, Brian I., Peterson, Lisa H., Beer, Cathy M., Cioffi, Christopher, Lynch, Michael, Rennells, W. Martin, Richards, Justin J., Rust, Timothy, Khmelnitsky, Yuri L., Cohen, Marlene L., Manning, David D.

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A comparative study of the decomposition of o-alkynyl-substituted aryl diazo ketones. Synthesis of polysubstituted .beta.-naphthols via arylketene intermediates von Padwa, Albert, Chiacchio, Ugo, Fairfax, David J, Kassir, Jamal M, Litrico, Angelo, Semones, Mark A, Xu, Simon L

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An enantioselective synthesis of nitrogen protected 3-arylserine esters von Bourdon, Lisa H., Fairfax, David J., Martin, Gregory S., Mathison, Casey J., Zhichkin, Pavel

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Preparation of 5-(2-Methoxy-4-nitrophenyl)oxazole:  A Key Intermediate for the Construction of VX-497 von Herr, R. Jason, Fairfax, David J, Meckler, Harold, Wilson, Jeffrey D

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A General Procedure for the Synthesis of 2-Substituted Pyrimidine-5-Carboxylic Esters von Zhichkin, Pavel, Fairfax, David J., Eisenbeis, Shane A.

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Stereo and electronic effects in the rhodium(II)-mediated synthesis of polycyclic lactones and lactams from .alpha.-diazo ester and amide precursors von Padwa, Albert, Dean, Dennis C, Fairfax, David J, Xu, Simon L

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An efficient one-pot, two-step synthesis of 4-substituted 1-heteroarylpiperazines under microwave irradiation conditions von Wang, Hong-Jun, Earley, William G., Lewis, Robert M., Srivastava, Rajiv R., Zych, Andrew J., Jenkins, David M., Fairfax, David J.

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A One-Pot Method for the Synthesis of Naphthyridines via Modified Friedländer Reaction von Zhichkin, Pavel, Beer, Catherine M., Rennells, W. Martin, Fairfax, David J.

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Discovery of 2-substituted benzoxazole carboxamides as 5-HT sub(3) receptor antagonists von Yang, Zhicai, Fairfax, David J, Maeng, Jun-Ho, Masih, Liaqat, Usyatinsky, Alexander, Hassler, Carla, Isaacson, Soshanna, Fitzpatrick, Kevin, DeOrazio, Russell J, Chen, Jianqing, Harding, James P, Isherwood, Matthew, Dobritsa, Svetlana, Christensen, Kevin L, Wierschke, Jonathan D, Bliss, Brian I, Peterson, Lisa H, Beer, Cathy M, Cioffi, Christopher, Lynch, Michael

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Discovery and Preclinical Evaluation of [4-[[1-(3-fluorophenyl)methyl]-1 H -indazol-5-ylamino]-5-methylpyrrolo[2,1- f ][1,2,4]triazin-6-yl]carbamic Acid, (3 S )-3-Morpholinylmethyl... von Gavai, Ashvinikumar V., Fink, Brian E., Fairfax, David J., Martin, Gregory S., Rossiter, Lana M., Holst, Christian L., Kim, Soong-Hoon, Leavitt, Kenneth J., Mastalerz, Harold, Han, Wen-Ching, Norris, Derek, Goyal, Bindu, Swaminathan, Shankar, Patel, Bharat, Mathur, Arvind, Vyas, Dolatrai M., Tokarski, John S., Yu, Chiang, Oppenheimer, Simone, Zhang, Hongjian, Marathe, Punit, Fargnoli, Joseph, Lee, Francis Y., Wong, Tai W., Vite, Gregory D.

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STORAGE STABLE FORMULATIONS OF SULFATED GLYCOSAMINOGLYCANS AND FRAGMENTS DERIVED THEREFROM FOR THE TREATMENT OF PAIN AND OTHER MEDICAL CONDITIONS von FAIRFAX, David J, VAUGHN, Thomas Michael, QUINN, John, D'AMBRA, Thomas Edward, POPP, Karl F

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Storage stable formulations of sulfated glycosaminoglycans and fragments derived therefrom for the treatment of pain and other medical conditions von Vaughn, Thomas Michael, Quinn, John, D'Ambra, Thomas Edward, Fairfax, David J, Popp, Karl F

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Alternatives to α-diazo ketones for tandem cyclization-cycloaddition and carbenoid-alkyne metathesis strategies. Novel cyclic enol-ether formation via carbonyl ylide rearrangement... von FAIRFAX, D. J, AUSTIN, D. J, XU, S. L, PADWA, A

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STORAGE STABLE FORMULATIONS OF SULFATED GLYCOSAMINOGLYCANS AND FRAGMENTS DERIVED THEREFROM FOR THE TREATMENT OF PAIN AND OTHER MEDICAL CONDITIONS von FAIRFAX, David J, HARRISON, Joshua Alan, VAUGHN, Thomas Michael, QUINN, John, D'AMBRA, Thomas Edward, POPP, Karl F

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STORAGE STABLE FORMULATIONS OF SULFATED GLYCOSAMINOGLYCANS AND FRAGMENTS DERIVED THEREFROM FOR THE TREATMENT OF PAIN AND OTHER MEDICAL CONDITIONS von FAIRFAX, David J, HARRISON, Joshua Alan, VAUGHN, Thomas Michael, QUINN, John, D'AMBRA, Thomas Edward, POPP, Karl F

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composto, composição farmacêutica, e, método de tratamento de um distúrbio von ZHICAI YANG, DAVID J. FAIRFAX

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4-fluoro-4-arylpiperdin-1-yl derivatives as mu opioid function moderators von FAIRFAX DAVID J

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4-FLUORO-4-ARYLPIPERDIN-1-YL DERIVATIVES AS MU OPIOID FUNCTION MODERATORS von FAIRFAX DAVID J

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4-FLUORO-4-ARYLPIPERDIN-1-YL DERIVATIVES AS MU OPIOID FUNCTION MODERATORS von FAIRFAX, DAVID J

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