Macrocyclization as a Source of Desired Polypharmacology. Discovery of Triple PI3K/mTOR/PIM Inhibitors von Martínez-González, Sonia, Alvarez, Rosa M, Martín, José I, García, Ana Belén, Riesco-Fagundo, Concepción, Varela, Carmen, Rodríguez Hergueta, Antonio, González Cantalapiedra, Esther, Albarrán, M. I, Gómez-Casero, Elena, Cebriá, Antonio, Aguirre, Enara, Ajenjo, Nuria, Cebrián, David, Di Geronimo, Bruno, Cunningham, Darren, O’Neill, Michael, Dave, Harish P. G, Blanco-Aparicio, Carmen, Pastor, Joaquín

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Synthesis of C3 Benzo[1,2-e:3,4-e′:5,6-e′′]tribenzo[l]acephenanthrylenes ("Crushed Fullerene" Derivatives) by Intramolecular Palladium-Catalyzed Arylation von Gómez-Lor, Berta, González-Cantalapiedra, Esther, Ruiz, Marta, de Frutos, Óscar, Cárdenas, Diego J., Santos, Amelia, Echavarren, Antonio M.

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Synthesis of a Crushed Fullerene C60H24 through Sixfold Palladium-Catalyzed Arylation von Dorel, Ruth, de Mendoza, Paula, Calleja, Pilar, Pascual, Sergio, González-Cantalapiedra, Esther, Cabello, Noemí, Echavarren, Antonio M.

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PIM kinases as potential therapeutic targets in a subset of peripheral T cell lymphoma cases von Martín-Sánchez, Esperanza, Odqvist, Lina, Rodríguez-Pinilla, Socorro M, Sánchez-Beato, Margarita, Roncador, Giovanna, Domínguez-González, Beatriz, Blanco-Aparicio, Carmen, García Collazo, Ana M, Cantalapiedra, Esther González, Fernández, Joaquín Pastor, Curiel del Olmo, Soraya, Pisonero, Helena, Madureira, Rebeca, Almaraz, Carmen, Mollejo, Manuela, Alves, F Javier, Menárguez, Javier, González-Palacios, Fernando, Rodríguez-Peralto, José Luis, Ortiz-Romero, Pablo L, Real, Francisco X, García, Juan F, Bischoff, James R, Piris, Miguel A

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Synthesis of the Benzo[b]fluorene Core of the Kinamycins by Arylalkyne-Allene and Arylalkyne-Alkyne Cycloadditions von González-Cantalapiedra, Esther, de Frutos, Óscar, Atienza, Carmen, Mateo, Cristina, Echavarren, Antonio M.

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Omipalisib inspired macrocycles as dual PI3K/mTOR inhibitors von Álvarez, Rosa M., García, Ana Belén, Riesco-Fagundo, Concepción, Martín, José I., Varela, Carmen, Rodríguez Hergueta, Antonio, González Cantalapiedra, Esther, Oyarzabal, Julen, Di Geronimo, Bruno, Lorenzo, Milagros, Albarrán, M Isabel, Cebriá, Antonio, Cebrián, David, Martínez-González, Sonia, Blanco-Aparicio, Carmen, Pastor, Joaquín

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Discovery of novel triazolo[4,3-b]pyridazin-3-yl-quinoline derivatives as PIM inhibitors von Martínez-González, Sonia, Rodríguez-Arístegui, Sonsoles, Gómez de la Oliva, Cristina Ana, Hernández, Ana Isabel, González Cantalapiedra, Esther, Varela, Carmen, García, Ana Belén, Rabal, Obdulia, Oyarzabal, Julen, Bischoff, James R., Klett, Javier, Albarrán, María Isabel, Cebriá, Antonio, Ajenjo, Nuria, García-Serelde, Beatriz, Gómez-Casero, Elena, Cuadrado-Urbano, Manuel, Cebrián, David, Blanco-Aparicio, Carmen, Pastor, Joaquín

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Generation of tricyclic imidazo[1,2-a]pyrazines as novel PI3K inhibitors by application of a conformational restriction strategy von Martínez González, Sonia, Rodríguez-Arístegui, Sonsoles, Hernández, Ana Isabel, Varela, Carmen, González Cantalapiedra, Esther, Álvarez, Rosa María, Rodríguez Hergueta, Antonio, Bischoff, James R., Albarrán, María Isabel, Cebriá, Antonio, Cendón, Elena, Cebrián, David, Alfonso, Patricia, Pastor, Joaquín

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New Building Blocks Based on Truxene Cores: Synthesis of Functionalized syn-Tri- and -Hexasubstituted Derivatives von González-Cantalapiedra, Esther, Ruiz, Marta, Gómez-Lor, Berta, Alonso, Beatriz, García-Cuadrado, Domingo, Cárdenas, Diego J., Echavarren, Antonio M.

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Corrigendum to <’ Omipalisib inspired macrocycles as dual PI3K/mTOR inhibitors’ [Eur. J. Med. Chem. 211 (2021), 113109] von Alvarez, Rosa M., García, Ana Belén, Riesco-Fagundo, Concepción, Martín, José I., Varela, Carmen, Rodríguez Hergueta, Antonio, González Cantalapiedra, Esther, Oyarzabal, Julen, Di Geronimo, Bruno, Lorenzo, Milagros, Albarrán, M Isabel, Cebriá, Antonio, Cebrián, David, Martínez-González, Sonia, Blanco-Aparicio, Carmen, Pastor, Joaquín

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Molecular Panels for Energy Transduction in C 60 -Based Conjugates von Sánchez, Luis, Martín, Nazario, González-Cantalapiedra, Esther, Echavarren, Antonio M., Aminur Rahman, G. M., Guldi, Dirk M.

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Synthesis of C 3 Benzo[1,2‐ e :3,4‐ e ′:5,6‐ e ′′]tribenzo[ l ]acephenanthrylenes (“Crushed Fullerene” Derivatives) by Intramolecular Palladium‐Catalyzed Arylation... von Gómez‐Lor, Berta, González‐Cantalapiedra, Esther, Ruiz, Marta, de Frutos, Óscar, Cárdenas, Diego J., Santos, Amelia, Echavarren, Antonio M.

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Molecular Panels for Energy Transduction in C60-Based Conjugates von Sánchez, Luis, Martín, Nazario, González-Cantalapiedra, Esther, Echavarren, Antonio M, Aminur Rahman, G. M, Guldi, Dirk M

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COMPOUNDS von BLANCO APARICIO, Carmen, CEBRIÁ GÓMEZ, Antonio, ALBARRÁN SANTIÑO, María Isabel, ÁLVAREZ ESCOBAR, Rosa María, MARTÍN HERNANDO, Jose Ignacio, RIESCO FAGUNDO, Rosario Concepción, GARCÍA GARCÍA, Ana Belén, GONZÁLEZ CANTALAPIEDRA, Esther, HERNÁNDEZ ENCINAS, Elena, RAMOS LIMA, Francisco Javier, GÓMEZ DE LA OLIVA, Cristina Ana, FERNÁNDEZ, Joaquin Pastor, CEBRIÁN MUÑOZ, David Álvaro, MARTÍNEZ GONZÁLEZ, Sonia

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COMPOUNDS von BLANCO APARICIO, Carmen, CEBRIÁ GÓMEZ, Antonio, ALBARRÁN SANTIÑO, María Isabel, ÁLVAREZ ESCOBAR, Rosa María, MARTÍN HERNANDO, Jose Ignacio, RIESCO FAGUNDO, Rosario Concepción, GARCÍA GARCÍA, Ana Belén, GONZÁLEZ CANTALAPIEDRA, Esther, HERNÁNDEZ ENCINAS, Elena, RAMOS LIMA, Francisco Javier, GÓMEZ DE LA OLIVA, Cristina Ana, FERNÁNDEZ, Joaquin Pastor, CEBRIÁN MUÑOZ, David Álvaro, MARTÍNEZ GONZÁLEZ, Sonia

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IMIDAZO[1,2-A]PYRAZINES AS INHIBITORS OF HASPIN AND THERAPEUTIC USES THEREOF von GONZÁLEZ CANTALAPIEDRA, Esther, PASTOR FERNÁNDEZ, Joaquín, CEBRIÁ GÓMEZ, Antonio, PASTOR FERNÁNDEZ, Miryam, BLANCO-APARICIO, Carmen, ALBARRÁN SANTIÑO, María Isabel, MALUMBRES MARTÍNEZ, Marcos, GARCÍA GARCÍA, Ana Belén, MARTÍNEZ GONZÁLEZ, Sonia, HERNÁNDEZ HIGUERAS, Ana Isabel

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IMIDAZO[1,2-A]PYRAZINES AS INHIBITORS OF HASPIN AND THERAPEUTIC USES THEREOF von GONZÁLEZ CANTALAPIEDRA, Esther, PASTOR FERNÁNDEZ, Joaquín, CEBRIÁ GÓMEZ, Antonio, PASTOR FERNÁNDEZ, Miryam, BLANCO-APARICIO, Carmen, ALBARRÁN SANTIÑO, María Isabel, GARCÍA GARCÍA, Ana Belén, MARTÍNEZ GONZÁLEZ, Sonia, HERNÁNDEZ HIGUERAS, Ana Isabel

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COMPOUNDS von BLANCO APARICIO, Carmen, CEBRIÁ GÓMEZ, Antonio, ALBARRÁN SANTIÑO, María Isabel, ÁLVAREZ ESCOBAR, Rosa María, MARTÍN HERNANDO, Jose Ignacio, RIESCO FAGUNDO, Rosario Concepción, GARCÍA GARCÍA, Ana Belén, GONZÁLEZ CANTALAPIEDRA, Esther, HERNÁNDEZ ENCINAS, Elena, RAMOS LIMA, Francisco Javier, GÓMEZ DE LA OLIVA, Cristina Ana, FERNÁNDEZ, Joaquin Pastor, CEBRIÁN MUÑOZ, David Álvaro, MARTÍNEZ GONZÁLEZ, Sonia

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Synthesis of a Crushed Fullerene C60H24 through Sixfold Palladium-Catalyzed Arylation von Dorel, Ruth, de Mendoza, Paula, Calleja, Pilar, Pascual, Sergio, González-Cantalapiedra, Esther, Cabello, Noemí, Echavarren, Antonio M

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PIM Kinases as Potential Therapeutic Targets in a Subset of Peripheral T Cell Lymphoma Cases: e112148 von Martin-Sanchez, Esperanza, Odqvist, Lina, Rodriguez-Pinilla, Socorro M, Sanchez-Beato, Margarita, Roncador, Giovanna, Dominguez-Gonzalez, Beatriz, Blanco-Aparicio, Carmen, Collazo, Ana MGarcia, Cantalapiedra, Esther Gonzalez, Fernandez, Joaquin Pastor

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