Pharmacokinetic-pharmacodynamic correlation from mouse to human with pazopanib, a multikinase angiogenesis inhibitor with potent antitumor and antiangiogenic activity von Kumar, Rakesh, Knick, Victoria B, Rudolph, Sharon K, Johnson, Jennifer H, Crosby, Renae M, Crouthamel, Ming-Chih, Hopper, Teresa M, Miller, Charles G, Harrington, Laura E, Onori, James A, Mullin, Robert J, Gilmer, Tona M, Truesdale, Anne T, Epperly, Andrea H, Boloor, Amogh, Stafford, Jeffrey A, Luttrell, Deirdre K, Cheung, Mui

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Discovery of 5-[[4-[(2,3-Dimethyl-2H-indazol-6-yl)methylamino]-2-pyrimidinyl]amino]-2-methyl-benzenesulfonamide (Pazopanib), a Novel and Potent Vascular Endothelial Growth Factor R... von Harris, Philip A, Boloor, Amogh, Cheung, Mui, Kumar, Rakesh, Crosby, Renae M, Davis-Ward, Ronda G, Epperly, Andrea H, Hinkle, Kevin W, Hunter, Robert N, Johnson, Jennifer H, Knick, Victoria B, Laudeman, Christopher P, Luttrell, Deirdre K, Mook, Robert A, Nolte, Robert T, Rudolph, Sharon K, Szewczyk, Jerzy R, Truesdale, Anne T, Veal, James M, Wang, Liping, Stafford, Jeffrey A

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Discovery of thiophene inhibitors of polo-like kinase von Emmitte, Kyle A., Andrews, C. Webb, Badiang, Jennifer G., Davis-Ward, Ronda G., Dickson, Hamilton D., Drewry, David H., Emerson, Holly K., Epperly, Andrea H., Hassler, Daniel F., Knick, Victoria B., Kuntz, Kevin W., Lansing, Timothy J., Linn, James A., Mook, Robert A., Nailor, Kristen E., Salovich, James M., Spehar, Glenn M., Cheung, Mui

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Discovery and Evaluation of 2-Anilino-5-aryloxazoles as a Novel Class of VEGFR2 Kinase Inhibitors von Harris, Philip A, Cheung, Mui, Hunter, Robert N, Brown, Matthew L, Veal, James M, Nolte, Robert T, Wang, Liping, Liu, Wendy, Crosby, Renae M, Johnson, Jennifer H, Epperly, Andrea H, Kumar, Rakesh, Luttrell, Deirdre K, Stafford, Jeffrey A

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The identification of pyrazolo[1,5- a]pyridines as potent p38 kinase inhibitors von Cheung, Mui, Harris, Philip A., Badiang, Jennifer G., Peckham, Gregory E., Chamberlain, Stanley D., Alberti, Michael J., Jung, David K., Harris, Stephanie S., Bramson, Neal H., Epperly, Andrea H., Stimpson, Stephen A., Peel, Michael R.

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Tetrahydroquinoline derivatives as opioid receptor antagonists von Zhang, Cunyu, Westaway, Susan M., Speake, Jason D., Bishop, Michael J., Goetz, Aaron S., Carballo, Luz Helena, Hu, Mike, Epperly, Andrea H.

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Phenoxyacetic acids as PPARδ partial agonists: Synthesis, optimization, and in vivo efficacy von Evans, Karen A., Shearer, Barry G., Wisnoski, David D., Shi, Dongchuan, Sparks, Steven M., Sternbach, Daniel D., Winegar, Deborah A., Billin, Andrew N., Britt, Christy, Way, James M., Epperly, Andrea H., Leesnitzer, Lisa M., Merrihew, Raymond V., Xu, Robert X., Lambert, Millard H., Jin, Jian

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Amino acid anthranilamide derivatives as a new class of glycogen phosphorylase inhibitors von Evans, Karen A., Li, Yue H., Coppo, Frank T., Graybill, Todd L., Cichy-Knight, Maria, Patel, Mehul, Gale, Jennifer, Li, Hu, Thrall, Sara H., Tew, David, Tavares, Francis, Thomson, Stephen A., Weiel, James E., Boucheron, Joyce A., Clancy, Daphne C., Epperly, Andrea H., Golden, Pamela L.

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Regulation of Ingestive Behaviors in the Rat by GSK1521498, a Novel μ-Opioid Receptor-Selective Inverse Agonist von Ignar, Diane M., Goetz, Aaron S., Noble, Kimberly Nichols, Carballo, Luz Helena, Stroup, Andrea E., Fisher, Julie C., Boucheron, Joyce A., Brainard, Tracy A., Larkin, Andrew L., Epperly, Andrea H., Shearer, Todd W., Sorensen, Scott D., Speake, Jason D., Hommel, Jonathan D.

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Phenoxyacetic acids as PPAR[delta] partial agonists: Synthesis, optimization, and in vivo efficacy von Evans, Karen A, Shearer, Barry G, Wisnoski, David D, Shi, Dongchuan, Sparks, Steven M, Sternbach, Daniel D, Winegar, Deborah A, Billin, Andrew N, Britt, Christy, Way, James M, Epperly, Andrea H, Leesnitzer, Lisa M, Merrihew, Raymond V, Xu, Robert X, Lambert, Millard H, Jin, Jian

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Regulation of ingestive behaviors in the rat by GSK1521498, a novel micro-opioid receptor-selective inverse agonist von Ignar, Diane M, Goetz, Aaron S, Noble, Kimberly Nichols, Carballo, Luz Helena, Stroup, Andrea E, Fisher, Julie C, Boucheron, Joyce A, Brainard, Tracy A, Larkin, Andrew L, Epperly, Andrea H, Shearer, Todd W, Sorensen, Scott D, Speake, Jason D, Hommel, Jonathan D

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Reviews von Van Ness, Peter H., Madden, Kathryn, Barbre, Claude, Dixon, Andrea, Kirby, Jill Carlen, Epperly, Bruce G., DuBose, Todd, Dal Maso, Donald F., Ulanov, Barry

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