Applications of tert-butanesulfinamide in the asymmetric synthesis of amines von Ellman, J. A.

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Inhibition of STEP61 ameliorates deficits in mouse and hiPSC-based schizophrenia models von Xu, J, Hartley, B J, Kurup, P, Phillips, A, Topol, A, Xu, M, Ononenyi, C, Foscue, E, Ho, S-M, Baguley, T D, Carty, N, Barros, C S, Müller, U, Gupta, S, Gochman, P, Rapoport, J, Ellman, J A, Pittenger, C, Aronow, B, Nairn, A C, Nestor, M W, Lombroso, P J, Brennand, K J

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Annulation of Aromatic Imines via Directed C−H Activation with Wilkinson's Catalyst von Thalji, R. K, Ahrendt, K. A, Bergman, R. G, Ellman, J. A

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Annulation of Alkenyl-Substituted Heterocycles via Rhodium-Catalyzed Intramolecular C−H Activated Coupling Reactions von Tan, K. L, Bergman, R. G, Ellman, J. A

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Synthesis of positional-scanning libraries of fluorogenic peptide substrates to define the extended substrate specificity of plasmin and thrombin von Craik, Charles S, Ellman, Jonathan A, Backes, Bradley J, Harris, Jennifer L, Leonetti, Francesco

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Asymmetric Synthesis of Protected 1,2-Amino Alcohols Using tert-Butanesulfinyl Aldimines and Ketimines von Tang, Tony P, Volkman, Steven K, Ellman, Jonathan A

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Inhibition of STEP 61 ameliorates deficits in mouse and hiPSC-based schizophrenia models von Xu, J, Hartley, B J, Kurup, P, Phillips, A, Topol, A, Xu, M, Ononenyi, C, Foscue, E, Ho, S-M, Baguley, T D, Carty, N, Barros, C S, Müller, U, Gupta, S, Gochman, P, Rapoport, J, Ellman, J A, Pittenger, C, Aronow, B, Nairn, A C, Nestor, M W, Lombroso, P J, Brennand, K J

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Potent, Low-Molecular-Weight Non-Peptide Inhibitors of Malarial Aspartyl Protease Plasmepsin II von Haque, Tasir S, Skillman, A. Geoffrey, Lee, Christina E, Habashita, Hiromu, Gluzman, Ilya Y, Ewing, Todd J. A, Goldberg, Daniel E, Kuntz, Irwin D, Ellman, Jonathan A

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The Combinatorial Synthesis and Chemical and Biological Evaluation of a 1,4-Benzodiazepine Library von Bunin, Barry A., Plunkett, Matthew J., Ellman, Jonathan A.

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Design, Synthesis, and Utility of a Support-Bound tert-Butanesulfinamide von Dragoli, Dean R, Burdett, Matthew T, Ellman, Jonathan A

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Combinatorial Target-Guided Ligand Assembly: Identification of Potent Subtype-Selective c-Src Inhibitors von Maly, D J, Choong, I C, Ellman, J A

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Compounds That Activate the Mouse Melanocortin-1 Receptor Identified by Screening a Small Molecule Library Based upon the β-Turn von Haskell-Luevano, Carrie, Rosenquist, Åsa, Souers, Andrew, Khong, Kathy C, Ellman, Jonathon A, Cone, Roger D

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Rapid and General Profiling of Protease Specificity by Using Combinatorial Fluorogenic Substrate Libraries von Harris, Jennifer L., Backes, Bradley J., Leonetti, Francesco, Mahrus, Sami, Ellman, Jonathan A., Craik, Charles S.

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Novel Cathepsin D Inhibitors Block the Formation of Hyperphosphorylated Tau Fragments in Hippocampus von Bi, Xiaoning, Haque, Tasir S., Zhou, Jun, Skillman, A. Geoffrey, Lin, Bin, Lee, Christine E., Kuntz, Irwin D., Ellman, Jonathan A., Lynch, Gary

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Synthesis of Enantiomerically Pure N-tert-Butanesulfinyl Imines (tert-Butanesulfinimines) by the Direct Condensation of tert-Butanesulfinamide with Aldehydes and Ketones von Liu, Guangcheng, Cogan, Derek A, Owens, Timothy D, Tang, Tony P, Ellman, Jonathan A

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Site-Specific Incorporation of Novel Backbone Structures into Proteins von Ellman, Jonathan A., Mendel, David, Schultz, Peter G.

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Catalytic Asymmetric Synthesis of tert-Butanesulfinamide. Application to the Asymmetric Synthesis of Amines von Liu, Guangcheng, Cogan, Derek A, Ellman, Jonathan A

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An Alkanesulfonamide “Safety-Catch” Linker for Solid-Phase Synthesis von Backes, Bradley J, Ellman, Jonathan A

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Synthesis and Crystal Structure of a Unique and Homochiral N,S-Bonded N,N ‘-Bis(tert-butanesulfinyl)amidinate Rhodium(I) Complex von Souers, Andrew J, Owens, Timothy D, Oliver, Allen G, Hollander, Frederick J, Ellman, Jonathan A

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Synthesis, Utility, and Structure of Novel Bis(sulfinyl)imidoamidine Ligands for Asymmetric Lewis Acid Catalysis von Owens, Timothy D, Hollander, Frederick J, Oliver, Allen G, Ellman, Jonathan A

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