Novel M2‐selective, Gi‐biased agonists of muscarinic acetylcholine receptors von Randáková, Alena, Nelic, Dominik, Ungerová, Dana, Nwokoye, Peter, Su, Qiwen, Doležal, Vladimír, El‐Fakahany, Esam E., Boulos, John, Jakubík, Jan

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Current Advances in Allosteric Modulation of Muscarinic Receptors von Jakubik, Jan, El-Fakahany, Esam E

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Analysis of equilibrium binding of an orthosteric tracer and two allosteric modulators von Dolezal, Vladimír, Jakubík, Jan, El-Fakahany, Esam E, Randáková, Alena

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Allosteric Modulation of GPCRs of Class A by Cholesterol von Jakubík, Jan, El-Fakahany, Esam E

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A randomized controlled pilot study of the University of Minnesota mentoring excellence training academy: A hybrid learning approach to research mentor training von Weber-Main, Anne Marie, Shanedling, Janet, Kaizer, Alexander M, Connett, John, Lamere, Michelle, El-Fakahany, Esam E

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Long-term activation upon brief exposure to xanomleline is unique to M1 and M4 subtypes of muscarinic acetylcholine receptors von Šantrůčková, Eva, Doležal, Vladimír, El-Fakahany, Esam E, Jakubík, Jan

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The operational model of allosteric modulation of pharmacological agonism von Jakubík, Jan, Randáková, Alena, Chetverikov, Nikolai, El-Fakahany, Esam E., Doležal, Vladimír

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Subtype differences in pre-coupling of muscarinic acetylcholine receptors von Dolezal, Vladimír, Jakubík, Jan, El-Fakahany, Esam E, Janícková, Helena, Randáková, Alena

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Allosteric Modulation of Muscarinic Acetylcholine Receptors von Jakubík, Jan, El-Fakahany, Esam E

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Agonist-Specific Conformations of the M 2 Muscarinic Acetylcholine Receptor Assessed by Molecular Dynamics von Randáková, Alena, Nelic, Dominik, Doležal, Vladimír, El-Fakahany, Esam E, Boulos, John, Jakubík, Jan

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Neuroactive steroids, WIN-compounds and cholesterol share a common binding site on muscarinic acetylcholine receptors von Dolejší, Eva, Chetverikov, Nikolai, Szánti-Pintér, Eszter, Nelic, Dominik, Randáková, Alena, Doležal, Vladimír, El-Fakahany, Esam E., Kudová, Eva, Jakubík, Jan

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Novel M 2 -selective, G i -biased agonists of muscarinic acetylcholine receptors von Randáková, Alena, Nelic, Dominik, Ungerová, Dana, Nwokoye, Peter, Su, Qiwen, Doležal, Vladimír, El-Fakahany, Esam E, Boulos, John, Jakubík, Jan

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Applications and limitations of fitting of the operational model to determine relative efficacies of agonists von Jakubík, Jan, Randáková, Alena, Rudajev, Vladimír, Zimčík, Pavel, El-Fakahany, Esam E., Doležal, Vladimír

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Changes in Membrane Cholesterol Differentially Influence Preferential and Non-preferential Signaling of the M1 and M3 Muscarinic Acetylcholine Receptors von Michal, Pavel, El-Fakahany, Esam E., Doležal, Vladimír

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Role of membrane cholesterol in differential sensitivity of muscarinic receptor subtypes to persistently bound xanomeline von Randáková, Alena, Dolejší, Eva, Rudajev, Vladimír, Zimčík, Pavel, Doležal, Vladimír, El-Fakahany, Esam E., Jakubík, Jan

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Towards predictive docking at aminergic G-protein coupled receptors von Jakubík, Jan, El-Fakahany, Esam E., Doležal, Vladimír

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Binding of N-methylscopolamine to the extracellular domain of muscarinic acetylcholine receptors von Jakubík, Jan, Randáková, Alena, Zimčík, Pavel, El-Fakahany, Esam E., Doležal, Vladimír

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Molecular Mechanisms of Methoctramine Binding and Selectivity at Muscarinic Acetylcholine Receptors von Jakubík, Jan, Zimčík, Pavel, Randáková, Alena, Fuksová, Květoslava, El-Fakahany, Esam E., Doležal, Vladimír

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Synthesis and evaluation of xanomeline analogs : Probing the wash-resistant phenomenon at the M1 muscarinic acetylcholine receptor von KANE, Brian E, GRANT, Marianne K. O, EL-FAKAHANY, Esam E, FERGUSON, David M

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Uncoupling of M1 muscarinic receptor/G-protein interaction by amyloid β(1-42) von Janíčková, Helena, Rudajev, Vladimír, Zimčík, Pavel, Jakubík, Jan, Tanila, Heikki, El-Fakahany, Esam E, Doležal, Vladimír

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