A Convenient Synthesis of 2-Cyanoimidazoles von Dudfield, P. J., Ekwuru, C. T., Hamilton, K., Osbourn, C. E., Simpson, D. J.

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Chronic diazepam treatment in rats causes long-lasting changes in central ( super(3)H)-5-hydroxytryptamine and ( super(14)C)- gamma -aminobutyric acid release von Hitchcott, P K, File, SE, Ekwuru, M, Neal, MJ

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Abstract P056: Polθ inhibitors elicit BRCA -gene synthetic lethality and target PARP inhibitor resistance von Zatreanu, Diana A., Robinson, Helen M. R., Alkhatib, Omar, Boursier, Marie, Finch, Harry, Geo, Lerin, Grande, Diego, Grinkevich, Vera, Heald, Robert, Langdon, Sophie, Majithiya, Jayesh, McWhirter, Claire, Martin, Niall M. B., Moore, Shaun, Neves, Joana, Rajendra, Eeson, Ranzani, Marco, Schaedler, Theresia, Stockley, Martin, Wiggins, Kimberley, Brough, Rachel, Sridhar, Sandhya, Gulati, Aditi, Shao, Nan, Badder, Luned M, Novo, Daniela, Knight, Eleanor G., Marlow, Rebecca, Haider, Syed, Callen, Elsa, Hewitt, Graeme, Schimmel, Joost, Prevo, Remko, Alli, Christina, Ferdinand, Amanda, Bell, Cameron, Blencowe, Peter, Calder, Mathew, Charles, Mark, Curry, Jayne, Ekwuru, Tennyson, Ewings, Katherine, Nussenzweig, Andre, Tijsterman, Marcel, Tutt, Andrew, Boulton, Simon J., Higgins, Geoff S., Pettitt, Steve, Smith, Graeme C. M., Lord, Christopher J.

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Abstract 5697: Targeting PARP inhibitor resistance with Polθ inhibitors von Zatreanu, Diana, Robinson, Helen, Alkhatib, Omar, Boursier, Marie, Finch, Harry, Geo, Lerin, Grande, Diego, Grinkevich, Vera, Heald, Robert, Langdon, Sophie, Majithiya, Jayesh, McWhirter, Claire, Martin, Niall, Moore, Shaun, Neves, Joana, Rajendra, Eeson, Ranzani, Marco, Schaedler, Theresia, Stockley, Martin, Wiggins, Kimberley, Brough, Rachel, Sridhar, Sandhya, Gulati, Aditi, Shao, Nan, Badder, Luted, Novo, Daniela, Knight, Eleanor, Marlow, Rebecca, Haider, Syed, Callen, Elsa, Hewitt, Graeme, Schimmel, Joost, Prevo, Remko, Alli, Christina, Ferdinand, Amanda, Bell, Cameron, Blencowe, Peter, Bot, Chris, Calder, Mathew, Charles, Mark, Curry, Jayne, Ekwuru, Tennyson, Nussenzweig, Andre, Tijsterman, Marcel, Tutt, Andrew N., Boulton, Simon, Higgins, Geoff, Pettitt, Stephen J., Smith, Graeme C., Lord, Christopher J.

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Discovery, Development, and SAR of Aminothiazoles as LIMK Inhibitors with Cellular Anti-Invasive Properties von Charles, Mark D, Brookfield, Joanna L, Ekwuru, Tennyson C, Stockley, Martin, Dunn, John, Riddick, Michelle, Hammonds, Tim, Trivier, Elisabeth, Greenland, Gavin, Wong, Ai Ching, Cheasty, Anne, Boyd, Susan, Crighton, Diane, Olson, Michael F

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Discovery, Characterization, and Structure-Based Optimization of Small-Molecule In Vitro and In Vivo Probes for Human DNA Polymerase Theta von Stockley, Martin L., Ferdinand, Amanda, Benedetti, Giovanni, Blencowe, Peter, Boyd, Susan M., Calder, Mat, Charles, Mark D., Edwardes, Lucy V., Ekwuru, Tennyson, Finch, Harry, Galbiati, Alessandro, Geo, Lerin, Grande, Diego, Grinkevich, Vera, Holliday, Nicholas D., Krajewski, Wojciech W., MacDonald, Ellen, Majithiya, Jayesh B., McCarron, Hollie, McWhirter, Claire L., Patel, Viral, Pedder, Chris, Rajendra, Eeson, Ranzani, Marco, Rigoreau, Laurent J. M., Robinson, Helen M. R., Schaedler, Theresia, Sirina, Julija, Smith, Graeme C. M., Swarbrick, Martin E., Turnbull, Andrew P., Willis, Simon, Heald, Robert A.

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Correction to “Discovery, Characterization, and Structure-Based Optimization of Small-Molecule In Vitro and In Vivo Probes for Human DNA Polymerase Theta” von Stockley, Martin L., Benedetti, Giovanni, Blencowe, Peter, Boulton, Simon J., Boyd, Susan M., Calder, Mat, Charles, Mark D., Edwardes, Lucy V., Ekwuru, Tennyson, Ferdinand, Amanda, Finch, Harry, Galbiati, Alessandro, Geo, Lerin, Grande, Diego, Grinkevich, Vera, Higgins, Geoff S., Holliday, Nicholas D., Krajewski, Wojciech W., MacDonald, Ellen, Majithiya, Jayesh B., McCarron, Hollie, McWhirter, Claire L., Patel, Viral, Pedder, Chris, Rajendra, Eeson, Ranzani, Marco, Rigoreau, Laurent J. M., Robinson, Helen M. R., Schaedler, Theresia, Sirina, Julija, Smith, Graeme C. M., Swarbrick, Martin E., Turnbull, Andrew P., Willis, Simon, Zemla, Aleksandra, Heald, Robert A.

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Pol theta inhibitors elicit BRCA-gene synthetic lethality and target PARP inhibitor resistance von Zatreanu, D., Robinson, H.M.R., Alkhatib, O., Boursier, M., Finch, H., Geo, L., Grande, D., Grinkevich, V., Heald, R.A., Langdon, S., Majithiya, J., McWhirter, C., Martin, N.M.B., Moore, S., Neves, J., Rajendra, E., Ranzani, M., Schaedler, T., Stockley, M., Wiggins, K., Brough, R., Sridhar, S., Gulati, A., Shao, N., Badder, L.M., Novo, D., Knight, E.G., Marlow, R., Haider, S., Callen, E., Hewitt, G., Schimmel, J., Prevo, R., Alli, C., Ferdinand, A., Bell, C., Blencowe, P., Bot, C., Calder, M., Charles, M., Curry, J., Ekwuru, T., Ewings, K., Krajewski, W., MacDonald, E., McCarron, H., Pang, L., Pedder, C., Rigoreau, L., Swarbrick, M., Wheatley, E., Willis, S., Wong, A.C., Nussenzweig, A., Tijsterman, M., Tutt, A., Boulton, S.J., Higgins, G.S., Pettitt, S.J., Smith, G.C.M., Lord, C.J.

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Chronic diazepam treatment in rats causes long‐lasting changes in central [3H]‐5‐hydroxytryptamine and [14C]‐γ‐aminobutyric acid release von Hitchcott, P.K., File, Sandra E., Ekwuru, M., Neal, M.J.

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Differential cardiovascular effects of propranolol, atenolol, and pindolol measured by impedance cardiography von THOMAS, S. H. L, COOPER, R. C, EKWURU, M, FLETCHER, S, GILBODY, J, HUSSEYIN, T. S, ISHAQUE, M, JAGATHESAN, R, REDDY, G, SMITH, S. E

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FUNGICIDE von COOKE TRACEY, EKWURU TENNYSON, TURNER RICHAR MICHAEEL, HARDY DAVID, PETTINGER ANDREW, MILLWARD PETER, MARONEY BRIAN, THOMAS PETER STANLEY

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Protein kinase D as a potential new target for cancer therapy von LaValle, Courtney R., George, Kara M., Sharlow, Elizabeth R., Lazo, John S., Wipf, Peter, Wang, Q. Jane

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Synthesis of isotope-labeled HSP90 inhibitor: [13CD3] and [14C]-TAK-459 von Plesescu, Mihaela, Elliott, Eric L., Li, Yuexian, Prakash, Shimoga R.

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Preparation of Polyfunctionalized Aromatic Nitriles from Aryl Oxazolines von Hess, A., Guelen, H. C., Alandini, N., Mourati, A., Guersoy, Y. C., Knochel, P.

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3,5-Diarylazoles as novel and selective inhibitors of protein kinase D von Gamber, Gabriel G., Meredith, Erik, Zhu, Qingming, Yan, Wanlin, Rao, Chang, Capparelli, Michael, Burgis, Robin, Enyedy, Istvan, Zhang, Ji-Hu, Soldermann, Nicolas, Beattie, Kimberley, Rozhitskaya, Olga, Koch, Keith A., Pagratis, Nikos, Hosagrahara, Vinayak, Vega, Richard B., McKinsey, Timothy A., Monovich, Lauren

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A Reconstruction of the Idea and Practice of Masquerading among Igbo People of South-Eastern Nigeria von Asiegbu, Martin F., Dimonye, Simeon C.

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Recent advances in the rational design and development of LIM kinase inhibitors are not enough to enter clinical trials von Manetti, Fabrizio

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The evaluation of drug-induced changes in cardiac inotropy in dogs: Results from a HESI-sponsored consortium von Guth, Brian D., Chiang, Alan Y., Doyle, Jennifer, Engwall, Michael J., Guillon, Jean-Michel, Hoffmann, Peter, Koerner, John, Mittelstadt, Scott, Ottinger, Sean, Pierson, Jennifer Beck, Pugsley, Michael K., Rossman, Eric I., Walisser, Jacqueline, Sarazan, R. Dustan

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Synthesis of 2-aminothiazoles via rhodium-catalyzed carbenoid insertion/annulation of sulfoxonium ylides with thioureas von Chen, Yuncan, Lv, Shan, Lai, Ruizhi, Xu, Yingying, Huang, Xin, Li, Jianglian, Lv, Guanghui, Wu, Yong

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Effects of sodium valproate on synaptic transmission and neuronal excitability in rat hippocampus von Yong, Wu, Zhang, Min-Min, Wang, Shu, Ruan, Di-Yun

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