Mechanism of Active Renal Tubular Efflux of Tenofovir von RAY, Adrian S, CIHLAR, Tomas, ROBINSON, Kelly L, TONG, Leah, VELA, Jennifer E, FULLER, Michael D, WIEMAN, Lani M, EISENBERG, Eugene J, RHODES, Gerry R

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Quantification of Phosphonate Drugs by 1H–31P HSQC Shows That Rats Are Better Models of Primate Drug Exposure than Mice von Barekatain, Yasaman, Khadka, Sunada, Harris, Kristen, Delacerda, Jorge, Yan, Victoria C., Chen, Ko-Chien, Pham, Cong-Dat, Uddin, Md. Nasir, Avritcher, Rony, Eisenberg, Eugene J., Kalluri, Raghu, Millward, Steven W., Muller, Florian L.

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Discovery of an Oral Respiratory Syncytial Virus (RSV) Fusion Inhibitor (GS-5806) and Clinical Proof of Concept in a Human RSV Challenge Study von Mackman, Richard L, Sangi, Michael, Sperandio, David, Parrish, Jay P, Eisenberg, Eugene, Perron, Michel, Hui, Hon, Zhang, Lijun, Siegel, Dustin, Yang, Hai, Saunders, Oliver, Boojamra, Constantine, Lee, Gary, Samuel, Dharmaraj, Babaoglu, Kerim, Carey, Anne, Gilbert, Brian E, Piedra, Pedro A, Strickley, Robert, Iwata, Quynh, Hayes, Jaclyn, Stray, Kirsten, Kinkade, April, Theodore, Dorothy, Jordan, Robert, Desai, Manoj, Cihlar, Tomas

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Antiviral Efficacy of a Respiratory Syncytial Virus (RSV) Fusion Inhibitor in a Bovine Model of RSV Infection von Jordan, Robert, Shao, Matt, Mackman, Richard L, Perron, Michel, Cihlar, Tomas, Lewis, Sandy A, Eisenberg, Eugene J, Carey, Anne, Strickley, Robert G, Chien, Jason W, Anderson, Mark L, McEligot, Heather A, Behrens, Nicole E, Gershwin, Laurel J

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Selective Intracellular Activation of a Novel Prodrug of the Human Immunodeficiency Virus Reverse Transcriptase Inhibitor Tenofovir Leads to Preferential Distribution and Accumulat... von LEE, William A, HE, Gong-Xin, EISENBERG, Eugene, CIHLAR, Tomas, SWAMINATHAN, Swami, MULATO, Andrew, CUNDY, Kenneth C

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RNase H Active Site Inhibitors of Human Immunodeficiency Virus Type 1 Reverse Transcriptase: Design, Biochemical Activity, and Structural Information von Kirschberg, Thorsten A, Balakrishnan, Mini, Squires, Neil H, Barnes, Tiffany, Brendza, Katherine M, Chen, Xiaowu, Eisenberg, Eugene J, Jin, Weili, Kutty, Nilima, Leavitt, Stephanie, Liclican, Albert, Liu, Qi, Liu, Xiaohong, Mak, John, Perry, Jason K, Wang, Michael, Watkins, William J, Lansdon, Eric B

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The Drug–Drug Interaction Profile of Presatovir von Xin, Yan, Weng, Winnie, Murray, Bernard P., Eisenberg, Eugene J., Chien, Jason W., Ling, John, Silverman, Jeffrey A.

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Identification of GS 4104 as an Orally Bioavailable Prodrug of the Influenza Virus Neuraminidase Inhibitor GS 4071 von WEIXING LI, ESCARPE, P. A, KIM, C. U, BISCHOFBERGER, N, CHEN, M. S, MENDEL, D. B, EISENBERG, E. J, CUNDY, K. C, SWEET, C, JAKEMAN, K. J, MERSON, J, LEW, W, WILLIAMS, M, LIJUN ZHANG

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Optimization of Pharmacokinetics through Manipulation of Physicochemical Properties in a Series of HCV Inhibitors von Lazerwith, Scott E, Bahador, Gina, Canales, Eda, Cheng, Guofeng, Chong, Lee, Clarke, Michael O, Doerffler, Edward, Eisenberg, Eugene J, Hayes, Jaclyn, Lu, Bing, Liu, Qi, Matles, Mike, Mertzman, Michael, Mitchell, Michael L, Morganelli, Philip, Murray, Bernard P, Robinson, Margaret, Strickley, Robert G, Tessler, Megan, Tirunagari, Neeraj, Wang, Jianhong, Wang, Yujin, Zhang, Jennifer R, Zheng, Xubin, Zhong, Weidong, Watkins, William J

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Antiviral Efficacy and Pharmacokinetics of Oral Adefovir Dipivoxil in Chronically Woodchuck Hepatitis Virus-Infected Woodchucks von CULLEN, John M, LI, Daniel H, BROWN, Cynthia, EISENBERG, Eugene J, CUNDY, Kenneth C, WOLFE, Julie, TOOLE, J. A. Y, GIBBS, Craig

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GS-5806 Inhibits a Broad Range of Respiratory Syncytial Virus Clinical Isolates by Blocking the Virus-Cell Fusion Process von Perron, Michel, Stray, Kirsten, Kinkade, April, Theodore, Dorothy, Lee, Gary, Eisenberg, Eugene, Sangi, Michael, Gilbert, Brian E, Jordan, Robert, Piedra, Pedro A, Toms, Geoffery L, Mackman, Richard, Cihlar, Tomas

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Quantification of Phosphonate Drugs by 1 H– 31 P HSQC Shows That Rats Are Better Models of Primate Drug Exposure than Mice von Barekatain, Yasaman, Khadka, Sunada, Harris, Kristen, Delacerda, Jorge, Yan, Victoria C., Chen, Ko-Chien, Pham, Cong-Dat, Uddin, Md. Nasir, Avritcher, Rony, Eisenberg, Eugene J., Kalluri, Raghu, Millward, Steven W., Muller, Florian L.

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Lack of a metabolic and antiviral drug interaction between tenofovir, abacavir and lamivudine von RAY, Adrian S, MYRICK, Florence, VELA, Jennifer E, OLSON, Loren Y, EISENBERG, Eugene J, BORROTO-ESODA, Katyna, MILLER, Michael D, FRIDLAND, Arnold

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High-performance liquid chromatographic determination of cytosine-containing compounds by precolumn fluorescence derivatization with phenacyl bromide: application to antiviral nucl... von Eisenberg, Eugene J., Cundy, Kenneth C.

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Drug Interaction Profile of GS-5806 von Xin, Yan, Toback, Seth, Weng, Winnie, Grycz, Krysia, Eisenberg, Eugene, Weston, Jonna, Murray, Bernard, Chien, Jason, Ramanathan, Srini, Silverman, Jeffrey

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Isolation and identification of a metabolite of cidofovir from rat kidney von Eisenberg, Eugene J, Lynch, Geoffrey R, Bidgood, Alison M, Krishnamurty, Krish, Cundy, Kenneth C

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765Drug Interaction Profile of GS-5806 von Xin, Yan, Toback, Seth, Weng, Winnie, Grycz, Krysia, Eisenberg, Eugene, Weston, Jonna, Murray, Bernard, Chien, Jason, Ramanathan, Srini, Silverman, Jeffrey

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Influence of Treatment Schedule and Viral Challenge Dose on the in Vivo Influenza Virus-Inhibitory Effects of the Orally Administered Neuraminidase Inhibitor GS 4104 von Sidwell, Robert W, Bailey, Kevin W, Bemis, Paul A, Wong, Min-Hui, Eisenberg, Eugene J, Huffman, John H

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Amperometric high-performance liquid chromatographic detection of NADH at a base-activated glassy carbon electrode von Eisenberg, Eugene J, Cundy, Kenneth C

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Penetration of GS4071, a novel influenza neuraminidase inhibitor, into rat bronchoalveolar lining fluid following oral administration of the prodrug GS4104 von EISENBERG, E. J, BIDGOOD, A, CUNDY, K. C

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