The inophyllums, novel inhibitors of HIV-1 reverse transcriptase isolated from the Malaysian tree, Calophyllum inophyllum Linn von Patil, Ashok D, Freyer, Alan J, Eggleston, Drake S, Haltiwanger, R. Curtis, Bean, Mark F, Taylor, Paul B, Caranfa, Mary Jo, Breen, Ann L, Bartus, Henry R

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New roles for structure in biology and drug discovery von Russell, R B, Eggleston, D S

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Discovery of a Novel Class of Substituted Pyrrolooctahydroisoquinolines as Potent and Selective δ Opioid Agonists, Based on an Extension of the Message−Address Concept von Dondio, Giulio, Ronzoni, Silvano, Eggleston, Drake S, Artico, Marco, Petrillo, Paola, Petrone, Giuseppe, Visentin, Luciano, Farina, Carlo, Vecchietti, Vittorio, Clarke, Geoffrey D

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Inhibitors of bacterial tyrosyl tRNA synthetase: synthesis of four stereoisomeric analogues of the natural product SB-219383 von Berge, John M, Copley, Royston C.B, Eggleston, Drake S, Hamprecht, Dieter W, Jarvest, Richard L, Mensah, Lucy M, O'Hanlon, Peter J, Pope, Andrew J

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Synthesis and Recognition Properties of Aromatic Amide Oligomers:  Molecular Zippers von Bisson, Adrian P, Carver, Fiona J, Eggleston, Drake S, Haltiwanger, R. Curtis, Hunter, Christopher A, Livingstone, David L, McCabe, James F, Rotger, Carmen, Rowan, Alan E

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Non-thiazolidinedione antihyperglycaemic agents. Part 3: the effects of stereochemistry on the potency of α-methoxy-β-phenylpropanoic acids von Haigh, David, Allen, Graham, Birrell, Helen C., Buckle, Derek R., Cantello, Barrie C.C., Eggleston, Drake S., Haltiwanger, R.Curtis, Holder, Julie C., Lister, Carolyn A., Pinto, Ivan L., Rami, Harshad K., Sime, John T., Smith, Stephen A., Sweeney, John D.

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1,4-Cyclohexanecarboxylates:  Potent and Selective Inhibitors of Phosophodiesterase 4 for the Treatment of Asthma von Christensen, Siegfried B, Guider, Aimee, Forster, Cornelia J, Gleason, John G, Bender, Paul E, Karpinski, Joseph M, DeWolf, Walter E, Barnette, Mary S, Underwood, David C, Griswold, Don E, Cieslinski, Lenora B, Burman, Miriam, Bochnowicz, Steven, Osborn, Ruth R, Manning, Carol D, Grous, Marilyn, Hillegas, Leonard M, Bartus, Joan O'Leary, Ryan, M. Dominic, Eggleston, Drake S, Haltiwanger, R. Curtis, Torphy, Theodore J

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The crystal structure, absolute configuration, and phosphodiesterase inhibitory activity of (+)-1-(4-bromobenzyl)-4-(3-cyclopentyloxy)-4-methoxyphenyl-pyrrolidin-2-one von BAURES, P. W, EGGLESTON, D. S, ERHARD, K. F, CIESLINSKI, L. B, TORPHY, T. J, CHRISTENSEN, S. B

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Investigation of conformational specificity at GPIIb/IIIa: evaluation of conformationally constrained RGD peptides von Peishoff, Catherine E, Ali, Fadia E, Bean, John W, Calvo, Raul, D'Ambrosio, Cynthia A, Eggleston, Drake S, Kline, Tammy Page, Koster, Paul F, Hwang, S. M

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ATP-Citrate Lyase as a Target for Hypolipidemic Intervention. 2. Synthesis and Evaluation of (3R,5S)-ω-Substituted-3-carboxy-3,5-dihydroxyalkanoic Acids and Their γ-Lactone Prodrug... von Gribble, Andrew D, Ife, Robert J, Shaw, Antony, McNair, David, Novelli, Christine E, Bakewell, Susan, Shah, Virendra P, Dolle, Roland E, Groot, Pieter H, Pearce, Nigel, Yates, John, Tew, David, Boyd, Helen, Ashman, Stephen, Eggleston, Drake S, Haltiwanger, R. Curtis, Okafo, George

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Apakaochtodenes A and B:  Two Tetrahalogenated Monoterpenes from the Red Marine Alga Portieria hornemannii von Gunatilaka, A. A. Leslie, Paul, Valerie J, Park, Peter U, Puglisi, Melany P, Gitler, Aaron D, Eggleston, Drake S, Haltiwanger, R. Curtis, Kingston, David G. I

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The structure of ribonuclease P protein from Staphylococcus aureus reveals a unique binding site for single-stranded RNA von Spitzfaden, Claus, Nicholson, Neville, Jones, Jo J, Guth, Sabine, Lehr, Ruth, Prescott, Cathy D, Hegg, Lisa A, Eggleston, Drake S

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Two New Nitrogenous Sesquiterpenes from the Sponge Axinyssa aplysinoides von Patil, Ashok D, Freyer, Alan J, Reichwein, Rex, Bean, Mark F, Faucette, Leo, Johnson, Randall K, Haltiwanger, R. Curtis, Eggleston, Drake S

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New Polyhydroxylated Pregnadienes from the South African Soft Coral Pieterfaurea unilobata von Beukes, Denzil R, Davies-Coleman, Michael T, Eggleston, Drake S, Haltiwanger, R. Curtis, Tomkowicz, Brian

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Structure–activity analysis of truncated orexin-A analogues at the orexin-1 receptor von Darker, John G, Porter, Roderick A, Eggleston, Drake S, Smart, Darren, Brough, Stephen J, Sabido-David, Cibele, Jerman, Jeffrey C

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Conformational Preferences in a Benzodiazepine Series of Potent Nonpeptide Fibrinogen Receptor Antagonists von Keenan, Richard M, Callahan, James F, Samanen, James M, Bondinell, William E, Calvo, Raul R, Chen, Lichong, DeBrosse, Charles, Eggleston, Drake S, Haltiwanger, R. Curtis, Hwang, Shing Mei, Jakas, Dalia R, Ku, Thomas W, Miller, William H, Newlander, Kenneth A, Nichols, Andrew, Parker, Michael F, Southhall, Linda S, Uzinskas, Irene, Vasko-Moser, Janice A, Venslavsky, Joseph W, Wong, Angela S, Huffman, William F

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Structure determination of racemic trichogin A IV using centrosymmetric crystals von Toniolo, Claudio, Peggion, Cristina, Crisma, Marco, Formaggio, Fernando, Shui, Xiuqi, Eggleston, Drake S

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Molecular structures of l-Leu-l-Tyr, Gly-d,l-Met.p-toluenesulfonate and l-His-l-Leu von Krause, J. A., Baures, P. W., Eggleston, D. S.

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Imidazole-5-acrylic acids: potent nonpeptide angiotensin II receptor antagonists designed using a novel peptide pharmacophore model von Keenan, R. M, Weinstock, J, Finkelstein, J. A, Franz, R. G, Gaitanopoulos, D. E, Girard, G. R, Hill, D. T, Morgan, T. M, Samanen, J. M

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Synthesis of imidazoles via hetero-Cope rearrangements von Lantos, Ivan, Zhang, Wei Yuan, Shui, Xiuqi, Eggleston, Drake S

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