Nucleophilic (Radio)Fluorination of Redox-Active Esters via Radical-Polar Crossover Enabled by Photoredox Catalysis von Webb, Eric W, Park, John B, Cole, Erin L, Donnelly, David J, Bonacorsi, Samuel J, Ewing, William R, Doyle, Abigail G

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Decarboxylative alkylation for site-selective bioconjugation of native proteins via oxidation potentials von Bloom, Steven, Liu, Chun, Kölmel, Dominik K., Qiao, Jennifer X., Zhang, Yong, Poss, Michael A., Ewing, William R., MacMillan, David W. C.

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Site-Selective Functionalization of Methionine Residues via Photoredox Catalysis von Kim, Junyong, Li, Beryl X, Huang, Richard Y.-C, Qiao, Jennifer X, Ewing, William R, MacMillan, David W. C

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Catalytic Ring Expansions of Cyclic Alcohols Enabled by Proton-Coupled Electron Transfer von Zhao, Kuo, Yamashita, Kenji, Carpenter, Joseph E, Sherwood, Trevor C, Ewing, William R, Cheng, Peter T. W, Knowles, Robert R

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Site-selective tyrosine bioconjugation via photoredox catalysis for native-to-bioorthogonal protein transformation von Li, Beryl X., Kim, Daniel K., Bloom, Steven, Huang, Richard Y.-C., Qiao, Jennifer X., Ewing, William R., Oblinsky, Daniel G., Scholes, Gregory D., MacMillan, David W. C.

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meta C–H Arylation of Electron-Rich Arenes: Reversing the Conventional Site Selectivity von Liu, Luo-Yan, Qiao, Jennifer X, Yeung, Kap-Sun, Ewing, William R, Yu, Jin-Quan

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meta‐Selective C−H Arylation of Fluoroarenes and Simple Arenes von Liu, Luo‐Yan, Qiao, Jennifer X., Yeung, Kap‐Sun, Ewing, William R., Yu, Jin‐Quan

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Milvexian, an orally bioavailable, small‐molecule, reversible, direct inhibitor of factor XIa: In vitro studies and in vivo evaluation in experimental thrombosis in rabbits von Wong, Pancras C., Crain, Earl J., Bozarth, Jeffrey M., Wu, Yiming, Dilger, Andrew K., Wexler, Ruth R., Ewing, William R., Gordon, David, Luettgen, Joseph M.

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Ligand-Enabled Pd(II)-Catalyzed C(sp3)–H Lactonization Using Molecular Oxygen as Oxidant von Qian, Shaoqun, Li, Zi-Qi, Li, Minyan, Wisniewski, Steven R, Qiao, Jennifer X, Richter, Jeremy M, Ewing, William R, Eastgate, Martin D, Chen, Jason S, Yu, Jin-Quan

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PdII‐Catalyzed Enantioselective C(sp3)–H Arylation of Cyclobutyl Ketones Using a Chiral Transient Directing Group von Xiao, Li‐Jun, Hong, Kai, Luo, Fan, Hu, Liang, Ewing, William R., Yeung, Kap‐Sun, Yu, Jin‐Quan

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Hemilabile Benzyl Ether Enables γ‑C(sp3)–H Carbonylation and Olefination of Alcohols von Tanaka, Keita, Ewing, William R, Yu, Jin-Quan

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Overcoming the Limitations of γ- and δ‑C–H Arylation of Amines through Ligand Development von Chen, Yan-Qiao, Wang, Zhen, Wu, Yongwei, Wisniewski, Steven R, Qiao, Jennifer X, Ewing, William R, Eastgate, Martin D, Yu, Jin-Quan

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A tautomeric ligand enables directed C-H hydroxylation with molecular oxygen von Li, Zhen, Wang, Zhen, Chekshin, Nikita, Qian, Shaoqun, Qiao, Jennifer X., Cheng, Peter T., Yeung, Kap-Sun, Ewing, William R., Yu, Jin-Quan

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Anti-Markovnikov Hydroamination of Unactivated Alkenes with Primary Alkyl Amines von Miller, David C, Ganley, Jacob M, Musacchio, Andrew J, Sherwood, Trevor C, Ewing, William R, Knowles, Robert R

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Pd-II-Catalyzed Enantioselective C(sp(3))-H Arylation of Cyclobutyl Ketones Using a Chiral Transient Directing Group von Xiao, Li-Jun, Hong, Kai, Luo, Fan, Hu, Liang, Ewing, William R., Yeung, Kap-Sun, Yu, Jin-Quan

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Selective C−H Halogenation with a Highly Fluorinated Manganese Porphyrin von Li, Gang, Dilger, Andrew K., Cheng, Peter T., Ewing, William R., Groves, John T.

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Potent and selective biphenyl azole inhibitors of adipocyte fatty acid binding protein (aFABP) von Sulsky, Richard, Magnin, David R., Huang, Yanting, Simpkins, Ligaya, Taunk, Prakash, Patel, Manorama, Zhu, Yeheng, Stouch, Terry R., Bassolino-Klimas, Donna, Parker, Rex, Harrity, Thomas, Stoffel, Robert, Taylor, David S., Lavoie, Thomas B., Kish, Kevin, Jacobson, Bruce L., Sheriff, Steven, Adam, Leonard P., Ewing, William R., Robl, Jeffrey A.

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Ni-Catalyzed Carbon–Carbon Bond-Forming Reductive Amination von Heinz, Christoph, Lutz, J. Patrick, Simmons, Eric M, Miller, Michael M, Ewing, William R, Doyle, Abigail G

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Ligand Enabled Pd(II)-Catalyzed γ‑C(sp3)–H Lactamization of Native Amides von Liu, Shuang, Zhuang, Zhe, Qiao, Jennifer X, Yeung, Kap-Sun, Su, Shun, Cherney, Emily C, Ruan, Zheming, Ewing, William R, Poss, Michael A, Yu, Jin-Quan

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Discovery of Milvexian, a High-Affinity, Orally Bioavailable Inhibitor of Factor XIa in Clinical Studies for Antithrombotic Therapy von Dilger, Andrew K, Pabbisetty, Kumar B, Corte, James R, De Lucca, Indawati, Fang, Tianan, Yang, Wu, Pinto, Donald J. P, Wang, Yufeng, Zhu, Yeheng, Mathur, Arvind, Li, Jianqing, Hou, Xiaoping, Smith, Daniel, Sun, Dawn, Zhang, Huiping, Krishnananthan, Subramaniam, Wu, Dauh-Rurng, Myers, Joseph E, Sheriff, Steven, Rossi, Karen A, Chacko, Silvi, Zheng, Joanna J, Galella, Michael A, Ziemba, Theresa, Dierks, Elizabeth A, Bozarth, Jeffrey M, Wu, Yiming, Crain, Earl, Wong, Pancras C, Luettgen, Joseph M, Wexler, Ruth R, Ewing, William R

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