Elucidation of Resistance Mechanisms to Second-Generation ALK Inhibitors Alectinib and Ceritinib in Non–Small Cell Lung Cancer Cells von Dong, Xuyuan, Fernandez-Salas, Ester, Li, Enxiao, Wang, Shaomeng

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Discovery of ARD-69 as a Highly Potent Proteolysis Targeting Chimera (PROTAC) Degrader of Androgen Receptor (AR) for the Treatment of Prostate Cancer von Han, Xin, Wang, Chao, Qin, Chong, Xiang, Weiguo, Fernandez-Salas, Ester, Yang, Chao-Yie, Wang, Mi, Zhao, Lijie, Xu, Tianfeng, Chinnaswamy, Krishnapriya, Delproposto, James, Stuckey, Jeanne, Wang, Shaomeng

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Discovery of QCA570 as an Exceptionally Potent and Efficacious Proteolysis Targeting Chimera (PROTAC) Degrader of the Bromodomain and Extra-Terminal (BET) Proteins Capable of Induc... von Qin, Chong, Hu, Yang, Zhou, Bing, Fernandez-Salas, Ester, Yang, Chao-Yie, Liu, Liu, McEachern, Donna, Przybranowski, Sally, Wang, Mi, Stuckey, Jeanne, Meagher, Jennifer, Bai, Longchuan, Chen, Zhuo, Lin, Mei, Yang, Jiuling, Ziazadeh, Danya N, Xu, Fuming, Hu, Jiantao, Xiang, Weiguo, Huang, Liyue, Li, Siwei, Wen, Bo, Sun, Duxin, Wang, Shaomeng

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Androgen receptor degraders overcome common resistance mechanisms developed during prostate cancer treatment von Kregel, Steven, Wang, Chao, Han, Xin, Xiao, Lanbo, Fernandez-Salas, Ester, Bawa, Pushpinder, McCollum, Brooke L., Wilder-Romans, Kari, Apel, Ingrid J., Cao, Xuhong, Speers, Corey, Wang, Shaomeng, Chinnaiyan, Arul M.

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A potent small-molecule inhibitor of the DCN1-UBC12 interaction that selectively blocks cullin 3 neddylation von Zhou, Haibin, Lu, Jianfeng, Liu, Liu, Bernard, Denzil, Yang, Chao-Yie, Fernandez-Salas, Ester, Chinnaswamy, Krishnapriya, Layton, Stephanie, Stuckey, Jeanne, Yu, Qing, Zhou, Weihua, Pan, Zhenqiang, Sun, Yi, Wang, Shaomeng

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Septin Dynamics Are Essential for Exocytosis von Tokhtaeva, Elmira, Capri, Joe, Marcus, Elizabeth A., Whitelegge, Julian P., Khuzakhmetova, Venera, Bukharaeva, Ellya, Deiss-Yehiely, Nimrod, Dada, Laura A., Sachs, George, Fernandez-Salas, Ester, Vagin, Olga

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Corrigendum to “Androgen receptor degraders overcome common resistance mechanisms developed during prostate cancer treatment” [Neoplasia, Volume 22, Issue 2 (2020) 111–119] von Kregel, Steven, Wang, Chao, Han, Xin, Xiao, Lanbo, Fernandez-Salas, Ester, Bawa, Pushpinder, McCollum, Brooke L., Wilder-Romans, Kari, Apel, Ingrid J., Cao, Xuhong, Speers, Corey, Wang, Shaomeng, Chinnaiyan, Arul M.

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EEDi-5285: An Exceptionally Potent, Efficacious, and Orally Active Small-Molecule Inhibitor of Embryonic Ectoderm Development von Rej, Rohan Kalyan, Wang, Changwei, Lu, Jianfeng, Wang, Mi, Petrunak, Elyse, Zawacki, Kaitlin P, McEachern, Donna, Fernandez-Salas, Ester, Yang, Chao-Yie, Wang, Lu, Li, Ruiting, Chinnaswamy, Krishnapriya, Wen, Bo, Sun, Duxin, Stuckey, Jeanne, Zhou, Yunlong, Chen, Jianyong, Tang, Guozhi, Wang, Shaomeng

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Corrigendum to ‘Androgen receptor degraders overcome common resistance mechanisms developed during prostate cancer treatment’ Neoplasia, Volume 22, Issue 2 (2020) 111–119 von Kregel, Steven, Wang, Chao, Han, Xin, Xiao, Lanbo, Fernandez-Salas, Ester, Bawa, Pushpinder, McCollum, Brooke L., Wilder-Romans, Kari, Apel, Ingrid J., Cao, Xuhong, Speers, Corey, Wang, Shaomeng, Chinnaiyan, Arul M.

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Design of the First‐in‐Class, Highly Potent Irreversible Inhibitor Targeting the Menin‐MLL Protein–Protein Interaction von Xu, Shilin, Aguilar, Angelo, Xu, Tianfeng, Zheng, Ke, Huang, Liyue, Stuckey, Jeanne, Chinnaswamy, Krishnapriya, Bernard, Denzil, Fernández‐Salas, Ester, Liu, Liu, Wang, Mi, McEachern, Donna, Przybranowski, Sally, Foster, Caroline, Wang, Shaomeng

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787 AB598, a CD39 inhibitory antibody, promotes immune-mediated tumor control von Clor, Julie, Jin, Ke, Parashar, Kaustubh, Anderson, Amy E, Kates, Lance, Guan, Yihong, Schwager, Sam, Talukdar, Priyanka, Kushwaha, Ritu, Kline, Janine, Fernandez-Salas, Ester, Bowman, Christine

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880 Inhibition of AXL signaling with AB801 augments anti-tumor immune responses von Leslie, Jhansi, Goshayeshi, Armon, Park, Eugene, Flores, Ruben, Barajas, Gonzalo, Schwager, Samantha C, Stagnaro, Enzo, Kaplan, Angelo, Kline, Janine, Fernandez-Salas, Ester, Paprcka, Susan L

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Botulinum neurotoxin serotype A specific cell-based potency assay to replace the mouse bioassay von Fernández-Salas, Ester, Wang, Joanne, Molina, Yanira, Nelson, Jeremy B, Jacky, Birgitte P S, Aoki, K Roger

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Identification of fibroblast growth factor receptor 3 (FGFR3) as a protein receptor for botulinum neurotoxin serotype A (BoNT/A) von Jacky, Birgitte P S, Garay, Patton E, Dupuy, Jérôme, Nelson, Jeremy B, Cai, Brian, Molina, Yanira, Wang, Joanne, Steward, Lance E, Broide, Ron S, Francis, Joseph, Aoki, K Roger, Stevens, Raymond C, Fernández-Salas, Ester

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The Organellular Chloride Channel Protein CLIC4/mtCLIC Translocates to the Nucleus in Response to Cellular Stress and Accelerates Apoptosis von Suh, Kwang S., Mutoh, Michihiro, Nagashima, Kunio, Fernandez-Salas, Ester, Edwards, Lindsay E., Hayes, Daniel D., Crutchley, John M., Marin, Keith G., Dumont, Rebecca A., Levy, Joshua M., Cheng, Christina, Garfield, Susan, Yuspa, Stuart H.

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A Highly Specific Monoclonal Antibody for Botulinum Neurotoxin Type A-Cleaved SNAP25 von Rhéaume, Catherine, Cai, Brian B, Wang, Joanne, Fernández-Salas, Ester, Aoki, K Roger, Francis, Joseph, Broide, Ron S

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CLIC4 is a tumor suppressor for cutaneous squamous cell cancer von SUH, K. Stephen, MALIK, Mariam, SIMPSON, R. Mark, YUSPA, Stuart H, SHUKLA, Anjali, RYSCAVAGE, Andrew, WRIGHT, Lisa, JIVIDEN, Kasey, CRUTCHLEY, John M, DUMONT, Rebecca A, FERNANDEZ-SALAS, Ester, WEBSTER, Joshua D

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The antiapoptotic decoy receptor TRID/TRAIL-R3 is a p53-regulated DNA damage-inducible gene that is overexpressed in primary tumors of the gastrointestinal tract von SAEED SHEIKH, M, YING HUANG, FERNANDEZ-SALAS, E. A, EL-DEIRY, W. S, FRIESS, H, AMUNDSON, S, JING YIN, MELTZER, S. J, HOLBROOK, N. J, FORNACE, A. J

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Plasma Membrane Localization Signals in the Light Chain of Botulinum Neurotoxin von Fernández-Salas, Ester, Steward, Lance E., Ho, Helen, Garay, Patton E., Sun, Sarah W., Gilmore, Marcella A., Ordas, Joseph V., Wang, Joanne, Francis, Joseph, Aoki, K. Roger, Boyer, Herbert W.

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mtCLIC/CLIC4, an Organellular Chloride Channel Protein, Is Increased by DNA Damage and Participates in the Apoptotic Response to p53 von Fernández-Salas, Ester, Suh, Kwang S., Speransky, Vladislav V., Bowers, Wendy L., Levy, Joshua M., Adams, Tracey, Pathak, Kamal R., Edwards, Lindsay E., Hayes, Daniel D., Cheng, Christina, Steven, Alasdair C., Weinberg, Wendy C., Yuspa, Stuart H.

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